|
558 |
E.Reichert Raguram; J.C. Dahl; K.F. Jensen; S.L. Buchwald |
Kinetic Modeling Enables Understanding of Off-Cycle Processes in Pd-Catalyzed Amination of Five-Membered Heteroaryl Halides |
J. Am. Chem. Soc. |
2024 |
Link |
|
557 |
K. Feng; E.Reichert Raguram; J.R. Howard; E. Peters; C. Liu; M.S. Sigman; S.L. Buchwald |
Development of a Deactivation-Resistant Dialkylbiarylphosphine Ligand for Pd-Catalyzed Arylation of Secondary Amines |
J. Am. Chem. Soc. |
2024 |
Link |
|
556 |
H.J. Ai; S.T. Kim; C. Liu; S.L. Buchwald |
Copper-Catalyzed Amination of Aryl Chlorides under Mild Reaction Conditions |
J. Am. Chem. Soc. |
2024 |
Link |
|
555 |
J. Tao; H.H. Dhanjee; M.W. Gribble; V. Kottisch; J. Rodriguez; J.S. Brown; H. Schmidt; J. Juneja; F. Denhez; P.S. Lee; D. Lipovšek; S. Krystek; Y. Zhang; P. Bousquet; Y. Zhang; B.L. Petelute; S.L. Buchwald |
Site-Specific Antibody Prodrugs via S‑Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues |
J. Am. Chem. Soc. |
2024 |
Link |
|
554 |
M.J. Strauss; K.X. Liu; M.E. Greaves; J.C. Dahl; S.T. Kim; Y.J. Wu; M.A. Schmidt; P.M. Scola; S.L. Buchwald |
Cu-Catalyzed Amination of Base-Sensitive Aryl Bromides and the Chemoselective N- and O-Arylation of Amino Alcohols |
J. Am. Chem. Soc. |
2024 |
Link |
|
553 |
S. Garhwal; Y. Dong; B.Khanh Mai; P. Liu; S.L. Buchwald |
CuH-Catalyzed Regio- and Enantioselective Formal Hydroformylation of Vinyl Arenes |
J. Am. Chem. Soc. |
2024 |
Link |
|
552 |
M.J. Strauss; M.E. Greaves; S.T. Kim; C.N. Teijaro; M.A. Schmidt; P.M. Scola; S.L. Buchwald |
Room-Temperature Copper-Catalyzed Etherification of Aryl Bromides |
Angewandte Chemie |
2024 |
Link |
|
551 |
N.M. Grob; C. Remarcik; S.L. Rössler; J.Y.K. Wong; J.C.K. Wong; J. Tao; C.L. Smith; A. Loas; S.L. Buchwald; D.L. Eaton; M.P. López; B.L. Pentelute |
Electrophile Scanning Reveals Reactivity Hotspots for the Design of Covalent Peptide Binders |
ACS Chem. Biol. |
2024 |
Link |
|
550 |
D.A. Kutateladze; B.Khanh Mai; Y. Dong; Y. Zhang; P. Liu; S.L. Buchwald |
Stereoselective Synthesis of Trisubstituted Alkenes via Copper Hydride-Catalyzed Alkyne Hydroalkylation |
J. Am. Chem. Soc. |
2023 |
Link |
|
549 |
S.T. Kim; M.J. Strauss; A. Cabré; S.L. Buchwald |
Room-Temperature Cu-Catalyzed Amination of Aryl Bromides Enabled by DFT-Guided Ligand Design |
J. Am. Chem. Soc. |
2023 |
Link |
|
548 |
S.L. Rössler; N.M. Grob; S.L. Buchwald; B.L. Pentelute |
Abiotic peptides as carriers of information for the encoding of small-molecule library synthesis |
Science |
2023 |
Link |
|
547 |
Y. Ye; S.T. Kim; R.P. King; M.H. Baik; S.L. Buchwald |
Studying Regioisomer Formation in the Pd-Catalyzed Fluorination of Cyclic Vinyl Triflates: Evidence for in situ Ligand Modification |
Angew. Chem. Int. Ed. |
2023 |
Link |
|
546 |
E.C. Reichert; K. Feng; A. Sather; S.L. Buchwald |
Pd-Catalyzed Amination of Base-Sensitive Five-Membered Heteroaryl Halides with Aliphatic Amines |
J. Am. Chem. Soc. |
2023 |
Link |
|
545 |
J.Levi Knippel; A.Z. Ni; A.W. Schuppe; S.L. Buchwald |
A General Strategy for the Asymmetric Preparation of α-Stereogenic Allyl Silanes, Germanes, and Boronate Esters via Dual Copper Hydride- and Palladium-Catalysis |
Angew. Chem. Int. Ed. |
2022 |
Link |
|
544 |
A.Jose Rojas; J.M. Wolfe; H.H. Dhanjee; I. Buslov; N.L. Truex; R.Y. Liu; W. Massefski; B. Pentelute; S.L. Buchwald |
Palladium−Peptide Oxidative Addition Complexes for Bioconjugation |
Chem. Sci. |
2022 |
Link |
|
543 |
Y. Dong; K. Shin; B.Khanh Mai; P. Liu; S.L. Buchwald |
Copper Hydride-Catalyzed Enantioselective Olefin Hydromethylation |
J. Am. Chem. Soc. |
2022 |
Link |
|
542 |
J. Rodriguez; H.H. Dhanjee; B.L. Pentelute; S.L. Buchwald |
Palladium Mediated Synthesis of Protein–Polyarene Conjugates |
J. Am. Chem. Soc. |
2022 |
Link |
|
541 |
S. Feng; Y. Dong; S.L. Buchwald |
Enantioselective Hydrocarbamoylation of Alkenes |
Angew. Chem. Int. Ed. |
2022 |
Link |
|
540 |
M. Gazvoda; H.H. Dhanjee; J. Rodriguez; J.S. Brown; C.E. Farquhar; N.L. Truex; A. Loas; S.L. Buchwald; B.L. Pentelute |
Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins |
J. Am. Chem. Soc. |
2022 |
Link |
|
539 |
Y. Dong; A.W. Schuppe; B.Khah Mai; P. Liu; S.L. Buchwald |
Confronting the Challenging Asymmetric Carbonyl 1,2-Addition Using Vinyl Heteroarene Pronucleophiles: Ligand-Controlled Regiodivergent Processes through a Dearomatized Allyl–Cu Species |
J. Am. Chem. Soc. |
2022 |
Link |
|
538 |
C.J. Hou; A.W. Schuppe; J.Levi Knippel; A.Z. Ni; S.L. Buchwald |
A Dual CuH- and Pd-Catalyzed Stereoselective Synthesis of Highly Substituted 1,3-Dienes |
Org. Lett. |
2021 |
Link |
|
537 |
R.P. King; S.W. Krska; S.L. Buchwald |
A Neophyl Palladacycle as an Air- and Thermally Stable Precursor to Oxidative Addition Complexes |
Org. Lett. |
2021 |
Link |
|
536 |
R.P. King; S.W. Krska; S.L. Buchwald |
A Ligand Exchange Process for the Diversification of Palladium Oxidative Addition Complexes |
Org. Lett. |
2021 |
Link |
|
535 |
M. Jbara; S. Pomplun; C.K. Schissel; S.Wilson Hawken; A. Boija; I. Klein; J. Rodriguez; S.L. Buchwald; B.L. Pentelute |
Engineering Bioactive Dimeric Transcription Factor Analogs via Palladium Rebound Reagents |
J. Am. Chem. Soc. |
2021 |
Link |
|
534 |
A. Mallek; B.L. Pentelute; S.L. Buchwald |
Selective N-Arylation of p-Aminophenylalanine in Unprotected Peptides with Organometallic Palladium Reagents |
Angew. Chem. Int. Ed. |
2021 |
Link |
|
533 |
A.W. Schuppe; J.Levi Knippel; G.M. Borrajo-Calleja; S.L. Buchwald |
Enantioselective Hydroalkenylation of Olefins with Enol Sulfonates Enabled by Dual Copper Hydride and Palladium Catalysis |
J. Am. Chem. Soc. |
2021 |
Link |
|
532 |
S. Feng; S.L. Buchwald |
CuH-Catalyzed Regio- and Enantioselective Hydrocarboxylation of Allenes; Toward Carboxylic Acids with Acyclic Quarternary Centers |
J. Am. Chem. Soc. |
2021 |
Link |
|
531 |
M. Jbara; J. Rodriguez; H.H. Dhanjee; A. Loas; S.L. Buchwald; B.L. Pentelute |
Oligonucleotide Bioconjugation with Bifunctional Palladium Reagents |
Angew. Chem., Int. Ed. |
2021 |
Link |
|
530 |
J.Levi Knippel; Y. Ye; S.L. Buchwald |
Enantioselective C2-Allylation of Benzimidazoles Using 1,3-Diene Pronucleophiles |
Org. Lett. |
2021 |
Link |
|
529 |
J. Rodriguez; H.H. Dhanjee; S.L. Buchwald |
Amphiphilic Biaryl Monophosphine Ligands by Regioselective Sulfonation |
Org. Lett. |
2021 |
Link |
|
528 |
H.H. Dhanjee; I. Buslov; I.W. Windsor; R.T. Raines; B.L. Pentelute; S.L. Buchwald |
Palladium–Protein Oxidative Addition Complexes by Amine-Selective Acylation |
J. Am. Chem. Soc. |
2020 |
Link |
|
527 |
S.D. McCann; E.C. Reichert; P.Luis Arrechea; S.L. Buchwald |
Development of an Aryl Amination Catalyst with Broad Scope Guided by Consideration of Catalyst Stability |
J. Am. Chem. Soc. |
2020 |
Link |
|
526 |
A. Link; Y. Zhou; S.L. Buchwald |
CuH-Catalyzed Asymmetric Reductive Amidation of α,β-Unsaturated Carboxylic Acids |
Org. Lett. |
2020 |
Link |
|
525 |
S. Guo; J. Zhu; S.L. Buchwald |
Enantioselective Synthesis of β-Amino Acid Derivatives Enabled by Ligand-Controlled Reversal of Hydrocupration Regiochemistry |
Angew. Chem. Int. Ed. |
2020 |
Link |
|
524 |
H. Zhang; P. Ruiz-Castillo; A.W. Schuppe; S.L. Buchwald |
Improved Process for the Palladium-Catalyzed C–O Cross-Coupling of Secondary Alcohols |
Org. Lett. |
2020 |
Link |
|
523 |
Y. Mo; Z. Lu; G. Rughoobur; P. Patil; N. Gershenfeld; A.I. Akinwande; S.L. Buchwald; K.F. Jensen |
Microfluidic electrochemistry for single-electron transfer redox-neutral reactions |
Science |
2020 |
Link |
|
522 |
M.W. Gribble; R.Y. Liu; S.L. Buchwald |
Evidence for Simultaneous Dearomatization of Two Aromatic Rings Under Mild Conditions in Cu(I)-Catalyzed Direct Asymmetric Dearomatization of Pyridine |
J. Am. Chem. Soc. |
2020 |
Link |
|
521 |
Z. Lu; S.L. Buchwald |
The Enantioselective Preparation of Arenes with β-Stereogenic Centers: Confronting the 1,1-Disubstituted Olefin Problem Using CuH/Pd Cooperative Catalysis |
Angew. Chem. Int. Ed. |
2020 |
Link |
|
520 |
Y. Ye; I. Kevlishvili; S. Feng; P. Liu; S.L. Buchwald |
Highly Enantioselective Synthesis of Indazoles with a C3-Quaternary Chiral Center Using CuH Catalysis |
J. Am. Chem. Soc. |
2020 |
Link |
|
519 |
R.Y. Liu; S.L. Buchwald |
CuH-Catalyzed Olefin Functionalization: From Hydroamination to Carbonyl Addition |
Acc. Chem. Res. |
2020 |
Link |
|
518 |
Y. Zhou; L. Zhou; L.T. Jesikiewicz; P. Liu; S.L. Buchwald |
Synthesis of Pyrroles Through the CuH-Catalyzed Coupling of Enynes and Nitriles |
J. Am. Chem. Soc. |
2020 |
Link |
|
517 |
H.H. Dhanjee; A. Saebi; I. Buslov; A.R. Loftis; S.L. Buchwald; B.L. Pentelute |
Protein–Protein Cross-Coupling via Palladium–Protein Oxidative Addition Complexes from Cysteine Residues |
J. Am. Chem. Soc |
2020 |
Link |
|
516 |
R.Y. Liu; J.M. Dennis; S.L. Buchwald |
The Quest for the Ideal Base: Rational Design of a Nickel Precatalyst Enables Mild, Homogeneous C–N Cross-Coupling |
J. Am. Chem. Soc. |
2020 |
Link |
|
515 |
B.Y. Park; M.T. Pirnot; S.L. Buchwald |
Visible Light-Mediated (Hetero)aryl Amination Using Ni(II) Salts and Photoredox Catalysis in Flow: A Synthesis of Tetracaine |
J. Org. Chem. |
2020 |
Link |
|
514 |
S. Feng; H. Hao; P. Liu; S.L. Buchwald |
Diastereo- and Enantioselective CuH-Catalyzed Hydroamination of Strained Trisubstituted Alkenes |
ACS Catal |
2020 |
Link |
|
513 |
A.W. Schuppe; G.M. Borrajo-Calleja; S.L. Buchwald |
Enantioselective Olefin Hydrocyanation Without Cyanide |
J. Am. Chem. Soc. |
2019 |
Link |
|
512 |
S. Ichikawa; S.L. Buchwald |
Asymmetric Synthesis of γ-Amino Alcohols by Copper-Catalyzed Hydroamination |
Organic Letters |
2019 |
Link |
|
511 |
R.P. King; S.L. Buchwald |
Synthesis of (MeCN)2Pd(CF3)OTs, a General Precursor to Palladium(II) Trifluoromethyl Complexes LPd(CF3)X |
Organometallics |
2019 |
Link |
|
510 |
C. Li*; K. Shin*; R. Y.Liu; S.L. Buchwald |
Engaging Aldehydes in CuH-Catalyzed Reductive Coupling Reactions: Stereoselective Allylation with Unactivated 1,3-Diene Pronucleophiles |
Angew. Chem. Int. Ed. |
2019 |
Link |
|
509 |
C.C. Wagen; B.T. Ingoglia; S.L. Buchwald |
Unexpected Formation of Hexasubstituted Arenes through a Twofold Palladium-Mediated Ligand Arylation |
J. Org. Chem. |
2019 |
Link |
|
508 |
L. Bayeh-Romero; S.L. Buchwald |
Copper Hydride-Catalyzed Enantioselective Synthesis of Axially Chiral 1,3-Disubstituted Allenes |
J. Am. Chem. Soc. |
2019 |
Link |
|
507 |
W. Huang; M. Einzinger; A. Maurano; T. Zhu; J. Tiepelt; C. Yu; H.Sik Chae; T. Van Voorhis; M.A. Baldo; S.L. Buchwald |
Large Increase in External Quantum Efficiency by Dihedral Angle Tuning in a Sky-Blue Thermally Activated Delayed Fluorescence Emitter |
Adv. Optical Mater. |
2019 |
Link |
|
506 |
L.M. Baumgartner; J.M. Dennis; N.A. White; S.L. Buchwald; K.F. Jensen |
Use of a Droplet Platform To Optimize Pd-Catalyzed C–N Coupling Reactions Promoted by Organic Bases |
Org. Process Res. Dev. |
2019 |
Link |
|
505 |
J. Xu; R.Y. Liu; C.S. Yeung; S.L. Buchwald |
Monophosphine Ligands Promote Pd-Catalyzed C–S Cross-Coupling Reactions at Room Temperature with Soluble Bases |
ACS Catalysis |
2019 |
Link |
|
504 |
S. Ichikawa; X.J. Dai; S.L. Buchwald |
Regio- and Enantioselective Synthesis of 1,2-Diamine Derivatives by Copper-Catalyzed Hydroamination |
Org. Lett. |
2019 |
Link |
|
503 |
B.T. Ingoglia; C.C. Wagen; S.L. Buchwald |
Biaryl monophosphine ligands in palladium-catalyzed C–N coupling: An updated User's guide |
Tetrahedron |
2019 |
Link |
|
502 |
J.M. Dennis; N.A. White; R.Y. Liu; S.L. Buchwald |
Pd-Catalyzed C–N Coupling Reactions Facilitated by Organic Bases: Mechanistic Investigation Leads to Enhanced Reactivity in the Arylation of Weakly Binding Amines |
ACS Catalysis |
2019 |
Link |
|
501 |
C. Li; R.Y. Liu; L.T. Jesikiewicz; Y. Yang; P. Liu; S.L. Buchwald |
CuH-Catalyzed Enantioselective Ketone Allylation with 1,3-Dienes: Scope, Mechanism, and Applications |
J. Am. Chem. Soc. |
2019 |
Link |
|
500 |
Y. Ye; S.T. Kim; J. Jeong; M.H. Baik; S.L. Buchwald |
CuH-Catalyzed Enantioselective Alkylation of Indole Derivatives with Ligand-Controlled Regiodivergence |
J. Am. Chem. Soc. |
2019 |
Link |
|
499 |
R.Y. Liu; Y. Zhou; Y. Yang; S.L. Buchwald |
Enantioselective Allylation Using Allene, a Petroleum Cracking Byproduct |
J. Am. Chem. Soc. |
2019 |
Link |
|
498 |
X.J. Dai; O.D. Engl; T. León; S.L. Buchwald |
Catalytic Asymmetric Synthesis of α-Arylpyrrolidines and Benzo-fused Nitrogen Heterocycles |
Angew. Chem. Int. Ed. |
2019 |
Link |
|
497 |
M.R. Uehling; R.P. King; S.W. Krska; T. Cernak; S.L. Buchwald |
Pharmaceutical diversification via palladium oxidative addition complexes |
Science |
2019 |
Link |
|
496 |
D.T. Cohen; C. Zhang; C.M. Fadzen; A.J. Mijalis; L. Hie; K.D. Johnson; Z. Shriver; O. Plante; S.J. Miller; S.L. Buchwald; B.L. Pentelute |
A chemoselective strategy for late-stage functionalization of complex small molecules with polypeptides and proteins |
