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K. Feng; E.Reichert Raguram; J.R. Howard; E. Peters; C. Liu; M.S. Sigman; S.L. Buchwald |
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J. Am. Chem. Soc. |
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Site-Specific Antibody Prodrugs via S‑Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues |
J. Am. Chem. Soc. |
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M.J. Strauss; K.X. Liu; M.E. Greaves; J.C. Dahl; S.T. Kim; Y.J. Wu; M.A. Schmidt; P.M. Scola; S.L. Buchwald |
Cu-Catalyzed Amination of Base-Sensitive Aryl Bromides and the Chemoselective N- and O-Arylation of Amino Alcohols |
J. Am. Chem. Soc. |
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J. Am. Chem. Soc. |
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M.J. Strauss; M.E. Greaves; S.T. Kim; C.N. Teijaro; M.A. Schmidt; P.M. Scola; S.L. Buchwald |
Room-Temperature Copper-Catalyzed Etherification of Aryl Bromides |
Angewandte Chemie |
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N.M. Grob; C. Remarcik; S.L. Rössler; J.Y.K. Wong; J.C.K. Wong; J. Tao; C.L. Smith; A. Loas; S.L. Buchwald; D.L. Eaton; M.P. López; B.L. Pentelute |
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J. Am. Chem. Soc. |
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J. Am. Chem. Soc. |
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S.L. Rössler; N.M. Grob; S.L. Buchwald; B.L. Pentelute |
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Y. Ye; S.T. Kim; R.P. King; M.H. Baik; S.L. Buchwald |
Studying Regioisomer Formation in the Pd-Catalyzed Fluorination of Cyclic Vinyl Triflates: Evidence for in situ Ligand Modification |
Angew. Chem. Int. Ed. |
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J. Am. Chem. Soc. |
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J.Levi Knippel; A.Z. Ni; A.W. Schuppe; S.L. Buchwald |
A General Strategy for the Asymmetric Preparation of α-Stereogenic Allyl Silanes, Germanes, and Boronate Esters via Dual Copper Hydride- and Palladium-Catalysis |
Angew. Chem. Int. Ed. |
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A.Jose Rojas; J.M. Wolfe; H.H. Dhanjee; I. Buslov; N.L. Truex; R.Y. Liu; W. Massefski; B. Pentelute; S.L. Buchwald |
Palladium−Peptide Oxidative Addition Complexes for Bioconjugation |
Chem. Sci. |
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Palladium Mediated Synthesis of Protein–Polyarene Conjugates |
J. Am. Chem. Soc. |
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Enantioselective Hydrocarbamoylation of Alkenes |
Angew. Chem. Int. Ed. |
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Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins |
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Org. Lett. |
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M. Jbara; S. Pomplun; C.K. Schissel; S.Wilson Hawken; A. Boija; I. Klein; J. Rodriguez; S.L. Buchwald; B.L. Pentelute |
Engineering Bioactive Dimeric Transcription Factor Analogs via Palladium Rebound Reagents |
J. Am. Chem. Soc. |
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A. Mallek; B.L. Pentelute; S.L. Buchwald |
Selective N-Arylation of p-Aminophenylalanine in Unprotected Peptides with Organometallic Palladium Reagents |
Angew. Chem. Int. Ed. |
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A.W. Schuppe; J.Levi Knippel; G.M. Borrajo-Calleja; S.L. Buchwald |
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J. Am. Chem. Soc. |
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CuH-Catalyzed Regio- and Enantioselective Hydrocarboxylation of Allenes; Toward Carboxylic Acids with Acyclic Quarternary Centers |
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Oligonucleotide Bioconjugation with Bifunctional Palladium Reagents |
Angew. Chem., Int. Ed. |
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Enantioselective C2-Allylation of Benzimidazoles Using 1,3-Diene Pronucleophiles |
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H.H. Dhanjee; I. Buslov; I.W. Windsor; R.T. Raines; B.L. Pentelute; S.L. Buchwald |
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J. Am. Chem. Soc. |
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S.D. McCann; E.C. Reichert; P.Luis Arrechea; S.L. Buchwald |
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Enantioselective Synthesis of β-Amino Acid Derivatives Enabled by Ligand-Controlled Reversal of Hydrocupration Regiochemistry |
Angew. Chem. Int. Ed. |
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Y. Mo; Z. Lu; G. Rughoobur; P. Patil; N. Gershenfeld; A.I. Akinwande; S.L. Buchwald; K.F. Jensen |
Microfluidic electrochemistry for single-electron transfer redox-neutral reactions |
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M.W. Gribble; R.Y. Liu; S.L. Buchwald |
Evidence for Simultaneous Dearomatization of Two Aromatic Rings Under Mild Conditions in Cu(I)-Catalyzed Direct Asymmetric Dearomatization of Pyridine |
J. Am. Chem. Soc. |
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Z. Lu; S.L. Buchwald |
The Enantioselective Preparation of Arenes with β-Stereogenic Centers: Confronting the 1,1-Disubstituted Olefin Problem Using CuH/Pd Cooperative Catalysis |
Angew. Chem. Int. Ed. |
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Highly Enantioselective Synthesis of Indazoles with a C3-Quaternary Chiral Center Using CuH Catalysis |
J. Am. Chem. Soc. |
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CuH-Catalyzed Olefin Functionalization: From Hydroamination to Carbonyl Addition |
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Synthesis of Pyrroles Through the CuH-Catalyzed Coupling of Enynes and Nitriles |
J. Am. Chem. Soc. |
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H.H. Dhanjee; A. Saebi; I. Buslov; A.R. Loftis; S.L. Buchwald; B.L. Pentelute |
Protein–Protein Cross-Coupling via Palladium–Protein Oxidative Addition Complexes from Cysteine Residues |
J. Am. Chem. Soc |
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R.Y. Liu; J.M. Dennis; S.L. Buchwald |
The Quest for the Ideal Base: Rational Design of a Nickel Precatalyst Enables Mild, Homogeneous C–N Cross-Coupling |
J. Am. Chem. Soc. |
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B.Y. Park; M.T. Pirnot; S.L. Buchwald |
Visible Light-Mediated (Hetero)aryl Amination Using Ni(II) Salts and Photoredox Catalysis in Flow: A Synthesis of Tetracaine |
J. Org. Chem. |
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Diastereo- and Enantioselective CuH-Catalyzed Hydroamination of Strained Trisubstituted Alkenes |
ACS Catal |
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Enantioselective Olefin Hydrocyanation Without Cyanide |
J. Am. Chem. Soc. |
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S. Ichikawa; S.L. Buchwald |
Asymmetric Synthesis of γ-Amino Alcohols by Copper-Catalyzed Hydroamination |
Organic Letters |
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R.P. King; S.L. Buchwald |
Synthesis of (MeCN)2Pd(CF3)OTs, a General Precursor