Nat. Chem. |
2019 |
Link |
|
495 |
C. Zhang; E.V. Vinogradova; A.M. Spokoyny; S.L. Buchwald; B.L. Pentelute |
Arylation Chemistry for Bioconjugation |
Angew. Chem. Int. Ed. |
2018 |
Link |
|
494 |
S. Guo; J.C. Yang; S.L. Buchwald |
A Practical Electrophilic Nitrogen Source for the Synthesis of Chiral Primary Amines by Copper-Catalyzed Hydroamination |
J. Am. Chem. Soc. |
2018 |
Link |
|
493 |
A.A. Thomas; K. Speck; I. Kevlishvili; Z. Lu; P. Liu; S.L. Buchwald |
Mechanistically Guided Design of Ligands that Significantly Improve the Efficiency of CuH-Catalyzed Hydroamination Reactions |
J. Am. Chem. Soc. |
2018 |
Link |
|
492 |
K.M. Khan; Y. Zhao; T. Scully; S.L. Buchwald |
Catalytic Arylhydroxylation of Dehydroalanine in Continuous Flow for Simple Access to Unnatural Amino Acids |
Chem. Eur. J. |
2018 |
Link |
|
491 |
S. Ichikawa; S. Zhu; S.L. Buchwald |
A Modified System for the Synthesis of Enantioenriched N‐Arylamines through Copper‐Catalyzed Hydroamination |
Angew. Chem. Int. Ed. |
2018 |
Link |
|
490 |
Y. Zhou; O.D. Engl; J.S. Bandar; E.D. Chant; S.L. Buchwald |
CuH‐Catalyzed Asymmetric Hydroamidation of Vinylarenes |
Angew. Chem. Int. Ed. |
2018 |
Link |
|
489 |
R.Y. Liu; S.L. Buchwald |
Copper-Catalyzed Enantioselective Hydroamination of Alkenes |
Org. Syn. |
2018 |
Link |
|
488 |
M.W. Gribble; S. Guo; S.L. Buchwald |
Asymmetric Cu-Catalyzed 1,4-Dearomatization of Pyridines and Pyridazines without Preactivation of the Heterocycle or Nucleophile |
J. Am. Chem. Soc. |
2018 |
Link |
|
487 |
J.M. Dennis; N.A. White; R.Y. Liu; S.L. Buchwald |
Breaking the Base Barrier: An Electron-Deficient Palladium Catalyst Enables the Use of a Common, Soluble Base in C–N Coupling |
J. Am. Chem. Soc. |
2018 |
Link |
|
486 |
H. Zhang; P. Ruiz-Castillo; S.L. Buchwald |
Palladium-Catalyzed C–O Cross-Coupling of Primary Alcohols |
Org. Lett. |
2018 |
Link |
|
485 |
W. Huang; M. Einzinger; T. Zhu; H.Sik Chae; S. Jeon; S.G. Ihn; M. Sim; S. Kim; M. Su; G. Teverovskiy; T. Wu; T. Van Voorhis; T.M. Swager; M.A. Baldo; S.L. Buchwald |
Molecular Design of Deep Blue Thermally Activated Delayed Fluorescence Materials Employing a Homoconjugative Triptycene Scaffold and Dihedral Angle Tuning |
Chem. Mater. |
2018 |
Link |
|
484 |
K. Kubota; P. Dai; B.L. Pentelute; S.L. Buchwald |
Palladium Oxidative Addition Complexes for Peptide and Protein Crosslinking |
J. Am. Chem. Soc. |
2018 |
Link |
|
483 |
E. Tsai; R.Y. Liu; Y. Yang; S.L. Buchwald |
A Regio- and Enantioselective CuH-Catalyzed Ketone Allylation with Terminal Allenes |
J. Am. Chem. Soc |
2018 |
Link |
|
482 |
R.Y. Liu; M. Bae; S. L. Buchwald |
Mechanistic Insight Facilitates Discovery of a Mild and Efficient Copper-Catalyzed Dehydration of Primary Amides to Nitriles Using Hydrosilanes |
J. Am. Chem. Soc. |
2018 |
Link |
|
481 |
Y. Zhou; J.S. Bandar; R.Y. Liu; S.L. Buchwald |
CuH-Catalyzed Asymmetric Reduction of α,β-Unsaturated Carboxylic Acids to β-Chiral Aldehydes |
J. Am. Chem. Soc |
2018 |
Link |
|
480 |
G. Lu; R.Y. Liu; Y. Yang; C. Fang; D.S. Lambrecht; S.L. Buchwald; P. Liu |
Ligand-Substrate Dispersion Facilitates the Copper-Catalyzed Hydroamination of Unactivated Olefins |
J. Am. Chem. Soc |
2017 |
Link |
|
479 |
A.J. Rojas; B.L. Pentelute; S.L. Buchwald |
Water-Soluble Palladium Reagents for Cysteine S-Arylation under Ambient Aqueous Conditions |
Org. Lett. |
2017 |
Link |
|
478 |
H. Zhang; S.L. Buchwald |
Palladium-Catalyzed Negishi Coupling of α-CF3 Oxiranyl Zincate: Access to Chiral CF3-substituted Benzylic Tertiary Alcohols |
J. Am. Chem. Soc |
2017 |
Link |
|
477 |
E.P.K. Olsen; P.L. Arrechea; S.L. Buchwald |
Mechanistic Insight Leads to a Ligand That Facilitates the Pd-Catalyzed Formation of 2-(Hetero)Arylaminooxazoles and 4-(Hetero)Arylaminothiazoles |
Angew. Chem. Int. Ed. |
2017 |
Link |
|
476 |
H. Wang; J.ChihYeh Yang; S.L. Buchwald |
CuH-Catalyzed Regioselective Intramolecular Hydroamination for the Synthesis of Alkyl-Substituted Chiral Aziridines |
J. Am. Chem. Soc |
2017 |
Link |
|
475 |
Y. Zhou; J.S. Bandar; S.L. Buchwald |
Enantioselective CuH-Catalyzed Hydroacylation Employing Unsaturated Carboxylic Acids as Aldehyde Surrogates |
J. Am. Chem. Soc |
2017 |
Link |
|
474 |
S.D. Friis; M.T. Pirnot; L.N. Dupuis; S.L. Buchwald |
A Dual Palladium and Copper Hydride Catalyzed Approach for Alkyl–Aryl Cross-Coupling of Aryl Halides and Olefins |
Angew. Chem. Int. Ed. |
2017 |
Link |
|
473 |
B.T. Ingoglia; S.L. Buchwald |
Oxidative Addition Complexes as Precatalysts for Cross-Coupling Reactions Requiring Extremely Bulky Biarylphosphine Ligands |
Org. Lett. |
2017 |
Link |
|
472 |
W. Zhao; H.Geun Lee; S.L. Buchwald; J.M. Hooker |
Direct 11CN-Labeling of Unprotected Peptides via Palladium-Mediated Sequential Cross-Coupling Reactions |
J. Am. Chem. Soc |
2017 |
Link |
|
471 |
A.J. Rojas; C. Zhang; E.V. Vinogradova; N. Buchwald; J. Reilly; B.L. Pentelute; S.L. Buchwald |
Divergent unprotected peptide macrocyclisation by palladium-mediated cysteine arylation |
Chem. Sci. |
2017 |
Link |
|
470 |
H.Geun Lee; G. Lautrette; B.L. Pentelute; S.L. Buchwald |
Palladium-Mediated Arylation of Lysine in Unprotected Peptides |
Angew. Chem. Int. Ed. |
2017 |
Link |
|
469 |
M.W. Gribble; M.T. Pirnot; J.S. Bandar; R.Y. Liu; S.L. Buchwald |
Asymmetric Copper Hydride-Catalyzed Markovnikov Hydrosilylation of Vinylarenes and Vinyl Heterocycles |
J. Am. Chem. Soc |
2017 |
Link |
|
468 |
Y. Ye; T. Takada; S.L. Buchwald |
Palladium-Catalyzed Fluorination of Cyclic Vinyl Triflates: Effect of TESCF3 as an Additive |
Angew. Chem. Int. Ed. |
2016 |
Link |
|
467 |
B.J. Reizman; Y.M. Wang; S.L. Buchwald; K.F. Jensen |
Suzuki-Miyaura cross-coupling optimization enabled by automated feedback |
Reaction Chemistry & Engineering |
2016 |
Link |
|
466 |
R.Y. Liu; Y. Yang; S.L. Buchwald |
Regiodivergent and Diastereoselective CuH-Catalyzed Allylation of Imines with Terminal Allenes |
Angew. Chem. Int. Ed. |
2016 |
Link |
|
465 |
P. Ruiz-Castillo; S.L. Buchwald |
Applications of Palladium-Catalyzed C–N Cross-Coupling Reactions |
Chem. Rev. |
2016 |
Link |
|
464 |
A.C. Sather; S.L. Buchwald |
The Evolution of Pd(0)/Pd(II)-Catalyzed Aromatic Fluorination |
Acc. of Chem. Res. |
2016 |
Link |
|
463 |
P.L. Arrechea; S.L. Buchwald |
Biaryl Phosphine Based Pd(II) Amido Complexes: The Effect of Ligand Structure on Reductive Elimination |
J. Am. Chem. Soc. |
2016 |
Link |
|
462 |
N.H. Park; T.J. Senter; S.L. Buchwald |
Rapid Synthesis of Aryl Fluorides in Continuous Flow through the Balz–Schiemann Reaction |
Angew. Chem. Int. Ed. |
2016 |
Link |
|
461 |
B. M. Vincent; J.B. Langlois; R. Srinivas; A. K. Lancaster; R. Scherz-Shouval; L. Whitesell; B. Tidor; S. L. Buchwald; S. Lindquist |
A Fungal-Selective Cytochrome bc1 Inhibitor Impairs Virulence and Prevents the Evolution of Drug Resistance |
Cell Chem. Bio. |
2016 |
Link |
|
460 |
S.M. King; S.L. Buchwald |
Development of a Method for the N-Arylation of Amino Acid Esters with Aryl Triflates |
Org. Lett. |
2016 |
Link |
|
459 |
W. Huang; S.L. Buchwald |
Palladium catalyzed N-Arylation of Iminodibenzyls and Iminostilbenes with Aryl and Hetero-Aryl Halides |
Chem. Eur. J. |
2016 |
Link |
|
458 |
Y. Yang; I.B. Perry; S.L. Buchwald |
Copper-Catalyzed Enantioselective Addition of Styrene-Derived Nucleophiles to Imines Enabled by Ligand-Controlled Chemoselective Hydrocupration |
J. Am. Chem. Soc. |
2016 |
Link |
|
457 |
S. Roesner; S.L. Buchwald |
Continuous-Flow Synthesis of Biaryls by Negishi Cross-Coupling of Fluoro- and Trifluoromethyl-Substituted (Hetero)arenes |
Angew. Chem. Int. Ed. |
2016 |
Link |
|
456 |
S.D. Friis; M.T. Pirnot; S.L. Buchwald |
Asymmetric Hydroarylation of Vinylarenes Using a Synergistic Combination of CuH and Pd Catalysis |
J. Am. Chem. Soc. |
2016 |
Link |
|
455 |
E.B. Corcoran; M.T. Pirnot; S. Lin; S.D. Dreher; D.A. DiRocco; I.W. Davies; S.L. Buchwald; D.W.C. MacMillan |
Aryl amination using ligand-free Ni(II) salts and photoredox catalysis |
Science |
2016 |
Link |
|
454 |
Y. Yang; I.B. Perry; G. Lu; P. Liu; S.L. Buchwald |
Copper-Catalyzed Asymmetric Addition of Olefin-Derived Nucleophiles to Ketones |
Science |
2016 |
Link |
|
453 |
J.S. Bandar; E. Ascic; S.L. Buchwald |
Enantioselective CuH-Catalyzed Reductive Coupling of Aryl Alkenes and Activated Carboxylic Acids |
J. Am. Chem. Soc. |
2016 |
Link |
|
452 |
S.M. Smith; S.L. Buchwald |
Regioselective 2-Amination of Polychloropyrimidines |
Org. Lett. |
2016 |
Link |
|
451 |
Y.M. Wang; S.L. Buchwald |
Enantioselective CuH-Catalyzed Hydroallylation of Vinylarenes |
J. Am. Chem. Soc. |
2016 |
Link |
|
450 |
S.L. Shi; Z.L. Wong; S.L. Buchwald |
Copper-catalysed enantioselective stereodivergent synthesis of amino alcohols |
Nature |
2016 |
Link |
|
449 |
J.C. Yang; D. Niu; B.P. Karsten; F. Lima; S.L. Buchwald |
Use of a “Catalytic” Cosolvent, N,N-Dimethyl Octanamide, Allows the Flow Synthesis of Imatinib with no Solvent Switch |
Angew. Chem. Int. Ed. |
2016 |
Link |
|
448 |
S. Zhu; N. Niljianskul; S.L. Buchwald |
A direct approach to amines with remote stereocentres by enantioselective CuH-catalysed reductive relay hydroamination |
Nat. Chem. |
2016 |
Link |
|
447 |
V.R. Bhonde; B.T. O'Neill; S.L. Buchwald |
An Improved System for the Aqueous Lipshutz–Negishi Cross-Coupling of Alkyl Halides with Aryl Electrophiles |
Angew. Chem. Int. Ed. |
2015 |
Link |
|
446 |
M.T. Pirnot; Y.M. Wang; S.L. Buchwald |
Copper Hydride-Catalyzed Hydroamination of Alkenes and Alkynes |
Angew. Chem. Int. Ed. |
2016 |
Link |
|
445 |
J.S. Bandar; M.T. Pirnot; S.L. Buchwald |
Mechanistic Studies Lead to Dramatically Improved Reaction Conditions for the Cu-Catalyzed Asymmetric Hydroamination of Olefins |
J. Am. Chem. Soc. |
2015 |
Link |
|
444 |
E.V. Vinogradova; C. Zhang; A.M. Spokoyny; B.L. Pentelute; S.L. Buchwald |
Organometallic palladium reagents for cysteine bioconjugation |
Nature |
2015 |
Link |
|
443 |
A.C. Sather; H.Geun Lee; V.Y. De La Rosa; Y. Yang; P. Müller; S.L. Buchwald |
A Fluorinated Ligand Enables Room-Temperature and Regioselective Pd-Catalyzed Fluorination of Aryl Triflates and Bromides |
J. Am. Chem. Soc. |
2015 |
Link |
|
442 |
P.J. Milner; Y. Yang; S.L. Buchwald |
In-Depth Assessment of the Palladium-Catalyzed Fluorination of Five-Membered Heteroaryl Bromides |
Organometallics |
2015 |
Link |
|
441 |
A.C. Sather; H.Geun Lee; J.R. Colombe; A. Zhang; S.L. Buchwald |
Dosage delivery of sensitive reagents enables glove-box-free synthesis |
Nature |
2015 |
Link |
|
440 |
Y.M. Wang; N.C. Bruno; Á.L. Placeres; S. Zhu; S.L. Buchwald |
Enantioselective Synthesis of Carbo- and Heterocycles Through a CuH-Catalyzed Hydroalkylation Approach |
J. Am. Chem. Soc. |
2015 |
Link |
|
439 |
D.T. Cohen; C. Zhang; B.L. Pentelute; S.L. Buchwald |
An Umpolung Approach for the Chemoselective Arylation of Selenocysteine in Unprotected Peptides |
J. Am. Chem. Soc. |
2015 |
Link |
|
438 |
D. Niu; S.L. Buchwald |
Design of Modified Amine Transfer Reagents Allows the Synthesis of α-Chiral Secondary Amines via CuH-Catalyzed Hydroamination |
J. Am. Chem. Soc. |
2015 |
Link |
|
437 |
Y. Yang; S.L. Shi; D. Niu; P. Liu; S.L. Buchwald |
Catalytic Asymmetric Hydroamination of Unactivated Internal Olefins to Aliphatic Amines |
Science |
2015 |
Link |
|
436 |
J.R. Colombe; R. DeBergh; S.L. Buchwald |
Synthesis of Heteroaryl Sulfonamides from Organozinc Reagents and 2,4,6-Trichlorophenyl Chlorosulfate |
Org. Lett. |
2015 |
Link |
|
435 |
R. Zhu; S.L. Buchwald |
Versatile Enantioselective Synthesis of Functionalized Lactones via Copper-Catalyzed Radical Oxyfunctionalization of Alkenes |
J. Am. Chem. Soc. |
2015 |
Link |
|
434 |
N.H. Park; E.V. Vinogradova; D.S. Surry; S.L. Buchwald |
Design of New Ligands for the Palladium-Catalyzed Arylation of α-Branched Secondary Amines |
Angew. Chem. Int. Ed. |
2015 |
Link |
|
433 |
E. Ascic; S.L. Buchwald |
Highly Diastereo- and Enantioselective CuH-Catalyzed Synthesis of 2,3-Disubstituted Indolines |
J. Am. Chem. Soc. |
2015 |
Link |
|
432 |
P. Ruiz-Castillo; D.G. Blackmond; S.L. Buchwald |
Rational Ligand Design for the Arylation of Hindered Primary Amines Guided by Reaction Progress Kinetic Analysis |
J. Am. Chem. Soc. |
2015 |
Link |
|
431 |
H.Geun Lee; P.J. Milner; M.S. Placzek; S.L. Buchwald; J.M. Hooker |
Virtually Instantaneous, Room-Temperature [11C]-Cyanation Using Biaryl Phosphine Pd(0) Complexes |
J. Am. Chem. Soc. |
2015 |
Link |
|
430 |
D.T. Cohen; S.L. Buchwald |
Mild Palladium-Catalyzed Cyanation of (Hetero)aryl Halides and Triflates in Aqueous Media |
Org. Lett. |
2015 |
Link |
|
429 |
S.L. Shi; S.L. Buchwald |
Palladium-Catalyzed Intramolecular C-H Difluoroalkylation: Synthesis of Substituted 3,3-Difluoro-2-oxindoles |
Angew. Chem. Int. Ed. |
2015 |
Link |
|
428 |
S.L. Shi; S.L. Buchwald |
Copper-catalysed Selective Hydroamination Reactions of Alkynes |
Nat. Chem. |
2015 |
Link |
|
427 |
N. Niljianskul; S. Zhu; S.L. Buchwald |
Enantioselective Synthesis of α-Aminosilanes by Copper-Catalyzed Hydroamination of Vinylsilanes |
Angew. Chem. Int. Ed. |
2015 |
Link |
|
426 |
S. Zhu; S.L. Buchwald |
Enantioselective CuH-Catalyzed Anti-Markovnikov Hydroamination of 1,1-Disubstituted Alkenes |
J. Am. Chem. Soc. |
2014 |
Link |
|
425 |
M. Chen; S. Ichikawa; S.L. Buchwald |
Rapid and Efficient Copper-Catalyzed Finkelstein Reaction of (Hetero)Aromatics under Continuous-Flow Conditions |
Angew. Chem. Int. Ed. |
2014 |
Link |
|
424 |
P.J. Milner; T. Kinzel; Y. Zhang; S.L. Buchwald |
Studying Regioisomer Formation in the Pd-Catalyzed Fluorination of Aryl Triflates by Deuterium Labeling |
J. Am. Chem. Soc. |
2014 |
Link |
|
423 |
Y. Yang; K. Niedermann; C. Han; S.L. Buchwald |
Highly Selective Palladium-Catalyzed Cross-Coupling of Secondary Alkylzinc Reagents with Heteroaryl Halides |
Org. Lett. |
2014 |
Link |
|
422 |
S.D. Friis; T. Skrydstrup; S.L. Buchwald |
Mild Pd-Catalyzed Aminocarbonylation of (Hetero)Aryl Bromides with a Palladacycle Precatalyst |
Org. Lett. |
2014 |
Link |
|
421 |
J.B. Ernst; N.E.S. Tay; N.T. Jui; S.L. Buchwald |
Regioselective Synthesis of Benzimidazolones via Cascade C–N Coupling of Monosubstituted Ureas |
Org. Lett. |
2014 |
Link |
|
420 |
H.Geun Lee; P.J. Milner; M.T. Colvin; L. Andreas; S.L. Buchwald |
Structure and reactivity of [(L·Pd)n·(1,5-cyclooctadiene)] (n = 1–2) complexes bearing biaryl phosphine ligands |
Inorganica Chimica Acta |
2014 |
Link |
|
419 |
C.Wai Cheung; S.L. Buchwald |
Palladium-Catalyzed Hydroxylation of Aryl and Heteroaryl Halides Enabled by the Use of a Palladacycle Precatalyst |
J. Org. Chem. |
2014 |
Link |
|
418 |
N.C. Bruno; N. Niljianskul; S.L. Buchwald |
N-Substituted 2-Aminobiphenylpalladium Methanesulfonate Precatalysts and Their Use in C–C and C–N Cross-Couplings |
J. Org. Chem. |
2014 |
Link |
|
417 |
Y. Yang; S.L. Buchwald |
Copper-Catalyzed Regioselective ortho C–H Cyanation of Vinylarenes |
Angew. Chem. Int. Ed. |
2014 |
Link |
|
416 |
Y. Zhu; S.L. Buchwald |
Ligand-Controlled Asymmetric Arylation of Aliphatic α-Amino Anion Equivalents |
J. Am. Chem. Soc. |
2014 |
Link |
|
415 |
H.Geun Lee; P.J. Milner; S.L. Buchwald |
Pd-Catalyzed Nucleophilic Fluorination of Aryl Bromides |
J. Am. Chem. Soc. |
2014 |
Link |
|
414 |
M.J. Su; N. Hoshiya; S.L. Buchwald |
Palladium-Catalyzed Amination of Unprotected Five-Membered Heterocyclic Bromides |
Org. Lett. |
2014 |
Link |
|
413 |
E.V. Vinogradova; P. Müller; S.L. Buchwald |
Structural Reevaluation of the Electrophilic Hypervalent Iodine Reagent for Trifluoromethylthiolation Supported by the Crystalline Sponge Method for X-ray Analysis |
Angew. Chem. Int. Ed. |
2014 |
Link |
|
412 |
N.H. Park; G. Teverovskiy; S.L. Buchwald |
Development of an Air-Stable Nickel Precatalyst for the Amination of Aryl Chlorides, Sulfamates, Mesylates, and Triflates |
Org. Lett. |
2014 |
Link |
|
411 |
C.Yeun Chung; V. Khurana; P.K. Auluck; D.F. Tardiff; J.R. Mazzulli; F. Soldner; V. Baru; Y. Lou; Y. Freyzon; S. Cho; A.E. Mungenast; J. Muffat; M. Mitalipova; M.D. Pluth; N.T. Jui; B. Schüle; S.J. Lippard; L.H. Tsai; D. Krainc; S.L. Buchwald; R. Jaenisch; S. Lindquist |
Identification and Rescue of α-Synuclein Toxicity in Parkinson Patient–Derived Neurons |
Science |
2013 |
Link |
|
410 |
D.F. Tardiff; N.T. Jui; V. Khurana; M.A. Tambe; M.L. Thompson; C.Yeun Chung; H.B. Kamadurai; H.Tae Kim; A.K. Lancaster; K.A. Caldwell; G.A. Caldwell; J.C. Rochet; S.L. Buchwald; S. Lindquist |
Yeast Reveal a “Druggable” Rsp5/Nedd4 Network that Ameliorates α-Synuclein Toxicity in Neurons |
Science |
2013 |
Link |
|
409 |
J.R. Colombe; S. Bernhardt; C. Stathakis; S.L. Buchwald; P. Knochel |
Synthesis of Solid 2-Pyridylzinc Reagents and Their Application in Negishi Reactions |
Org. Lett. |
2013 |
Link |
|
408 |
Y. Yang; T.J.L. Mustard; P.HaYeon Cheong; S.L. Buchwald |
Palladium-Catalyzed Completely Linear-Selective Negishi Cross-Coupling of Allylzinc Halides with Aryl and Vinyl Electrophiles |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
407 |
H.Geun Lee; P.J. Milner; S.L. Buchwald |
An Improved Catalyst System for the Pd-Catalyzed Fluorination of (Hetero)Aryl Triflates |
Org. Lett. |
2013 |
Link |
|
406 |
S. Zhu; N. Niljianskul; S.L. Buchwald |
Enantio- and Regioselective CuH-Catalyzed Hydroamination of Alkenes |
J. Am. Chem. Soc. |
2013 |
Link |
|
405 |
R. Zhu; S.L. Buchwald |
Enantioselective Functionalization of Radical Intermediates in Redox Catalysis: Copper-Catalyzed Asymmetric Oxytrifluoromethylation of Alkenes |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
404 |
M. Chen; S.L. Buchwald |
Rapid and Efficient Trifluoromethylation of Aromatic and Heteroaromatic Compounds Using Potassium Trifluoroacetate Enabled by a Flow System |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
403 |
N.T. Jui; S.L. Buchwald |
Cascade Palladium Catalysis: A Predictable and Selectable Regiocontrolled Synthesis of N-Arylbenzimidazoles |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
402 |
T.D. Senecal; W. Shu; S.L. Buchwald |
A General, Practical Palladium-Catalyzed Cyanation of (Hetero)Aryl Chlorides and Bromides |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
401 |
A. Düfert; K.L. Billingsley; S.L. Buchwald |
Suzuki-Miyaura Cross-Coupling of Unprotected, Nitrogen-Rich Heterocycles: Substrate Scope and Mechanistic Investigation |
J. Am. Chem. Soc. |
2013 |
Link |
|
400 |
C.Wai Cheung; S.L. Buchwald |
Mild and General Palladium-Catalyzed Synthesis of Methyl Aryl Ethers Enabled by the Use of a Palladacycle Precatalyst |
Org. Lett. |
2013 |
Link |
|
399 |
R. DeBergh; N. Niljianskul; S.L. Buchwald |
Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids |
J. Am. Chem. Soc. |
2013 |
Link |
|
398 |
Y. Yang; S.L. Buchwald |
Ligand-Controlled Palladium-Catalyzed Regiodivergent Suzuki–Miyaura Cross-Coupling of Allylboronates and Aryl Halides |
J. Am. Chem. Soc. |
2013 |
Link |
|
397 |
C.Wai Cheung; D.S. Surry; S.L. Buchwald |
Mild and Highly Selective Palladium-Catalyzed Monoarylation of Ammonia Enabled by the Use of Bulky Biarylphosphine Ligands and Palladacycle Precatalysts |
Org. Lett. |
2013 |
Link |
|
396 |
N.C. Bruno; S.L. Buchwald |
Synthesis and Application of Palladium Precatalysts that Accommodate Extremely Bulky Di-tert-butylphosphino Biaryl Ligands |
Org. Lett. |
2013 |
Link |
|
395 |
E.V. Vinogradova; N.H. Park; B.P. Fors; S.L. Buchwald |
Palladium-Catalyzed Synthesis of N-Aryl Carbamates |
Org. Lett. |
2013 |
Link |
|
394 |
M. Chen; S.L. Buchwald |
Continuous-Flow Synthesis of 1-Substituted Benzotriazoles from Chloronitrobenzenes and Amines in a C—N Bond Formation/Hydrogenation/Diazotization/Cyclization Sequence |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
393 |
X. Wang; S.L. Buchwald |
Synthesis of Optically Pure 2-Trifluoromethyl Lactic Acid by Asymmetric Hydroformylation |
J. Org. Chem. |
2013 |
Link |
|
392 |
A. DeAngelis; D.H. Wang; S.L. Buchwald |
Mild and Rapid Pd-Catalyzed Cross-Coupling with Hydrazine in Continuous Flow: Application to the Synthesis of Functionalized Heterocycles |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
391 |
N.C. Bruno; M.T. Tudge; S.L. Buchwald |
Design and preparation of new palladium precatalysts for C-C and C-N cross-coupling reactions |
Chem. Sci. |
2013 |
Link |
|
390 |
A.M. Spokoyny; C.D. Lewis; G. Teverovskiy; S.L. Buchwald |
Extremely Electron-Rich, Boron-Functionalized, Icosahedral Carborane-Based Phosphinoboranes |
Organometallics |
2012 |
Link |
|
389 |
P.J. Milner; T.J. Maimone; M. Su; P. Müller; S.L. Buchwald |
Investigating the Dearomative Rearrangement of Biaryl Phosphine-Ligated Pd(II) Complexes |
J. Am. Chem. Soc. |
2012 |
Link |
|
388 |
Y. Yang; N.J. Oldenhuis; S.L. Buchwald |
Mild and General Conditions for Negishi Cross-Coupling Enabled by the Use of Palladacycle Precatalysts |
Angew. Chem. Int. Ed. |
2013 |
Link |
|
387 |
S. Ueda; S.L. Buchwald |
Catalyst-controlled chemoselective arylation of 2-aminobenzimidazoles |
Angew. Chem., Int. Ed. |
2012 |
Link |
|
386 |
M.A. Oberli; S.L. Buchwald |
A general method for Suzuki-Miyaura coupling reactions using lithium triisopropyl borates |
Org. Lett. |
2012 |
Link |
|
385 |
C.W. Cheung; S.L. Buchwald |
Room temperature copper(II)-catalyzed oxidative cyclization of enamides to 2,5-disubstituted oxazoles via vinylic C-H functionalization |
J. Org. Chem. |
2012 |
Link |
|
384 |
L. Pellegatti; S.L. Buchwald |
Continuous-Flow Preparation and Use of β-Chloro Enals Using the Vilsmeier Reagent |
Org. Process Res. Dev. |
2012 |
Link |
|
383 |
R. Zhu; S.L. Buchwald |
Copper-catalyzed oxytrifluoromethylation of unactivated alkenes |
J. Am. Chem. Soc. |
2012 |
Link |
|
382 |
N. Chernyak; S.L. Buchwald |
Continuous-flow synthesis of monoarylated acetaldehydes using aryldiazonium salts |
J. Am. Chem. Soc. |
2012 |
Link |
|
381 |
M.A. McGowan; C.Z. McAvoy; S.L. Buchwald |
Palladium-Catalyzed N-Monoarylation of Amidines and a One-Pot Synthesis of Quinazoline Derivatives |
Org. Lett. |
2012 |
Link |
|
380 |
E.V. Vinogradova; B.P. Fors; S.L. Buchwald |
Palladium-catalyzed cross-coupling of aryl chlorides and triflates with sodium cyanate: a practical synthesis of unsymmetrical ureas |
J. Am. Chem. Soc. |
2012 |
Link |
|
379 |
N. Hoshiya; S.L. Buchwald |
An Improved Synthesis of BrettPhos- and RockPhos-Type Biarylphosphine Ligands |
Adv. Synth. Catal. |
2012 |
Link |
|
378 |
W. Shu; S.L. Buchwald |
Enantioselective β-arylation of ketones enabled by lithiation/borylation/1,4-addition sequence under flow conditions |
Angew. Chem. Int. Ed. |
2012 |
Link |
|
377 |
M. Su; S.L. Buchwald |
A bulky biaryl phosphine ligand allows for palladium-catalyzed amidation of five-membered heterocycles as electrophiles |
Angew. Chem. Int. Ed. |
2012 |
Link |
|
376 |
A.T. Parsons; T.D. Senecal; S.L. Buchwald |
Iron(II)-Catalyzed Trifluoromethylation of Potassium Vinyltrifluoroborates |
Angew. Chem. Int. Ed. |
2012 |
Link |
|
375 |
M.A. McGowan; J.L. Henderson; S.L. Buchwald |
Palladium-Catalyzed N-Arylation of 2-Aminothiazoles |
Org. Lett. |
2012 |
Link |
|
374 |
S. Ueda; S. Ali; B.P. Fors; S.L. Buchwald |
Me3(OMe)tBuXPhos: a surrogate ligand for Me4tBuXPhos in palladium-catalyzed C-N and C-O bond-forming reactions |
J. Org. Chem. |
2012 |
Link |
|
373 |
L. Salvi; N. Davis; S. Ali; S.L. Buchwald |
A New Biarylphosphine Ligand for the Pd-Catalyzed Synthesis of Diaryl Ethers Under Mild Conditions |
Org. Lett. |
2012 |
Link |
|
372 |
R. Zhu; S.L. Buchwald |
Combined oxypalladation/C-H functionalization: palladium(II)-catalyzed intramolecular oxidative oxyarylation of hydroxyalkenes |
Angew. Chem. Int. Ed. |
2012 |
Link |
|
371 |
S. Ueda; M. Su; S.L. Buchwald |
Completely N1-selective palladium-catalyzed arylation of unsymmetric imidazoles: application to the synthesis of nilotinib |
J. Am. Chem. Soc. |
2012 |
Link |
|
370 |
A.T. Parsons; S.L. Buchwald |
Organic chemistry: A radical approach to diversity |
Nature |
2011 |
Link |
|
369 |
E.J. Cho; S.L. Buchwald |
The palladium-catalyzed trifluoromethylation of vinyl sulfonates |
Org. Lett. |
2011 |
|
|
368 |
X. Wang; S.L. Buchwald |
Rh-catalyzed asymmetric hydroformylation of functionalized 1,1-disubstituted olefins |
J. Am. Chem. Soc. |
2011 |
Link |
|
367 |
T.J. Maimone; P.J. Milner; T. Kinzel; Y. Zhang; M.K. Takase; S.L. Buchwald |
Evidence for<i> in situ</i> Catalyst Modification during the Pd-Catalyzed Conversion of Aryl Triflates to Aryl Fluorides |
J. Am. Chem. Soc. |
2011 |
Link |
|
366 |
J. Pan; X. Wang; Y. Zhang; S.L. Buchwald |
An improved palladium-catalyzed conversion of aryl and vinyl triflates to bromides and chlorides |
Org. Lett. |
2011 |
Link |
|
365 |
W. Shu; L. Pellegatti; M.A. Oberli; S.L. Buchwald |
Continuous-flow synthesis of biaryls enabled by multistep solid-handling in a lithiation/borylation/Suzuki-Miyaura cross-coupling sequence |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
364 |
D. Tsvelikhovsky; S.L. Buchwald |
Concise palladium-catalyzed synthesis of dibenzodiazepines and structural analogues |
J. Am. Chem. Soc. |
2011 |
Link |
|
363 |
W. Shu; S.L. Buchwald |
Use of precatalysts greatly facilitate palladium-catalyzed alkynylations in batch and continuous-flow conditions |
Chem. Sci. |
2011 |
Link |
|
362 |
X. Wu; B.P. Fors; S.L. Buchwald |
A single phosphine ligand allows palladium-catalyzed intermolecular C-O bond formation with secondary and primary alcohols |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
361 |
A.T. Parsons; S.L. Buchwald |
Copper-catalyzed trifluoromethylation of unactivated olefins |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
360 |
T. Noël; T.J. Maimone; S.L. Buchwald |
Accelerating Palladium-Catalyzed C-F Bond Formation: Use of a Microflow Packed-Bed Reactor |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
359 |
S. Ueda; M. Su; S.L. Buchwald |
Highly N2-selective palladium-catalyzed arylation of 1,2,3-triazoles |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
358 |
J. Pan; M. Su; S.L. Buchwald |
Palladium(0)-catalyzed intermolecular amination of unactivated C(sp(3))-H bonds |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
357 |
T. Noel; S.L. Buchwald |
Cross-coupling in flow |
Chem. Soc. Rev. |
2011 |
Link |
|
356 |
P. Li; S.L. Buchwald |
Continuous-flow synthesis of 3,3-disubstituted oxindoles by a palladium-catalyzed α-arylation/alkylation sequence |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
355 |
S. Rousseaux; J. Garcia-Fortanet; M.A.Del Agu Sanchez; S.L. Buchwald |
Palladium(0)-catalyzed arylative dearomatization of phenols |
J. Am. Chem. Soc. |
2011 |
Link |
|
354 |
S. Breitler; N.J. Oldenhuis; B.P. Fors; S.L. Buchwald |
Synthesis of Unsymmetrical Diarylureas via Pd-Catalyzed C–N Cross-Coupling Reactions |
Org. Lett. |
2011 |
Link |
|
353 |
G. Teverovskiy; D.S. Surry; S.L. Buchwald |
Pd-catalyzed synthesis of Ar-SCF3 compounds under mild conditions |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
352 |
T. Noël; S. Kuhn; A.J. Musacchio; K.F. Jensen; S.L. Buchwald |
Suzuki–Miyaura Cross-Coupling Reactions in Flow: Multistep Synthesis Enabled by a Microfluidic Extraction |
Angew. Chem. Int. Ed. |
2011 |
Link |
|
351 |
T.D. Senecal; A.T. Parsons; S.L. Buchwald |
Room temperature aryl trifluoromethylation via copper-mediated oxidative cross-coupling |
J. Org. Chem. |
2011 |
Link |
|
350 |
B.P. Fors; S.L. Buchwald |
Commentary on "A New, Efficient and Recyclable Lanthanum(III) Oxide-Catalyzed C-N Cross-Coupling" by S. Narayana Murthy, B. Madhav, V. Prakash Reddy, and Y. V. D. Nageswar, Adv. Synth. Catal. 2010, 352, 3241-3245 |
Adv. Synth. Catal. |
2010 |
Link |
|
349 |
T. Noël; J.R. Naber; R.L. Hartman; J.P. McMullen; K.F. Jensen; S.L. Buchwald |
Palladium-catalyzed amination reactions in flow: overcoming the challenges of clogging via acoustic irradiation |
Chem. Sci. |
2011 |
Link |
|
348 |
B.P. Fors; S.L. Buchwald |
A Multiligand Based Pd Catalyst for C−N Cross-Coupling Reactions |
J. Am. Chem. Soc. |
2010 |
Link |
|
347 |
J.R. Naber; S.L. Buchwald |
Packed-bed reactors for continuous-flow C-N cross-coupling |
Angew. Chem. Int. Ed. |
2010 |
Link |
|
346 |
J.L. Henderson; S.L. Buchwald |
Efficient Pd-Catalyzed Amination Reactions for Heterocycle Functionalization |
Org. Lett. |
2010 |
Link |
|
345 |
J.L. Henderson; S.M. McDermott; S.L. Buchwald |
Palladium-Catalyzed Amination of Unprotected Halo-7-azaindoles |
Org. Lett. |
2010 |
Link |
|
344 |
X. Shen; A.M. Hyde; S.L. Buchwald |
Palladium-Catalyzed Conversion of Aryl and Vinyl Triflates to Bromides and Chlorides |
J. Am. Chem. Soc. |
2010 |
Link |
|
343 |
D. Tsvelikhovsky; S.L. Buchwald |
Synthesis of Heterocycles via Pd-Ligand Controlled Cyclization of 2-Chloro-N-(2-vinyl)aniline: Preparation of Carbazoles, Indoles, Dibenzazepines and Acridines |
J. Am. Chem. Soc. |
2010 |
Link |
|
342 |
T. Kinzel; Y. Zhang; S.L. Buchwald |
A New Palladium Precatalyst Allows for the Fast Suzuki−Miyaura Coupling Reactions of Unstable Polyfluorophenyl and 2-Heteroaryl Boronic Acids |
J. Am. Chem. Soc. |
2010 |
Link |
|
341 |
R.L. Hartman; J.R. Naber; N. Zaborenko; S.L. Buchwald; K.F. Jensen |
Overcoming the Challenges of Solid Bridging and Constriction during Pd-Catalyzed C-N Bond Formation in Microreactors |
Org. Process Res. Dev. |
2010 |
Link |
|
340 |
D.S. Surry; S.L. Buchwald |
Dialkylbiaryl Phosphines in Pd-Catalyzed Amination: A User's Guide |
Chem. Sci. |
2011 |
Link |
|
339 |
D. Maiti; B.P. Fors; J.L. Henderson; Y. Nakamura; S.L. Buchwald |
Palladium-Catalyzed Coupling of Functionalized Primary and Secondary Amines with Aryl and Heteroaryl Halides: Two Ligands Suffice in Most Cases |
Chem. Sci. |
2011 |
Link |
|
338 |
T.J. Maimone; S.L. Buchwald |
Pd-Catalyzed O-Arylation of Ethyl Acetohydroximate: Synthesis of O-Arylhydroxylamines and Substituted Benzofurans |
J. Am. Chem. Soc. |
2010 |
Link |
|
337 |
X. Shen; G.O. Jones; D.A. Watson; B. Bhayana; S.L. Buchwald |
Enantioselective Synthesis of Axially Chiral Biaryls by the Pd-Catalyzed Suzuki−Miyaura Reaction: Substrate Scope and Quantum Mechanical Investigations |
J. Am. Chem. Soc. |
2010 |
Link |
|
336 |
J.P. McMullen; M.T. Stone; S.L. Buchwald; K.F. Jensen |
An integrated microreactor system for self-optimization of a Heck reaction: from micro- to mesoscale flow systems |
Angew. Chem. Int. Ed. |
2010 |
Link |
|
335 |
E.J. Cho; T.D. Senecal; T. Kinzel; Y. Zhang; D.A. Watson; S.L. Buchwald |
The Palladium-Catalyzed Trifluoromethylation of Aryl Chlorides |
Science |
2010 |
Link |
|
334 |
K. Dooleweerdt; B.P. Fors; S.L. Buchwald |
Pd-Catalyzed Cross-Coupling Reactions of Amides and Aryl Mesylates |
Org. Lett. |
2010 |
Link |
|
333 |
D.S. Surry; S.L. Buchwald |
Diamine Ligands in Copper-Catalyzed Reactions |
Chem. Sci. |
2010 |
Link |
|
332 |
G.O. Jones; P. Liu; K.N. Houk; S.L. Buchwald |
Computational Explorations of Mechanisms and Ligand-Directed Selectivities of Copper-Catalyzed Ullmann-Type Reactions |
J. Am. Chem. Soc. |
2010 |
Link |
|
331 |
D. Maiti; S.L. Buchwald |
Cu-Catalyzed Arylation of Phenols: Synthesis of Sterically Hindered and Heteroaryl Diaryl Ethers |
J. Org. Chem. |
2010 |
Link |
|
330 |
R.L. Hartman; J.R. Naber; S.L. Buchwald; K.F. Jensen |
Multistep microchemical synthesis enabled by microfluidic distillation |
Angew. Chem. Int. Ed. |
2010 |
Link |
|
329 |
X. Shen; S.L. Buchwald |
Rhodium-catalyzed asymmetric intramolecular hydroamination of unactivated alkenes |
Angew. Chem. Int. Ed. |
2010 |
Link |
|
328 |
D. Maiti; S.L. Buchwald |
Orthogonal Cu- and Pd-Based Catalyst Systems for the O- and N-Arylation of Aminophenols |
J. Am. Chem. Soc. |
2009 |
Link |
|
327 |
J.D. Hicks; A.M. Hyde; A.Martinez Cuezva; S.L. Buchwald |
Pd-Catalyzed N-Arylation of Secondary Acyclic Amides: Catalyst Development, Scope, and Computational Study |
J. Am. Chem. Soc. |
2009 |
Link |
|
326 |
J. R. Naber; B.P. Fors; X. Wu; J.T. Gunn; S.L. Buchwald |
Stille Cross-Coupling Reactions of Aryl Mesylates and Tosylates Using a Biarylphosphine Based Catalyst System |
Heterocycles |
2010 |
Link |
|
325 |
B.P. Fors; S.L. Buchwald |
Pd-Catalyzed Conversion of Aryl Chlorides, Triflates, and Nonaflates to Nitroaromatics |
J. Am. Chem. Soc. |
2009 |
Link |
|
324 |
B. Bhayana; B.P. Fors; S.L. Buchwald |
A Versatile Catalyst System for Suzuki−Miyaura Cross-Coupling Reactions of C(sp2)-Tosylates and Mesylates |
Org. Lett. |
2009 |
Link |
|
323 |
D.A. Watson; M. Su; G. Teverovskiy; Y. Zhang; J. Garcia-Fortanet; T. Kinzel; S.L. Buchwald |
Formation of ArF from LPdAr(F): Catalytic Conversion of Aryl Triflates to Aryl Fluorides |
Science |
2009 |
Link |
|
322 |
S. L. Buchwald; C. Bolm |
On the Role of Metal Contaminants in Catalyses with FeCl3 |
Angew. Chem. Int. Ed. |
2009 |
Link |
|
321 |
A.M. Taylor; R.A. Altman; S.L. Buchwald |
Palladium-Catalyzed Enantioselective α-Arylation and α-Vinylation of Oxindoles Facilitated by an Axially Chiral P-Stereogenic Ligand |
J. Am. Chem. Soc. |
2009 |
Link |
|
320 |
A.M. Hyde; S.L. Buchwald |
Synthesis of 5,5-Disubstituted Butenolides Based on a Pd-Catalyzed γ-Arylation Strategy |
Org. Lett. |
2009 |
Link |
|
319 |
C. Han; S.L. Buchwald |
Negishi Coupling of Secondary Alkylzinc Halides with Aryl Bromides and Chlorides |
J. Am. Chem. Soc. |
2009 |
Link |
|
318 |
B.P. Fors; K. Dooleweerdt; Q. Zeng; S.L. Buchwald |
An efficient system for the Pd-catalyzed cross-coupling of amides and aryl chlorides |
Tetrahedron |
2009 |
Link |
|
317 |
J. García-Fortanet; F. Kessler; S.L. Buchwald |
Palladium-Catalyzed Asymmetric Dearomatization of Naphthalene Derivatives |
J. Am. Chem. Soc. |
2009 |
Link |
|
316 |
B.P. Fors; N.R. Davis; S.L. Buchwald |
An Efficient Process for Pd-Catalyzed C−N Cross-Coupling Reactions of Aryl Iodides: Insight Into Controlling Factors |
J. Am. Chem. Soc. |
2009 |
Link |
|
315 |
B.K. Lee; M.R. Biscoe; S.L. Buchwald |
Simple, efficient protocols for the Pd-catalyzed cross-coupling reaction of aryl chlorides and dimethylamine |
Tetrahedron Lett. |
2009 |
Link |
|
314 |
M.R. Biscoe; S.L. Buchwald |
Selective Monoarylation of Acetate Esters and Aryl Methyl Ketones Using Aryl Chlorides |
Org. Lett. |
2009 |
Link |
|
313 |
E.R. Strieter; B. Bhayana; S.L. Buchwald |
Mechanistic Studies on the Copper-Catalyzed N-Arylation of Amides |
J. Am. Chem. Soc. |
2009 |
Link |
|
312 |
R. Martín; S.L. Buchwald |
An Improved Protocol for the Pd-Catalyzed α-Arylation of Aldehydes with Aryl Halides |
Org. Lett. |
2008 |
Link |
|
311 |
B.P. Fors; D.A. Watson; M.R. Biscoe; S.L. Buchwald |
A Highly Active Catalyst for Pd-Catalyzed Amination Reactions: Cross-Coupling Reactions Using Aryl Mesylates and the Highly Selective Monoarylation of Primary Amines Using Aryl Chlorides |
J. Am. Chem. Soc. |
2008 |
Link |
|
310 |
J. García-Fortanet; S. L. Buchwald |
Asymmetric Palladium-Catalyzed Intramolecular α-Arylation of Aldehydes |
Angew. Chem. Int. Ed. |
2008 |
Link |
|
309 |
W.C.Peter Tsang; R.H. Munday; G. Brasche; N. Zheng; S.L. Buchwald |
Palladium-Catalyzed Method for the Synthesis of Carbazoles via Tandem C−H Functionalization and C−N Bond Formation |
J. Org. Chem. |
2008 |
Link |
|
308 |
J.R. Martinelli; D.A. Watson; D.M.M. Freckmann; T.E. Barder; S.L. Buchwald |
Palladium-Catalyzed Carbonylation Reactions of Aryl Bromides at Atmospheric Pressure: A General System Based on Xantphos |
J. Org. Chem. |
2008 |
Link |
|
307 |
B.P. Fors; P. Krattiger; E. Strieter; S.L. Buchwald |
Water-Mediated Catalyst Preactivation: An Efficient Protocol for C−N Cross-Coupling Reactions |
Org. Lett. |
2008 |
Link |
|
306 |
D.A. Watson; X. Fan; S.L. Buchwald |
Carbonylation of Aryl Chlorides with Oxygen Nucleophiles at Atmospheric Pressure. Preparation of Phenyl Esters as Acyl Transfer Agents and the Direct Preparation of Alkyl Esters and Carboxylic Acids |
J. Org. Chem. |
2008 |
Link |
|
305 |
R.A. Altman; A.M. Hyde; X. Huang; S.L. Buchwald |
Orthogonal Pd- and Cu-Based Catalyst Systems for C- and N-Arylation of Oxindoles |
J. Am. Chem. Soc. |
2008 |
Link |
|
304 |
R.A. Altman; K.W. Anderson; S.L. Buchwald |
Pyrrole-2-carboxylic Acid as a Ligand for the Cu-Catalyzed Reactions of Primary Anilines with Aryl Halides |
J. Org. Chem. |
2008 |
Link |
|
303 |
H. Wang; M.L. Duennwald; B.E. Roberts; L.M. Rozeboom; Y.L. Zhang; A.D. Steele; R. Krishnan; L.J. Su; D. Griffin; S. Mukhopadhyay; E.J. Hennessy; P. Weigele; B.J. Blanchard; J. King; A.A. Deniz; S.L. Buchwald; V.M. Ingram; S. Lindquist; J. Shorter |
Direct and selective elimination of specific prions and amyloids by 4,5-dianilinophthalimide and analogs |
Proc Natl Acad Sci U S A |
2008 |
Link |
|
302 |
K.L. Billingsley; S.L. Buchwald |
An Improved System for the Palladium-Catalyzed Borylation of Aryl Halides with Pinacol Borane |
J. Org. Chem. |
2008 |
Link |
|
301 |
A. Minatti; S.L. Buchwald |
Synthesis of Indolines via a Domino Cu-Catalyzed Amidation/Cyclization Reaction |
Org. Lett. |
2008 |
Link |
|
300 |
R. Martin; S.L. Buchwald |
Palladium-Catalyzed Suzuki−Miyaura Cross-Coupling Reactions Employing Dialkylbiaryl Phosphine Ligands |
Acc. Chem. Res. |
2008 |
Link |
|
300 |
R. Martín; S.L. Buchwald |
Palladium-Catalyzed Suzuki−Miyaura Cross-Coupling Reactions Employing Dialkylbiaryl Phosphine Ligands |
Acc. Chem. Res. |
2008 |
Link |
|
299 |
K. L. Billingsley; S. L. Buchwald |
A General and Efficient Method for the Suzuki–Miyaura Coupling of 2-Pyridyl Nucleophiles |
Angew. Chem. Int. Ed. |
2008 |
Link |
|
298 |
G. Brasche; J. García-Fortanet; S.L. Buchwald |
Twofold C−H Functionalization: Palladium-Catalyzed Ortho Arylation of Anilides |
Org. Lett. |
2008 |
Link |
|
297 |
M.R. Biscoe; B.P. Fors; S.L. Buchwald |
A New Class of Easily Activated Palladium Precatalysts for Facile C−N Cross-Coupling Reactions and the Low Temperature Oxidative Addition of Aryl Chlorides |
J. Am. Chem. Soc. |
2008 |
Link |
|
296 |
D. S. Surry; S. L. Buchwald |
Biaryl Phosphane Ligands in Palladium-Catalyzed Amination |
Angew. Chem. Int. Ed. |
2008 |
Link |
|
295 |
J. R. Naber; S. L. Buchwald |
Palladium-Catalyzed Stille Cross-Coupling Reaction of Aryl Chlorides using a Pre-Milled Palladium Acetate and XPhos Catalyst System |
Adv. Synth. Cat. |
2008 |
Link |
|
294 |
R.H. Munday; J.R. Martinelli; S.L. Buchwald |
Palladium-Catalyzed Carbonylation of Aryl Tosylates and Mesylates |
J. Am. Chem. Soc. |
2008 |
Link |
|
293 |
G. Brasche; S. L. Buchwald |
C–H Functionalization/C–N Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines |
Angew. Chem. Int. Ed. |
2008 |
Link |
|
292 |
R. Martín; A. Cuenca; S.L. Buchwald |
Sequential Copper-Catalyzed Vinylation/Cyclization: An Efficient Synthesis of Functionalized Oxazoles |
Org. Lett. |
2007 |
Link |
|
291 |
A. M. Hyde; S. L. Buchwald |
Palladium-Catalyzed γ-Arylation of β,γ-Unsaturated Ketones: Application to a One-Pot Synthesis of Tricyclic Indolines |
Angew. Chem. Int. Ed. |
2008 |
Link |
|
290 |
R.A. Altman; A. Shafir; A. Choi; P.A. Lichtor; S.L. Buchwald |
An Improved Cu-Based Catalyst System for the Reactions of Alcohols with Aryl Halides |
J. Org. Chem. |
2008 |
Link |
|
289 |
N. Zheng; S.L. Buchwald |
Copper-Catalyzed Regiospecific Synthesis of N-Alkylbenzimidazoles |
Org. Lett. |
2007 |
Link |
|
288 |
R.A. Altman; B.P. Fors; S.L. Buchwald |
Pd-catalyzed amination reactions of aryl halides using bulky biarylmonophosphine ligands |
Nature Protocols |
2007 |
Link |
|
287 |
R.A. Altman; S.L. Buchwald |
Pd-catalyzed Suzuki–Miyaura reactions of aryl halides using bulky biarylmonophosphine ligands |
Nature Protocols |
2007 |
Link |
|
286 |
A. Minatti; X. Zheng; S.L. Buchwald |
Synthesis of Chiral 3-Substituted Indanones via an Enantioselective Reductive-Heck Reaction |
J. Org. Chem. |
2007 |
Link |
|
285 |
T. Ikawa; T.E. Barder; M.R. Biscoe; S.L. Buchwald |
Pd-Catalyzed Amidations of Aryl Chlorides Using Monodentate Biaryl Phosphine Ligands: A Kinetic, Computational, and Synthetic Investigation |
J. Am. Chem. Soc. |
2007 |
Link |
|
284 |
R.A. Altman; S.L. Buchwald |
Cu-catalyzed Goldberg and Ullmann reactions of aryl halides using chelating N- and O-based ligands |
Nature Protocols |
2007 |
Link |
|
283 |
J. R. Martinelli; T. P. Clark; D. A. Watson; R. H. Munday; S. L. Buchwald |
Palladium-Catalyzed Aminocarbonylation of Aryl Chlorides at Atmospheric Pressure: The Dual Role of Sodium Phenoxide |
Angew. Chem. Int. Ed. |
2007 |
Link |
|
282 |
R. Martín; S. L. Buchwald |
A General Method for the Direct α-Arylation of Aldehydes with Aryl Bromides and Chlorides |
Angew. Chem. Int. Ed. |
2007 |
Link |
|
281 |
C.P. Jones; K.W. Anderson; S.L. Buchwald |
Sequential Cu-Catalyzed Amidation-Base-Mediated Camps Cyclization: A Two-Step Synthesis of 2-Aryl-4-quinolones fromo-Halophenones |
J. Org. Chem. |
2007 |
Link |
|
280 |
E. McNeill; T.E. Barder; S.L. Buchwald |
Palladium-Catalyzed Silylation of Aryl Chlorides with Hexamethyldisilane |
Org. Lett. |
2007 |
Link |
|
279 |
N. Zheng; K. W. Anderson; X. Huang; H. N. Nguyen; S. L. Buchwald |
A Palladium-Catalyzed Regiospecific Synthesis of N-Aryl Benzimidazoles |
Angew. Chem. Int. Ed. |
2007 |
Link |
|
278 |
T.E. Barder; S.L. Buchwald |
Insights into Amine Binding to Biaryl Phosphine Palladium Oxidative Addition Complexes and Reductive Elimination from Biaryl Phosphine Arylpalladium Amido Complexes via Density Functional Theory |
J. Am. Chem. Soc. |
2007 |
Link |
|
277 |
D.S. Surry; S.L. Buchwald |
Selective Palladium-Catalyzed Arylation of Ammonia: Synthesis of Anilines as Well as Symmetrical and Unsymmetrical Di- and Triarylamines |
J. Am. Chem. Soc. |
2007 |
Link |
|
276 |
R. Martín; C.H. Larsen; A. Cuenca; S.L. Buchwald |
Cu-Catalyzed Tandem C−N Bond Formation for the Synthesis of Pyrroles and Heteroarylpyrroles |
Org. Lett. |
2007 |
Link |
|
275 |
M. R. Biscoe; T. E. Barder; S. L. Buchwald |
Electronic Effects on the Selectivity of Pd-Catalyzed C–N Bond-Forming Reactions Using Biarylphosphine Ligands: The Competitive Roles of Amine Binding and Acidity |
Angew. Chem. Int. Ed. |
2007 |
Link |
|
274 |
R.A. Altman; E.D. Koval; S.L. Buchwald |
Copper-Catalyzed N-Arylation of Imidazoles and Benzimidazoles |
J. Org. Chem. |
2007 |
Link |
|
273 |
K. L. Billingsley; T. E. Barder; S. L. Buchwald |
Palladium-Catalyzed Borylation of Aryl Chlorides: Scope, Applications, and Computational Studies |
Angew. Chem. Int. Ed. |
2007 |
Link |
|
272 |
R. Martín; S.L. Buchwald |
Pd-Catalyzed Kumada−Corriu Cross-Coupling Reactions at Low Temperatures Allow the Use of Knochel-type Grignard Reagents |
J. Am. Chem. Soc. |
2007 |
Link |
|
271 |
A. Shafir; P.A. Lichtor; S.L. Buchwald |
N- versus O-Arylation of Aminoalcohols: Orthogonal Selectivity in Copper-Based Catalysts |
J. Am. Chem. Soc. |
2007 |
Link |
|
270 |
M.Rodríguez Rivero; S.L. Buchwald |
Copper-Catalyzed Vinylation of Hydrazides. A Regioselective Entry to Highly Substituted Pyrroles |
Org. Lett. |
2007 |
Link |
|
269 |
R.A. Altman; S.L. Buchwald |
Cu-Catalyzed N- and O-Arylation of 2-, 3-, and 4-Hydroxypyridines and Hydroxyquinolines |
Org. Lett. |
2007 |
Link |
|
268 |
K. Billingsley; S.L. Buchwald |
Highly Efficient Monophosphine-Based Catalyst for the Palladium-Catalyzed Suzuki−Miyaura Reaction of Heteroaryl Halides and Heteroaryl Boronic Acids and Esters |
J. Am. Chem. Soc. |
2007 |
Link |
|
267 |
T.E. Barder; S.L. Buchwald |
Rationale Behind the Resistance of Dialkylbiaryl Phosphines toward Oxidation by Molecular Oxygen |
J. Am. Chem. Soc. |
2007 |
Link |
|
266 |
T.E. Barder; M.R. Biscoe; S.L. Buchwald |
Structural Insights into Active Catalyst Structures and Oxidative Addition to (Biaryl)phosphine−Palladium Complexes via Density Functional Theory and Experimental Studies |
Organometallics |
2007 |
Link |
|
265 |
T.E. Barder; S.L. Buchwald |
Benchtop Monitoring of Reaction Progress via Visual Recognition with a Handheld UV Lamp: In Situ Monitoring of Boronic Acids in the Suzuki−Miyaura Reaction |
Org. Lett. |
2007 |
Link |
|
264 |
E. R. Murphy; J. R. Martinelli; N. Zaborenko; S. L. Buchwald; K. F. Jensen |
Accelerating Reactions with Microreactors at Elevated Temperatures and Pressures: Profiling Aminocarbonylation Reactions |
Angew. Chem. Int. Ed. |
2007 |
Link |
|
263 |
J.R. Martinelli; D.M.M. Freckmann; S.L. Buchwald |
Convenient Method for the Preparation of Weinreb Amides via Pd-Catalyzed Aminocarbonylation of Aryl Bromides at Atmospheric Pressure |
Org. Lett. |
2006 |
Link |
|
262 |
R. Martín; M.Rodríguez Rivero; S.L. Buchwald |
Domino Cu-Catalyzed C–N Coupling/Hydroamidation: A Highly Efficient Synthesis of Nitrogen Heterocycles |
Angew. Chem. Int. Ed. |
2006 |
Link |
|
261 |
K.W. Anderson; T. Ikawa; R.E. Tundel; S.L. Buchwald |
The Selective Reaction of Aryl Halides with KOH: Synthesis of Phenols, Aromatic Ethers, and Benzofurans |
J. Am. Chem. Soc. |
2006 |
Link |
|
260 |
K.W. Anderson; R.E. Tundel; T. Ikawa; R.A. Altman; S.L. Buchwald |
Monodentate Phosphines Provide Highly Active Catalysts for Pd-Catalyzed C–N Bond-Forming Reactions of Heteroaromatic Halides/Amines and (H)N-Heterocycles |
Angew. Chem. Int. Ed. |
2006 |
Link |
|
259 |
A. Shafir; S.L. Buchwald |
Highly Selective Room-Temperature Copper-Catalyzed C−N Coupling Reactions |
J. Am. Chem. Soc. |
2006 |
Link |
|
258 |
R.A. Altman; S.L. Buchwald |
4,7-Dimethoxy-1,10-phenanthroline: An Excellent Ligand for the Cu-Catalyzed N-Arylation of Imidazoles |
Org. Lett. |
2006 |
Link |
|
257 |
S. Buchwald; C. Larsen; K. Anderson; R. Tundel |
Palladium-Catalyzed Heck Alkynylation of Benzyl Chlorides |
Synlett |
2006 |
Link |
|
256 |
C.H. Burgos; T.E. Barder; X. Huang; S.L. Buchwald |
Significantly Improved Method for the Pd-Catalyzed Coupling of Phenols with Aryl Halides: Understanding Ligand Effects |
Angew. Chem. Int. Ed. |
2006 |
Link |
|
255 |
C. Enguehard-Gueiffier; I. Thery; A. Gueiffier; S.L. Buchwald |
A general and efficient method for the copper-catalyzed cross-coupling of amides and thiophenols with 6-halogenoimidazo[1,2-a]pyridines |
Tetrahedron |
2006 |
Link |
|
254 |
K.L. Billingsley; K.W. Anderson; S.L. Buchwald |
A Highly Active Catalyst for Suzuki–Miyaura Cross-Coupling Reactions of Heteroaryl Compounds |
Angew. Chem. Int. Ed. |
2006 |
Link |
|
253 |
L.M. Klingensmith; E.R. Strieter; T.E. Barder; S.L. Buchwald |
New Insights into Xantphos/Pd-Catalyzed C−N Bond Forming Reactions: A Structural and Kinetic Study |
Organometallics |
2006 |
Link |
|
252 |
R.E. Tundel; K.W. Anderson; S.L. Buchwald |
Expedited Palladium-Catalyzed Amination of Aryl Nonaflates through the Use of Microwave-Irradiation and Soluble Organic Amine Bases |
J. Org. Chem. |
2006 |
Link |
|
251 |
S. Shekhar; P. Ryberg; J.F. Hartwig; J.S. Mathew; D.G. Blackmond; E.R. Strieter; S.L. Buchwald |
Reevaluation of the Mechanism of the Amination of Aryl Halides Catalyzed by BINAP-Ligated Palladium Complexes |
J. Am. Chem. Soc. |
2006 |
Link |
|
250 |
E.R. Strieter; S.L. Buchwald |
Evidence for the Formation and Structure of Palladacycles during Pd-Catalyzed C–N Bond Formation with Catalysts Derived from Bulky Monophosphinobiaryl Ligands |
Angew. Chem. Int. Ed. |
2006 |
Link |
|
249 |
W.C.Peter Tsang; N. Zheng; S.L. Buchwald |
Combined C−H Functionalization/C−N Bond Formation Route to Carbazoles |
J. Am. Chem. Soc. |
2005 |
Link |
|
248 |
S. L. Buchwald; C. Mauger; G. Mignani; U. Scholz |
Industrial-Scale Palladium-Catalyzed Coupling of Aryl Halides and Amines –A Personal Account |
Advanced Synthesis & Catalysis |
2006 |
Link |
|
247 |
M.D. Charles; P. Schultz; S.L. Buchwald |
Efficient Pd-Catalyzed Amination of Heteroaryl Halides |
Org. Lett. |
2005 |
Link |
|
246 |
E.J. Hennessy; S.L. Buchwald |
Synthesis of 4,5-Dianilinophthalimide and Related Analogues for Potential Treatment of Alzheimer's Disease via Palladium-Catalyzed Amination |
J. Org. Chem. |
2005 |
Link |
|
245 |
K.W. Anderson; S.L. Buchwald |
General Catalysts for the Suzuki-Miyaura and Sonogashira Coupling Reactions of Aryl Chlorides and for the Coupling of Challenging Substrate Combinations in Water |
Angew. Chem. Int. Ed. |
2005 |
Link |
|
244 |
M.P. Rainka; J.E. Milne; S.L. Buchwald |
Dynamic Kinetic Resolution of α,β-Unsaturated Lactones through Asymmetric Copper-Catalyzed Conjugate Reduction: Application to the Total Synthesis of Eupomatilone-3 |
Angew. Chem. Int. Ed. |
2005 |
Link |
|
243 |
A.V. Vorogushin; X. Huang; S.L. Buchwald |
Use of Tunable Ligands Allows for Intermolecular Pd-Catalyzed C−O Bond Formation |
J. Am. Chem. Soc. |
2005 |
Link |
|
242 |
E.R. Strieter; D.G. Blackmond; S.L. Buchwald |
The Role of Chelating Diamine Ligands in the Goldberg Reaction: A Kinetic Study on the Copper-Catalyzed Amidation of Aryl Iodides |
J. Am. Chem. Soc. |
2005 |
Link |
|
241 |
T.E. Barder; S.D. Walker; J.R. Martinelli; S.L. Buchwald |
Catalysts for Suzuki−Miyaura Coupling Processes: Scope and Studies of the Effect of Ligand Structure |
J. Am. Chem. Soc. |
2005 |
Link |
|
240 |
J. Chae; J. Yun; S.L. Buchwald |
One-Pot Sequential Cu-Catalyzed Reduction and Pd-Catalyzed Arylation of Silyl Enol Ethers |
Org. Lett. |
2004 |
Link |
|
239 |
J.E. Milne; S.L. Buchwald |
An extremely active catalyst for the Negishi cross-coupling reaction |
J. Am. Chem. Soc. |
2004 |
Link |
|
238 |
T.E. Barder; S.L. Buchwald |
Efficient Catalyst for the Suzuki−Miyaura Coupling of Potassium Aryl Trifluoroborates with Aryl Chlorides |
Org. Lett. |
2004 |
Link |
|
237 |
J.C. Antilla; J.M. Baskin; T.E. Barder; S.L. Buchwald |
Copper−Diamine-Catalyzed N-Arylation of Pyrroles, Pyrazoles, Indazoles, Imidazoles, and Triazoles |
J. Org. Chem. |
2004 |
Link |
|
236 |
M. Murata; S.L. Buchwald |
A general and efficient method for the palladium-catalyzed cross-coupling of thiols and secondary phosphines |
Tetrahedron |
2004 |
Link |
|
235 |
M.P. Rainka; Y. Aye; S.L. Buchwald |
Copper-catalyzed asymmetric conjugate reduction as a route to novel β-azaheterocyclic acid derivatives |
Proceedings of the National Academy of Sciences of the United States of America |
2004 |
Link |
|
234 |
J. Chae; S.L. Buchwald |
Palladium-Catalyzed Regioselective Hydrodebromination of Dibromoindoles: Application to the Enantioselective Synthesis of Indolodioxane U86192A |
J. Org. Chem. |
2004 |
Link |
|
233 |
A. Klapars; S. Parris; K.W. Anderson; S.L. Buchwald |
Synthesis of Medium Ring Nitrogen Heterocycles via a Tandem Copper-Catalyzed C−N Bond Formation−Ring-Expansion Process |
J. Am. Chem. Soc. |
2004 |
Link |
|
232 |
S.D. Walker; T.E. Barder; J.R. Martinelli; S.L. Buchwald |
A Rationally Designed Universal Catalyst for Suzuki–Miyaura Coupling Processes |
Angew. Chem. Int. Ed. |
2004 |
Link |
|
231 |
D. Gelman; S.L. Buchwald |
Efficient Palladium-Catalyzed Coupling of Aryl Chlorides and Tosylates with Terminal Alkynes: Use of a Copper Cocatalyst Inhibits the Reaction |
Angew. Chem. Int. Ed. |
2003 |
Link |
|
230 |
E.R. Strieter; D.G. Blackmond; S.L. Buchwald |
Insights into the Origin of High Activity and Stability of Catalysts Derived from Bulky, Electron-Rich Monophosphinobiaryl Ligands in the Pd-Catalyzed C−N Bond Formation |
J. Am. Chem. Soc. |
2003 |
Link |
|
229 |
K.W. Anderson; M. Mendez-Perez; J. Priego; S.L. Buchwald |
Palladium-Catalyzed Amination of Aryl Nonaflates |
J. Org. Chem. |
2003 |
Link |
|
228 |
L. Jiang; G.E. Job; A. Klapars; S.L. Buchwald |
Copper-Catalyzed Coupling of Amides and Carbamates with Vinyl Halides |
Org. Lett. |
2003 |
Link |
|
227 |
H.Nho Nguyen; X. Huang; S.L. Buchwald |
The First General Palladium Catalyst for the Suzuki−Miyaura and Carbonyl Enolate Coupling of Aryl Arenesulfonates |
J. Am. Chem. Soc. |
2003 |
Link |
|
226 |
E.J. Hennessy; S.L. Buchwald |
Synthesis of Substituted Oxindoles from α-Chloroacetanilides via Palladium-Catalyzed C−H Functionalization |
J. Am. Chem. Soc. |
2003 |
Link |
|
225 |
C. Enguehard; H. Allouchi; A. Gueiffier; S.L. Buchwald |
Ipso- or Cine-Substitutions of 6-Haloimidazo[1,2-a]pyridine Derivatives with Different Azoles Depending on the Reaction Conditions |
J. Org. Chem. |
2003 |
Link |
|
224 |
G. Hughes; M. Kimura; S.L. Buchwald |
Catalytic Enantioselective Conjugate Reduction of Lactones and Lactams |
J. Am. Chem. Soc. |
2003 |
Link |
|
223 |
V. Jurkauskas; J.P. Sadighi; S.L. Buchwald |
Conjugate Reduction of α,β-Unsaturated Carbonyl Compounds Catalyzed by a Copper Carbene Complex |
Org. Lett. |
2003 |
Link |
|
222 |
D. Zim; S.L. Buchwald |
An Air and Thermally Stable One- Component Catalyst for the Amination of Aryl Chlorides |
Org. Lett. |
2003 |
Link |
|
221 |
D. Gelman; L. Jiang; S.L. Buchwald |
Copper-Catalyzed C−P Bond Construction via Direct Coupling of Secondary Phosphines and Phosphites with Aryl and Vinyl Halides |
Org. Lett. |
2003 |
Link |
|
220 |
C. Enguehard; H. Allouchi; A. Gueiffier; S.L. Buchwald |
Easy Access to Novel Substituted 6-Aminoimidazo[1,2-a]pyridines Using Palladium- and Copper-Catalyzed Aminations |
J. Org. Chem. |
2003 |
Link |
|
219 |
X. Huang; K.W. Anderson; D. Zim; L. Jiang; A. Klapars; S.L. Buchwald |
Expanding Pd-Catalyzed C−N Bond-Forming Processes: The First Amidation of Aryl Sulfonates, Aqueous Amination, and Complementarity with Cu-Catalyzed Reactions |
J. Am. Chem. Soc. |
2003 |
Link |
|
218 |
G. Nordmann; S.L. Buchwald |
A Domino Copper-Catalyzed C−O Coupling−Claisen Rearrangement Process |
J. Am. Chem. Soc. |
2003 |
Link |
|
217 |
J. Zanon; A. Klapars; S.L. Buchwald |
Copper-Catalyzed Domino Halide Exchange-Cyanation of Aryl Bromides |
J. Am. Chem. Soc. |
2003 |
Link |
|
216 |
F.Yee Kwong; S.L. Buchwald |
Mild and Efficient Copper-Catalyzed Amination of Aryl Bromides with Primary Alkylamines |
Org. Lett. |
2003 |
Link |
|
215 |
J.L. Rutherford; M.P. Rainka; S.L. Buchwald |
An Annulative Approach to Highly Substituted Indoles: Unusual Effect of Phenolic Additives on the Success of the Arylation of Ketone Enolates |
J. Am. Chem. Soc. |
2002 |
Link |
|
214 |
A. Klapars; S.L. Buchwald |
Copper-Catalyzed Halogen Exchange in Aryl Halides: An Aromatic Finkelstein Reaction |
J. Am. Chem. Soc. |
2002 |
Link |
|
213 |
G.E. Job; S.L. Buchwald |
Copper-Catalyzed Arylation of β-Amino Alcohols |
Org. Lett. |
2002 |
Link |
|
212 |
F.Yee Kwong; S.L. Buchwald |
A General, Efficient, and Inexpensive Catalyst System for the Coupling of Aryl Iodides and Thiols |
Org. Lett. |
2002 |
Link |
|
211 |
U.K. Singh; E.R. Strieter; D.G. Blackmond; S.L. Buchwald |
Mechanistic Insights into the Pd(BINAP)-Catalyzed Amination of Aryl Bromides: Kinetic Studies under Synthetically Relevant Conditions |
J. Am. Chem. Soc. |
2002 |
Link |
|
210 |
J.C. Antilla; A. Klapars; S.L. Buchwald |
The Copper-Catalyzed N-Arylation of Indoles |
J. Am. Chem. Soc. |
2002 |
Link |
|
209 |
D.J. Spielvogel; W.M. Davis; S.L. Buchwald |
Preparation, Crystal Structure Analysis, and Catalytic Application of [(S)-BINAP]Ni(COD) and [(S)-BINAP]NiBr2 |
Organometallics |
2002 |
Link |
|
208 |
M.C. Harris; X. Huang; S.L. Buchwald |
Improved Functional Group Compatibility in the Palladium-Catalyzed Synthesis of Aryl Amines |
Org. Lett. |
2002 |
Link |
|
207 |
A. Klapars; X. Huang; S.L. Buchwald |
A General and Efficient Copper Catalyst for the Amidation of Aryl Halides |
J. Am. Chem. Soc. |
2002 |
Link |
|
206 |
J. Yin; S.L. Buchwald |
Pd-Catalyzed Intermolecular Amidation of Aryl Halides: The Discovery that Xantphos Can Be Trans-Chelating in a Palladium Complex |
J. Am. Chem. Soc. |
2002 |
Link |
|
205 |
S.J. Sturla; S.L. Buchwald |
Cobalt−Phosphite-Catalyzed Asymmetric Pauson−Khand Reaction |
J. Org. Chem. |
2002 |
Link |
|
204 |
D.J. Spielvogel; S.L. Buchwald |
Nickel-BINAP Catalyzed Enantioselective α-Arylation of α-Substituted γ-Butyrolactones |
J. Am. Chem. Soc. |
2002 |
Link |
|
203 |
V. Jurkauskas; S.L. Buchwald |
Dynamic Kinetic Resolution via Asymmetric Conjugate Reduction: Enantio- and Diastereoselective Synthesis of 2,4-Dialkyl Cyclopentanones |
J. Am. Chem. Soc. |
2002 |
Link |
|
202 |
T. Hamada; S.L. Buchwald |
P-Chirogenic Binaphthyl-Substituted Monophosphines: Synthesis and Use in Enolate Vinylation/Arylation Reactions |
Org. Lett. |
2002 |
Link |
|
201 |
M. Wolter; G. Nordmann; G.E. Job; S.L. Buchwald |
Copper-Catalyzed Coupling of Aryl Iodides with Aliphatic Alcohols |
Org. Lett. |
2002 |
Link |
|
200 |
F.Yee Kwong; A. Klapars; S.L. Buchwald |
Copper-Catalyzed Coupling of Alkylamines and Aryl Iodides: An Efficient System Even in an Air Atmosphere |
Org. Lett. |
2002 |
Link |
|
199 |
E.J. Hennessy; S.L. Buchwald |
A General and Mild Copper-Catalyzed Arylation of Diethyl Malonate |
Org. Lett. |
2002 |
Link |
|
198 |
J. Yin; M.P. Rainka; X.X. Zhang; S.L. Buchwald |
A highly active Suzuki catalyst for the synthesis of sterically hindered biaryls: novel ligand coordination |
J. Am. Chem. Soc. |
2002 |
Link |
|
197 |
S.J. Sturla; S.L. Buchwald |
Monocyclopentadienyltitanium Aryloxide Complexes: Preparation, Characterization, and Application in Cyclization Reactions |
Organometallics |
2002 |
Link |
|
196 |
O. Gaertzen; S.L. Buchwald |
Palladium-Catalyzed Intramolecular α-Arylation of α-Amino Acid Esters |
J. Org. Chem. |
2002 |
Link |
|
195 |
T. Hamada; A. Chieffi; J.Å. hman; S.L. Buchwald |
An Improved Catalyst for the Asymmetric Arylation of Ketone Enolates |
J. Am. Chem. Soc. |
2002 |
Link |
|
194 |
S.I. Kuwabe; K.E. Torraca; S.L. Buchwald |
Palladium-Catalyzed Intramolecular C−O Bond Formation |
J. Am. Chem. Soc. |
2001 |
Link |
|
193 |
E.M. Vogl; S.L. Buchwald |
Palladium-Catalyzed Monoarylation of Nitroalkanes |
J. Org. Chem. |
2002 |
Link |
|
192 |
M. Wolter; A. Klapars; S.L. Buchwald |
Synthesis of N-Aryl Hydrazides by Copper-Catalyzed Coupling of Hydrazides with Aryl Iodides |
Org. Lett. |
2001 |
Link |
|
191 |
X. Huang; S.L. Buchwald |
New Ammonia Equivalents for the Pd-Catalyzed Amination of Aryl Halides |
Org. Lett. |
2001 |
Link |
|
190 |
K.E. Torraca; X. Huang; C.A. Parrish; S.L. Buchwald |
An Efficient Intermolecular Palladium-Catalyzed Synthesis of Aryl Ethers |
J. Am. Chem. Soc. |
2001 |
Link |
|
189 |
S. Kaye; J.M. Fox; F.A. Hicks; S.L. Buchwald |
The Use of Catalytic Amounts of CuCl and Other Improvements in the Benzyne Route to Biphenyl-Based Phosphine Ligands |
Advanced Synthesis & Catalysis |
2001 |
Link |
|
188 |
J.P. Wolfe; S.L. Buchwald |
Palladium-Catalyzed Amination of Aryl Halides and Aryl Triflates: N-Hexyl-2-methyl-4-methoxy Aniline and N-Methyl-N-(4-chlorophenyl) Aniline |
Org. Syn. |
2000 |
Link |
|
187 |
A. Klapars; J.C. Antilla; X. Huang; S.L. Buchwald |
A General and Efficient Copper Catalyst for the Amidation of Aryl Halides and the N-Arylation of Nitrogen Heterocycles |
J. Am. Chem. Soc. |
2001 |
Link |
|
186 |
W.A. Moradi; S.L. Buchwald |
Palladium-Catalyzed α-Arylation of Esters |
J. Am. Chem. Soc. |
2001 |
Link |
|
185 |
X.X. Zhang; M.C. Harris; J.P. Sadighi; S.L. Buchwald |
The use of palladium chloride as a precatalyst for the amination of aryl bromides |
Can. J. Chem. |
2001 |
Link |
|
184 |
J.C. Antilla; S.L. Buchwald |
Copper-Catalyzed Coupling of Arylboronic Acids and Amines |
Org. Lett. |
2001 |
Link |
|
183 |
A. Chieffi; K. Kamikawa; J.Å. hman; J.M. Fox; S.L. Buchwald |
Catalytic Asymmetric Vinylation of Ketone Enolates |
Org. Lett. |
2001 |
Link |
|
182 |
C.A. Parrish; S.L. Buchwald |
Use of Polymer-Supported Dialkylphosphinobiphenyl Ligands for Palladium-Catalyzed Amination and Suzuki Reactions |
J. Org. Chem. |
2001 |
Link |
|
181 |
J. Yun; S.L. Buchwald |
One-Pot Synthesis of Enantiomerically Enriched 2,3-Disubstituted Cyclopentanones via Copper-Catalyzed 1,4-Reduction and Alkylation |
Org. Lett. |
2001 |
Link |
|
180 |
C.A. Parrish; S.L. Buchwald |
Palladium-Catalyzed Formation of Aryl tert-Butyl Ethers from Unactivated Aryl Halides |
J. Org. Chem. |
2001 |
Link |
|
179 |
M.H. Ali; S.L. Buchwald |
An Improved Method for the Palladium-Catalyzed Amination of Aryl Iodides |
J. Org. Chem. |
2001 |
Link |
|
178 |
K.E. Torraca; S.I. Kuwabe; S.L. Buchwald |
A High-Yield, General Method for the Catalytic Formation of Oxygen Heterocycles |
J. Am. Chem. Soc. |
2000 |
Link |
|
177 |
J. Yin; S.L. Buchwald |
A Catalytic Asymmetric Suzuki Coupling for the Synthesis of Axially Chiral Biaryl Compounds |
J. Am. Chem. Soc. |
2000 |
Link |
|
176 |
X.X. Zhang; S.L. Buchwald |
Efficient Synthesis of N-Aryl-Aza-Crown Ethers via Palladium-Catalyzed Amination |
J. Org. Chem. |
2000 |
Link |
|
175 |
H. Tomori; J.M. Fox; S.L. Buchwald |
An Improved Synthesis of Functionalized Biphenyl-Based Phosphine Ligands |
J. Org. Chem. |
2000 |
Link |
|
174 |
X.X. Zhang; J.P. Sadighi; T.W. Mackewitz; S.L. Buchwald |
Efficient Synthesis of Well-Defined, High Molecular Weight, and Processible Polyanilines under Mild Conditions via Palladium-Catalyzed Amination |
J. Am. Chem. Soc. |
2000 |
Link |
|
173 |
Y. Moritani; D.H. Appella; V. Jurkauskas; S.L. Buchwald |
Synthesis of β-Alkyl Cyclopentanones in High Enantiomeric Excess via Copper-Catalyzed Asymmetric Conjugate Reduction |
J. Am. Chem. Soc. |
2000 |
Link |
|
172 |
O.J. Plante; S.L. Buchwald; P.H. Seeberger |
Halobenzyl Ethers as Protecting Groups for Organic Synthesis |
J. Am. Chem. Soc. |
2000 |
Link |
|
171 |
M.C. Harris; S.L. Buchwald |
One-Pot Synthesis of Unsymmetrical Triarylamines from Aniline Precursors |
J. Org. Chem. |
2000 |
Link |
|
170 |
T. Hundertmark; A.F. Littke; S.L. Buchwald; G.C. Fu |
Pd(PhCN)2Cl2/P(t-Bu)3: A Versatile Catalyst for Sonogashira Reactions of Aryl Bromides at Room Temperature |
Org. Lett. |
2000 |
Link |
|
169 |
D.W. Old; M.C. Harris; S.L. Buchwald |
Efficient Palladium-CatalyzedN-Arylation of Indoles |
Org. Lett. |
2000 |
Link |
|
168 |
J. Yin; S.L. Buchwald |
Palladium-Catalyzed Intermolecular Coupling of Aryl Halides and Amides |
Org. Lett. |
2000 |
Link |
|
167 |
M.C. Hansen; S.L. Buchwald |
A method for the asymmetric hydrosilylation of N-aryl imines |
Org. Lett. |
2000 |
Link |
|
166 |
J. Yun; S.L. Buchwald |
Kinetic resolution and isomerization of 2,5-disubstituted pyrrolines |
Chirality |
2000 |
Link |
|
165 |
J.M. Fox; X. Huang; A. Chieffi; S.L. Buchwald |
Highly Active and Selective Catalysts for the Formation of α-Aryl Ketones |
J. Am. Chem. Soc. |
2000 |
Link |
|
164 |
J. Yun; S.L. Buchwald |
Efficient Kinetic Resolution in the Asymmetric Hydrosilylation of Imines of 3-Substituted Indanones and 4-Substituted Tetralones |
J. Org. Chem. |
2000 |
Link |
|
163 |
J.P. Wolfe; S.L. Buchwald |
Scope and Limitations of the Pd/BINAP-Catalyzed Amination of Aryl Bromides |
J. Org. Chem. |
2000 |
Link |
|
162 |
J.P. Wolfe; H. Tomori; J.P. Sadighi; J. Yin; S.L. Buchwald |
Simple, Efficient Catalyst System for the Palladium-Catalyzed Amination of Aryl Chlorides, Bromides, and Triflates |
J. Org. Chem. |
2000 |
Link |
|
161 |
D.H. Appella; Y. Moritani; R. Shintani; E.M. Ferreira; S.L. Buchwald |
Asymmetric Conjugate Reduction of α,β-Unsaturated Esters Using a Chiral Phosphine−Copper Catalyst |
J. Am. Chem. Soc. |
1999 |
Link |
|
160 |
S. Wagaw; B.H. Yang; S.L. Buchwald |
A Palladium-Catalyzed Method for the Preparation of Indoles via the Fischer Indole Synthesis |
J. Am. Chem. Soc. |
1999 |
Link |
|
159 |
M. Frid; D. Pérez; A.J. Peat; S.L. Buchwald |
A Combined Zirconocene Benzyne−Palladium Cross-Coupling Route to Substituted Biphenyls and Terphenyls |
J. Am. Chem. Soc. |
1999 |
Link |
|
158 |
J.P. Wolfe; R.A. Singer; B.H. Yang; S.L. Buchwald |
Highly Active Palladium Catalysts for Suzuki Coupling Reactions |
J. Am. Chem. Soc. |
1999 |
Link |
|
157 |
C. Gurtler; S.L. Buchwald |
A phosphane-free catalyst system for the Heck arylation of disubstituted alkenes: Application to the synthesis of trisubstituted olefins |
Chem. Eur. J. |
1999 |
Link |
|
156 |
M.C. Harris; O. Geis; S.L. Buchwald |
Sequential N-Arylation of Primary Amines as a Route To Alkyldiarylamines |
J. Org. Chem. |
1999 |
Link |
|
155 |
F.A. Hicks; S.L. Buchwald |
An Intramolecular Titanium-Catalyzed Asymmetric Pauson−Khand Type Reaction |
J. Am. Chem. Soc. |
1999 |
Link |
|
154 |
J.P. Wolfe; S.L. Buchwald |
A Highly Active Catalyst for the Room-Temperature Amination and Suzuki Coupling of Aryl Chlorides |
Angew. Chem. Int. Ed. |
1999 |
Link |
|
153 |
S.J. Sturla; S.L. Buchwald |
Catalytic Asymmetric Cyclocarbonylation of Nitrogen-Containing Enynes |
J. Org. Chem. |
1999 |
Link |
|
152 |
J. Yun; S.L. Buchwald |
Titanocene-catalyzed asymmetric ketone hydrosilylation: The effect of catalyst activation protocol and additives on the reaction rate and enantioselectivity |
J. Am. Chem. Soc. |
1999 |
Link |
|
151 |
B.H. Yang; S.L. Buchwald |
The development of efficient protocols for the palladium-catalyzed cyclization reactions of secondary amides and carbamates |
Org. Lett. |
1999 |
Link |
|
150 |
F.A. Hicks; N.M. Kablaoui; S.L. Buchwald |
Scope of the Intramolecular Titanocene-Catalyzed Pauson−Khand Type Reaction |
J. Am. Chem. Soc. |
1999 |
Link |
|
149 |
M.V. Troutman; D.H. Appella; S.L. Buchwald |
Asymmetric Hydrogenation of Unfunctionalized Tetrasubstituted Olefins with a Cationic Zirconocene Catalyst |
J. Am. Chem. Soc. |
1999 |
Link |
|
148 |
A. Aranyos; D.W. Old; A. Kiyomori; J.P. Wolfe; J.P. Sadighi; S.L. Buchwald |
Novel Electron-Rich Bulky Phosphine Ligands Facilitate the Palladium-Catalyzed Preparation of Diaryl Ethers |
J. Am. Chem. Soc. |
1999 |
Link |
|
147 |
A. Kiyomori; J.F. Marcoux; S.L. Buchwald |
An efficient copper-catalyzed coupling of aryl halides with imidazoles |
Tet. Lett. |
1999 |
Link |
|
146 |
M. Hansen; S. Buchwald |
Synthesis of NPS R-568 utilizing titanium-catalyzed asymmetric hydrosilylation |
Tetrahedron Lett. |
1999 |
Link |
|
145 |
S.J. Sturla; N.M. Kablaoui; S.L. Buchwald |
A Titanocene-Catalyzed Intramolecular Ene Reaction: Cycloisomerization of Enynes and Dienynes |
J. Am. Chem. Soc. |
1999 |
Link |
|
144 |
R. Singer; S. Buchwald |
Preparation of 2-amino-2′-hydroxy-1,1′-binaphthyl and N-arylated 2-amino-1,1′-binaphthyl derivatives via palladium-catalyzed amination |
Tet. Lett. |
1999 |
Link |
|
143 |
B. Yang; S. Buchwald |
Palladium-Catalyzed Amination of Aryl Halides and Sulfonates |
J. Organomet. Chem. |
1999 |
Link |
|
142 |
D.W. Old; J.P. Wolfe; S.L. Buchwald |
A Highly Active Catalyst for Palladium-Catalyzed Cross-Coupling Reactions: Room-Temperature Suzuki Couplings and Amination of Unactivated Aryl Chlorides |
J. Am. Chem. Soc. |
1998 |
Link |
|
141 |
S. Akai; A.J. Peat; S.L. Buchwald |
Regioselective, directed meta acylation of aromatic compounds |
J. Am. Chem. Soc. |
1998 |
Link |
|
140 |
J.P. Wolfe; S. Wagaw; J.F. Marcoux; S.L. Buchwald |
Rational Development of Practical Catalysts for Aromatic Carbon−Nitrogen Bond Formation |
Acc. Chem. Res. |
1998 |
Link |
|
139 |
M.T. Reding; S.L. Buchwald |
Short Enantioselective Total Syntheses of the Piperidine Alkaloids (S)-Coniine and (2R,6R)-trans-Solenopsin A via Catalytic Asymmetric Imine Hydrosilylation |
J. Org. Chem. |
1998 |
Link |
|
138 |
S. Wagaw; B.H. Yang; S.L. Buchwald |
A palladium-catalyzed strategy for the preparation of indoles: A novel entry into the Fischer indole synthesis |
J. Am. Chem. Soc. |
1998 |
Link |
|
137 |
J.P. Sadighi; M.C. Harris; S.L. Buchwald |
A highly active palladium catalyst system for the arylation of anilines |
Tet. Lett. |
1998 |
Link |
|
136 |
R.A. Widenhoefer; S.L. Buchwald |
Electronic Dependence of C−O Reductive Elimination from Palladium (Aryl)neopentoxide Complexes |
J. Am. Chem. Soc. |
1998 |
Link |
|
135 |
J.P. Sadighi; R.A. Singer; S.L. Buchwald |
Palladium-catalyzed synthesis of monodisperse, controlled-length, and functionalized oligoanilines |
J. Am. Chem. Soc. |
1998 |
Link |
|
134 |
J. Ahman; J.P. Wolfe; M.V. Troutman; M. Palucki; S.L. Buchwald |
Asymmetric arylation of ketone enolates |
J. Am. Chem. Soc. |
1998 |
Link |
|
133 |
X. Verdaguer; U.E.W. Lange; S.L. Buchwald |
Amine additives greatly expand the scope of asymmetric hydrosilylation of imines |
Angew. Chem. Int. Ed. |
1998 |
Link |
|
132 |
M.C. Hansen; X. Verdaguer; S.L. Buchwald |
Convenient two-step conversion of lactones into cyclic ethers |
J. Org. Chem. |
1998 |
Link |
|
131 |
K. Aoki; A.J. Peat; S.L. Buchwald |
Titanocene-based method for indole synthesis |
J. Am. Chem. Soc. |
1998 |
Link |
|
130 |
R.A. Singer; J.P. Sadighi; S.L. Buchwald |
A general synthesis of end-functionalized oligoanilines via palladium-catalyzed amination |
J. Am. Chem. Soc. |
1998 |
Link |
|
129 |
M. Palucki; S.L. Buchwald |
Palladium-catalyzed alpha-arylation of ketones |
J. Am. Chem. Soc. |
1997 |
Link |
|
128 |
X. Verdaguer; M.C. Hansen; S.C. Berk; S.L. Buchwald |
Titanocene-Catalyzed Reduction of Lactones to Lactols |
J. Org. Chem. |
1997 |
Link |
|
127 |
J.F. Marcoux; S. Doye; S.L. Buchwald |
A general copper-catalyzed synthesis of diaryl ethers |
J. Am. Chem. Soc. |
1997 |
Link |
|
126 |
J.P. Wolfe; J. Ahman; J.P. Sadighi; R.A. Singer; S.L. Buchwald |
An ammonia equivalent for the palladium-catalyzed amination of aryl halides and triflates |
Tet. Lett. |
1997 |
Link |
|
125 |
J.Å. hman; S.L. Buchwald |
An Improved Method for the Palladium-Catalyzed Amination of Aryl Triflates |
Tet. Lett. |
1997 |
Link |
|
124 |
J.P. Wolfe; S.L. Buchwald |
Improved functional group compatibility in the palladium-catalyzed amination of aryl bromides |
Tet. Lett. |
1997 |
Link |
|
123 |
S. Wagaw; R.A. Rennels; S.L. Buchwald |
Palladium-Catalyzed Coupling of Optically Active Amines with Aryl Bromides |
J. Am. Chem. Soc. |
1997 |
Link |
|
122 |
J.P. Wolfe; S.L. Buchwald |
Room temperature catalytic amination of aryl iodides |
J. Org. Chem. |
1997 |
Link |
|
121 |
J.P. Wolfe; S.L. Buchwald |
Nickel-Catalyzed Amination of Aryl Chlorides |
J. Am .Chem .Soc. |
1997 |
Link |
|
120 |
R.A. Widenhoefer; H.A. Zhong; S.L. Buchwald |
Direct observation of C-O reductive elimination from palladium aryl alkoxide complexes to form aryl ethers |
J. Am. Chem. Soc. |
1997 |
Link |
|
119 |
N.M. Kablaoui; F.A. Hicks; S.L. Buchwald |
Titanocene-catalyzed cyclocarbonylation of o-allyl aryl ketones to gamma-butyrolactones |
J. Am. Chem. Soc. |
1997 |
Link |
|
118 |
M. Palucki; J.P. Wolfe; S.L. Buchwald |
Palladium-catalyzed intermolecular carbon-oxygen bond formation: A new synthesis of aryl ethers |
J. Am. Chem. Soc. |
1997 |
Link |
|
117 |
J.F. Marcoux; S. Wagaw; S.L. Buchwald |
Palladium-catalyzed amination of aryl bromides: Use of phosphinoether ligands for the efficient coupling of acyclic secondary amines |
J. Org. Chem. |
1997 |
Link |
|
116 |
J.P. Wolfe; S.L. Buchwald |
Palladium-Catalyzed Amination of Aryl Triflates |
J. Org. Chem. |
1997 |
Link |
|
115 |
B. Chin; S.L. Buchwald |
Improved Procedure for the Preparation of Enantiomerically Pure Ethylenebis(tetrahydroindenyl)zirconium Derivatives |
J. Org. Chem. |
1997 |
Link |
|
114 |
F.A. Hicks; S.L. Buchwald |
Highly enantioselective catalytic Pauson-Khand type formation of bicyclic cyclopentenones |
J. Am. Chem. Soc. |
1996 |
Link |
|
113 |
M. Palucki; J.P. Wolfe; S.L. Buchwald |
Synthesis of oxygen heterocycles via a palladium-catalyzed C-O bond-forming reaction |
J. Am. Chem. Soc. |
1996 |
Link |
|
112 |
F.A. Hicks; N.M. Kablaoui; S.L. Buchwald |
Titanocene-catalyzed cyclocarbonylation of enynes to cyclopentenones |
J. Am. Chem. Soc. |
1996 |
Link |
|
111 |
S. Wagaw; S.L. Buchwald |
The Synthesis of Aminopyridines: A Method Employing Palladium-Catalyzed Carbon-Nitrogen Bond Formation |
J. Org. Chem. |
1996 |
Link |
|
110 |
N.S. Radu; S.L. Buchwald; B. Scott; C.J. Burns |
Carbon-hydrogen bond activation of aromatic imines by(Cp*2SmH)(2) |
Organometallics |
1996 |
Link |
|
109 |
J.P. Wolfe; S. Wagaw; S.L. Buchwald |
An improved catalyst system for aromatic carbon-nitrogen bond formation: The possible involvement of bis(phosphine) palladium complexes as key intermediates |
J. Am. Chem. Soc. |
1996 |
Link |
|
108 |
R.A. Widenhoefer; S.L. Buchwald |
Formation of palladium bis(amine) complexes from reaction of amine with palladium tris(o-tolyl)phosphine mono(amine) complexes |
Organometallics |
1996 |
Link |
|
107 |
B. Chin; S.L. Buchwald |
An improved procedure for the resolution of (rac)-ethylenebis(tetrahydroindenyl)-titanium derivatives |
J. Org. Chem. |
1996 |
Link |
|
106 |
X. Verdaguer; U.E.W. Lange; M.T. Reding; S.L. Buchwald |
Highly enantioselective imine hydrosilylation using (S,S)-ethylenebis(eta(5)-tetrahydroindenyl)titanium difluoride |
J. Am. Chem. Soc. |
1996 |
Link |
|
105 |
M. Zhang; S.L. Buchwald |
A Nickel(0)-Catalyzed Process for the Transformation of Enynes to Bicyclic Cyclopentenones |
J. Org. Chem. |
1996 |
Link |
|
104 |
S. Bower; K.A. Kreutzer; S.L. Buchwald |
A mild general procedure for the one-pot conversion of amides to aldehydes |
Angew. Chem. Int. Ed. |
1996 |
Link |
|
103 |
N.M. Kablaoui; F.A. Hicks; S.L. Buchwald |
Diastereoselective synthesis of gamma-butyrolactones from enones mediated or catalyzed by a titanocene complex |
J. Am. Chem. Soc. |
1996 |
Link |
|
102 |
R.A. Widenhoefer; S.L. Buchwald |
Halide and Amine Influence in the Equilibrium Formation of Palladium Tris(o-tolyl)phosphine Mono(amine) Complexes from Palladium Aryl Halide Dimers |
Organometallics |
1996 |
Link |
|
101 |
R.A. Widenhoefer; H.A. Zhong; S.L. Buchwald |
Synthesis and solution structure of palladium tris(o-tolyl)phosphine mono(amine) complexes |
Organometallics |
1996 |
Link |
|
100 |
N.M. Kablaoui; S.L. Buchwald |
Development of a method for the reductive cyclization of enones by a titanium catalyst |
J. Am. Chem. Soc. |
1996 |
Link |
|
99 |
F.A. Hicks; S.C. Berk; S.L. Buchwald |
A Practical Titanium-Catalyzed Synthesis of Bicyclic Cyclopentenones and Allylic Amines |
J. Org. Chem. |
1996 |
Link |
|
98 |
J.P. Wolfe; R.A. Rennels; S.L. Buchwald |
Intramolecular palladium-catalyzed aryl amination and aryl amidation |
Tetrahedron |
1996 |
Link |
|
97 |
A.J. Peat; S.L. Buchwald |
Novel syntheses of tetrahydropyrroloquinolines: Applications to alkaloid synthesis |
J. Am. Chem. Soc. |
1996 |
Link |
|
96 |
J.P. Wolfe; S.L. Buchwald |
Palladium-catalyzed amination of aryl iodides |
J. Org. Chem. |
1996 |
Link |
|
95 |
X. Verdaguer; S.C. Berk; S.L. Buchwald |
Catalytic method for the reduction of lactones to lactols |
J. Am. Chem. Soc. |
1995 |
Link |
|
94 |
C.A. Willoughby; R.R. Duff; W.M. Davis; S.L. Buchwald |
Preparation of novel titanium complexes bearing o-phosphinophenol ligands |
Organometallics |
1996 |
Link |
|
93 |
M.T. Reding; S.L. Buchwald |
An Inexpensive Air-Stable Titanium-Based System for the Conversion of Esters to Primary Alcohols |
J. Org. Chem. |
1995 |
Link |
|
92 |
F.M.G. Derege; W.M. Davis; S.L. Buchwald |
Synthesis and Structure of Zirconium Group-13 Heterobimetallic Compounds |
Organometallics |
1995 |
Link |
|
91 |
B.P. Warner; S.P. Millar; R.D. Broene; S.L. Buchwald |
Controlled acceleration and inhibition of bergman cyclization by metal chlorides |
Science |
1995 |
Link |
|
90 |
J.R. Johnson; G.D. Cuny; S.L. Buchwald |
Rhodium-Catalyzed Hydroformylation of Internal Alkynes to α,β-Unsaturated Aldehydes |
Angew. Chem. Int. Ed. |
1995 |
Link |
|
89 |
N.M. Kablaoui; S.L. Buchwald |
Reductive Cyclization of Enones by a Titanium Catalyst |
J. Am. Chem. Soc. |
1995 |
Link |
|
88 |
A.S. Guram; R.A. Rennels; S.L. Buchwald |
A Simple Catalytic Method for the Conversion of Aryl Bromides to Arylamines |
Angew. Chem. Int. Ed. |
1995 |
Link |
|
87 |
G.D. Cuny; S.L. Buchwald |
Regioselective Olefin Hydroformylation as a Route to Indolizidine and Pyrrolizidine Alkaloids |
Synlett |
1995 |
Link |
|
86 |
C.A. Willoughby; W.M. Davis; S.L. Buchwald |
Preparation and X-ray structure of a novel chiral methylene bridged titanocene complex |
J. Organomet. Chem. |
1995 |
Link |
|
85 |
J. Campora; S.L. Buchwald; E. Gutierrez-Puebla; A. Monge |
Kinetics and Mechanism of the Reductive Elimination of Cyclic Titanocene Iminoacyls |
Organometallics |
1995 |
Link |
|
84 |
F.M.G. de Rege; S.L. Buchwald |
The regioselective synthesis of halophenols |
Tetrahedron |
1995 |
Link |
|
83 |
C.A. Willoughby; S.L. Buchwald |
Catalytic Asymmetric Hydrogenation of Imines with a Chiral Titanocene Catalyst: Kinetic and Mechanistic Investigations |
J. Am. Chem. Soc. |
1994 |
Link |
|
82 |
J.H. Tidwell; S.L. Buchwald |
Synthesis of Polysubstituted Indoles and Indolines by Means of Zirconocene-Stabilized Benzyne Complexes |
J. Am. Chem. Soc. |
1994 |
Link |
|
81 |
J.H. Tidwell; A.J. Peat; S.L. Buchwald |
Synthesis and Reactions of 3-(Bromomethyl)-1-carbethoxy-4-iodoindole: The Preparation of 3,4-Differentially Substituted Indoles |
J. Org. Chem. |
1994 |
Link |
|
80 |
E. Spaltenstein; P. Palma; K.A. Kreutzer; C.A. Willoughby; W.M. Davis; S.L. Buchwald |
Preparation and X-ray Structure of Cp2Ti(Ph2SiH2)(PMe3) |
J. Am. Chem. Soc. |
1994 |
Link |
|
79 |
M.Beth Carter; B. Schiott; A. Gutierrez; S.L. Buchwald |
Enantioselective Hydrosilylation of Ketones with a Chiral Titanocene Catalyst |
J. Am. Chem. Soc. |
1994 |
Link |
|
78 |
A. Viso; N.E. Lee; S.L. Buchwald |
Kinetic resolution of racemic disubstituted 1-pyrrolines via asymmetric reduction with a chiral titanocene catalyst |
J. Am. Chem. Soc. |
1994 |
Link |
|
77 |
D.P. Hsu; B.P. Warner; R.A. Fisher; W.M. Davis; S.L. Buchwald |
Synthesis and Structure of a Novel Bis(stibole) |
Organometallics |
1994 |
Link |
|
76 |
C.A. Willoughby; S.L. Buchwald |
Catalytic Asymmetric Hydrogenation of Imines with a Chiral Titanocene Catalyst: Scope and Limitations |
J. Am. Chem. Soc. |
1994 |
Link |
|
75 |
B.P. Warner; S.L. Buchwald |
A Catalytic Method for the Conversion of Silanes to Stannanes |
J. Org. Chem. |
1994 |
Link |
|
74 |
S.C. Berk; R.B. Grossman; S.L. Buchwald |
Development of a Titanocene-Catalyzed Enyne Cyclization/Isocyanide Insertion Reaction |
J. Am. Chem. Soc. |
1994 |
Link |
|
73 |
A.F. England; C.J. Burns; S.L. Buchwald |
New Syntheses of Cp*2Th(Ph)2 and Cp*2Th(Me)(aryl) Derivatives |
Organometallics |
1994 |
Link |
|
72 |
R.B. Grossman; J.C. Tsai; W.M. Davis; A. Gutierrez; S.L. Buchwald |
Synthesis and Structure of a C2-Symmetric, Doubly Bridged ansa-Titanocene Complex |
Organometallics |
1994 |
Link |
|
71 |
A.S. Guram; S.L. Buchwald |
Palladium-Catalyzed Aromatic Aminations with in situ Generated Aminostannanes |
J. Am. Chem. Soc. |
1994 |
Link |
|
70 |
K.J. Barr; S.C. Berk; S.L. Buchwald |
Titanocene-Catalyzed Reduction of Esters Using Polymethylhydrosiloxane as the Stoichiometric Reductant |
J. Org. Chem. |
1994 |
Link |
|
69 |
N.E. Lee; S.L. Buchwald |
Asymmetric Hydrogenation of Enamines with a Chiral Titanocene Catalyst |
J. Am. Chem. Soc. |
1994 |
Link |
|
68 |
B.P. Warner; W.M. Davis; S.L. Buchwald |
Synthesis and X-ray Structure of a Zirconocene Complex of Two Alkynes |
J. Am. Chem. Soc. |
1994 |
Link |
|
67 |
C.A. Willoughby; S.L. Buchwald |
Synthesis of highly enantiomerically enriched cyclic amines by the catalytic asymmetric hydrogenation of cyclic imines |
J. Org. Chem. |
1993 |
Link |
|
66 |
R.D. Broene; S.L. Buchwald |
Asymmetric hydrogenation of unfunctionalized trisubstituted olefins with a chiral titanocene catalyst |
J. Am. Chem. Soc. |
1993 |
Link |
|
65 |
D.P. Hsu; W.M. Davis; S.L. Buchwald |
Synthesis and structure of seven-membered cyclic cumulene |
J. Am. Chem. Soc. |
1993 |
Link |
|
64 |
J. Campora; S.L. Buchwald |
Synthesis and reactivity of a titanocene-benzyne complex |
Organometallics |
1993 |
Link |
|
63 |
R.D. Broene; S.L. Buchwald |
Zirconocene complexes of unsaturated organic molecules: new vehicles for organic synthesis |
Science |
1993 |
Link |
|
62 |
S.C. Berk; R.B. Grossman; S.L. Buchwald |
Titanocene-catalyzed conversion of enynes to bicyclic cyclopentenones |
J. Am. Chem. Soc. |
1993 |
Link |
|
61 |
J.H. Tidwell; S.L. Buchwald |
A new approach to the synthesis of the CC-1065/duocarmycin pharmacophore |
J. Org. Chem. |
1992 |
Link |
|
60 |
G.D. Cuny; S.L. Buchwald |
Practical, high-yield, regioselective, rhodium-catalyzed hydroformylation of functionalized .alpha.-olefins |
J. Am. Chem. Soc. |
1993 |
Link |
|
59 |
R.B. Grossman; S.L. Buchwald |
Reductive cyclization of ester-containing enynes with a practical titanocene reagent. Synthesis of bicyclic cyclopentenones and iminocyclopentenes |
J. Org. Chem. |
1992 |
Link |
|
58 |
C.A. Willoughby; S.L. Buchwald |
Asymmetric titanocene-catalyzed hydrogenation of imines |
J. Am. Chem. Soc. |
1992 |
Link |
|
57 |
R.E. v H. Spence; D.P. Hsu; S.L. Buchwald |
Synthesis of thermochromic dibismuthines with nonthermochromic distibine analogs |
Organometallics |
1992 |
Link |
|
56 |
R.E. v H. Spence; S.L. Buchwald; J.F. Richardson |
The Unexpected Formation of 3,4,7,8-Tetramethyl-1,2,5,6-tetrahydrodicyclobuta[a, e]cyclooctene from a Zirconacyclopentadiene |
Acta Chem. Scand. |
1993 |
Link |
|
55 |
S.C. Berk; S.L. Buchwald |
An air-stable catalyst system for the conversion of esters to alcohols |
J. Org. Chem. |
1992 |
Link |
|
54 |
K.J. Barr; B.T. Watson; S.L. Buchwald |
Zirconocene(iso-butyl) chloride: In situ generation of a zirconocene(methyl) chloride equivalent for use in organic synthesis |
Tet. Lett. |
1991 |
Link |
|
53 |
S.C. Berk; K.A. Kreutzer; S.L. Buchwald |
A catalytic method for the reduction of esters to alcohols |
J. Am. Chem. Soc. |
1991 |
Link |
|
52 |
J.H. Tidwell; D.R. Senn; S.L. Buchwald |
Synthesis of 3,4-disubstituted indoles via a sequential olefin-insertion/ene route |
J. Am. Chem. Soc. |
1991 |
Link |
|
51 |
S.L. Buchwald; S.J. LaMaire; R.B. Nielsen; B.T. Watson; S.M. King |
Schwartz's Reagent |
Org. Synth. |
1993 |
Link |
|
50 |
K.A. Kreutzer; R.A. Fisher; W.M. Davis; E. Spaltenstein; S.L. Buchwald |
Synthesis, characterization, and reactivity of zirconocene and hafnocene silyl hydride complexes |
Organometallics |
1991 |
Link |
|
49 |
G.D. Cuny; A. Gutierrez; S.L. Buchwald |
Cis difunctionalization of cyclic olefins with use of organozirconium intermediates |
Organometallics |
1991 |
Link |
|
48 |
R.B. Grossman; W.M. Davis; S.L. Buchwald |
Enantioselective, zirconium-mediated synthesis of allylic amines |
J. Am. Chem. Soc. |
1991 |
Link |
|
47 |
R.B. Grossman; R.Ann Doyle; S.L. Buchwald |
Syntheses of [ethylene-1,2-bis(.eta.5-4,5,6,7-tetrahydro-1-indenyl)]zirconium and -hafnium hydride complexes. Improved syntheses of the corresponding dichlorides |
Organometallics |
1991 |
Link |
|
46 |
R.A. Fisher; R.B. Nielsen; W.M. Davis; S.L. Buchwald |
Stibathiolanes: synthesis, solid-state structure, and solution behavior |
J. Am. Chem. Soc. |
1991 |
Link |
|
45 |
S.L. Buchwald; S.M. King |
The regiospecific synthesis of polysubstituted naphthalenes and iodo(acyl)naphthoquinones via zirconocene complexes of naphthalynes |
J. Am. Chem. Soc. |
1991 |
Link |
|
44 |
G.D. Cuny; S.L. Buchwald |
Ring-opening reactions of cyclic allylic ethers by zirconocene complexes of cyclic alkynes |
Organometallics |
1991 |
Link |
|
43 |
D.P. Hsu; E.A. Lucas; S.L. Buchwald |
Synthesis and reactions of a zirconocene-benzdiyne equivalent |
Tet. Lett. |
1990 |
Link |
|
42 |
S.L. Buchwald; R.A. Fisher; B.M. Foxman |
The Synthesis and Structure of Stibaindoles |
Angew. Chem. Int. Ed. |
1990 |
Link |
|
41 |
R.A. Fisher; S.L. Buchwald |
Synthesis, structure, and reactivity of a zirconocene complex of cyclobutene |
Organometallics |
1990 |
Link |
|
40 |
S.L. Buchwald; K.A. Kreutzer; R.A. Fisher |
Synthesis, reactions, and x-ray crystal structure determination of hafnocene complex Cp2Hf(isobutylene).cntdot.PMe3 |
J. Am. Chem. Soc. |
1990 |
Link |
|
39 |
S.L. Buchwald; R.A. Fisher |
Zirconocene Complexes of Unsaturated Organic Molecules |
Chemica Scripta |
1989 |
Link |
|
38 |
S.L. Buchwald; R.T. Lum; R.A. Fisher; W.M. Davis |
Synthesis and x-ray crystal structure of a zirconocene complex of a cyclopentyne and its use to prepare bicyclic cyclopentenones |
J. Am. Chem. Soc. |
1989 |
Link |
|
37 |
S.L. Buchwald; R.A. Fisher; W.M. Davis |
Synthesis and structure of novel antimony thiametallacycles |
Organometallics |
1989 |
Link |
|
36 |
S.L. Buchwald; Q. Fang |
An efficient one-pot method for the preparation of polysubstituted benzothiophenes |
J. Org. Chem. |
1989 |
Link |
|
35 |
S.L. Buchwald; R.B. Nielsen; J.C. Dewan |
Synthesis of (alkoxymethyl)zirconocene chlorides: stereochemistry of carbon-carbon bond formation in a zirconocene-Wittig rearrangement |
Organometallics |
1989 |
Link |
|
34 |
S.L. Buchwald; B.T. Watson; W. Wannamaker; J.C. Dewan |
Zirconocene complexes of imines. General synthesis, structure, reactivity, and in situ generation to prepare geometrically pure allylic amines |
J. Am. Chem. Soc. |
1989 |
Link |
|
33 |
S.L. Buchwald; E.A. Lucas; W.M. Davis |
A bimetallic zirconium complex containing an in-plane bridging aromatic ring |
J. Am. Chem. Soc. |
1989 |
Link |
|
32 |
S.L. Buchwald; R.B. Nielsen |
Selective, zirconium-mediated cross-coupling of alkynes: the synthesis of isomerically pure 1,3-dienes and 1,4-diiodo-1,3-dienes |
J. Am. Chem. Soc. |
1989 |
Link |
|
31 |
S.L. Buchwald; W. Wannamaker; B.T. Watson |
Synthesis of substituted pyrroles via zirconocene complexes of imines |
J. Am. Chem. Soc. |
1989 |
Link |
|
30 |
A. Vaughan; G.L. Hillhouse; R.T. Lum; S.L. Buchwald; A.L. Rheingold |
Oxygen-atom transfer from nitrous oxide. Synthesis and structure of a zirconocene oxametallacyclobutene complex |
J. Am. Chem. Soc. |
1988 |
Link |
|
29 |
S.L. Buchwald; R.B. Nielsen |
Group 4 metal complexes of benzynes, cycloalkynes, acyclic alkynes, and alkenes |
Chemical Reviews |
1988 |
Link |
|
28 |
S.L. Buchwald; Q. Fang; S.M. King |
A new method for the preparation of 3,5-disubstituted butenolides |
Tet. Lett. |
1988 |
Link |
|
27 |
S.L. Buchwald; R.B. Nielsen; J.C. Dewan |
Synthesis, structure, and reactions of (1-ethoxyethyl)zirconocene chloride, a stable acyclic secondary zirconocene alkyl |
Organometallics |
1988 |
Link |
|
26 |
S.L. Buchwald; R.B. Nielsen |
Kinetics and substituent effects in the formation of zirconocene thioaldehyde complexes: .beta.-hydride elimination versus cyclometalation |
J. Am. Chem. Soc. |
1988 |
Link |
|
25 |
S.L. Buchwald; B.T. Watson; R.T. Lum; W.A. Nugent |
A general method for the preparation of zirconocene complexes of substituted benzynes: in situ generation, coupling reactions, and use in the synthesis of polyfunctionalized aromatic compounds |
J. Am. Chem. Soc. |
1987 |
Link |
|
24 |
S.L. Buchwald; S.J. LaMaire; R.B. Nielsen; B.T. Watson; S.M. King |
A Modified Procedure for the Preparation of Cp2Zr(H)Cl (Schwartz's Reagent) |
Tet. Lett. |
1987 |
Link |
|
23 |
J.C. Dewan; E.A. Lucas; S.L. Buchwald |
Synthesis, structure, and reactions of a zirconocene-benzdiyne complex |
J. Am. Chem. Soc. |
1987 |
Link |
|
22 |
S.L. Buchwald; A. Sayers; B.T. Watson; J.C. Dewan |
The zirconocene induced coupling of benzyne with nitriles: Synthesis, structure and reactions of novel azametallacyclopentenes |
Tet. Lett. |
1987 |
Link |
|
21 |
S.L. Buchwald; B.T. Watson; J.C. Huffman |
The synthesis, reactions and molecular structure of zirconocene-alkyne complexes |
J. Am. Chem. Soc. |
1987 |
Link |
|
20 |
S.L. Buchwald; R.B. Nielsen; J.C. Dewan |
The synthesis, structure and reactivity of trimethylphosphine-zirconocene thioaldehyde complexes |
J. Am. Chem. Soc. |
1987 |
Link |
|
19 |
S.L. Buchwald; S.J. LaMaire |
A regiospecific method for the hydrocyanation of olefins |
Tet. Lett. |
1987 |
Link |
|
18 |
S.L. Buchwald; R.T. Lum; J.C. Dewan |
Synthesis, structure, and reactions of a zirconocene-cyclohexyne complex |
J. Am. Chem. Soc. |
1986 |
Link |
|
17 |
S.L. Buchwald; B.T. Watson; J.C. Huffman |
Trimethylphosphine adduct of the zirconocene-benzyne complex: synthesis, reactions, and x-ray crystal structure |
J. Am. Chem. Soc. |
1986 |
Link |
|
16 |
L. Clawson; J. Soto; S.L. Buchwald; M.L. Steigerwald; R.H. Grubbs |
Olefin insertion in a metal alkyl in a Ziegler polymerization system |
J. Am. Chem. Soc. |
1985 |
Link |
|
15 |
S.L. Buchwald; E.V. Anslyn; R.H. Grubbs |
Reaction of dicyclopentadienylmethylenetitanium with organic halides: Evidence for a radical mechanism |
J. Am. Chem. Soc. |
1985 |
Link |
|
14 |
L. Clawson; S.L. Buchwald; R.H. Grubbs |
The methylenation of enolizable ketones and esters using organotitanium chemistry |
Tet. Lett. |
1984 |
Link |
|
13 |
S.L. Buchwald; M.S. Saini; J.R. Knowles; R.L. Van Etten |
Stereochemical course of phospho group transfer by human prostatic acid phosphatase |
J. Biol. Chem. |
1984 |
|
|
12 |
S.L. Buchwald; D.H. Pliura; J.R. Knowles |
Stereochemical evidence for pseudorotation in the reaction of a phosphoric monoester |
J. Am. Chem. Soc. |
1984 |
Link |
|
11 |
S.L. Buchwald; J.M. Friedman; J.R. Knowles |
Stereochemistry of nucleophilic displacement on two phosphoric monoesters and a phosphoguanidine: the role of metaphosphate |
J. Am. Chem. Soc. |
1984 |
Link |
|
10 |
K.A. Brown-Wensley; S.L. Buchwald; L. Cannizzo; L. Clawson; H. S.; D. Meinhardt; J.R. Stille; D. Straus; R.H. Grubbs |
CP2TiCH2 Complexes in Synthetic Applications |
Pure Appl. Chem. |
1983 |
Link |
|
9 |
S.L. Buchwald; R.H. Grubbs |
A titanium vinylidene route to substituted allenes |
J. Am. Chem. Soc. |
1983 |
Link |
|
8 |
K.A. Parker; J.J. Petraitis; R.W. Kosley; S.L. Buchwald |
Reactions of propargyl alcohols with amide acetals |
J. Org. Chem. |
1982 |
Link |
|
7 |
S.L. Buchwald; D.H. Pliura; J.R. Knowles |
Stereochemistry and mechanism of an acid-catalyzed 1,2-phospho group migration: evidence for pseudorotation in the reaction of a phosphoric monoester |
J. Am. Chem. Soc. |
1982 |
Link |
|
6 |
S.L. Buchwald; J.R. Knowles |
Nucleophilic displacements on phosphoric monoesters: stereochemical evidence |
J. Am. Chem. Soc. |
1982 |
Link |
|
5 |
S.L. Buchwald; D.E. Hansen; A. Hassett; J.R. Knowles |
Chiral [16O, 17O, 18O]phosphoric monoesters as stereochemical probes of phosphotransferases |
Methods Enzymol. |
1982 |
|
|
4 |
M.S. Saini; S.L. Buchwald; R.L. Van Etten; J.R. Knowles |
Stereochemistry of phospho transfer catalyzed by bovine liver acid phosphatase |
J. Biol. Chem. |
1981 |
|
|
3 |
S.L. Buchwald; J.R. Knowles |
Determination of the absolute configuration of [16O,17O,18O]phosphate monoesters by using phosphorus-31 NMR |
J. Am. Chem. Soc. |
1980 |
Link |
|
2 |
D.E. Cane; S.L. Buchwald |
Application of deuterium magnetic resonance to biosynthetic studies. 1. Biosynthesis of ovalicin |
J. Am. Chem. Soc. |
1977 |
Link |
|
1 |
K.A. Parker; R.W. Kosley; S.L. Buchwald; J.J. Petraitis |
The Reaction of Tertiary Ethynyl Alcohols with Formamide Acetals: Formation of Dienamines and Enamine Orthoformates |
J. Am. Chem. Soc. |
1976 |
Link |
|
|
|
|
|
Submitted |
|
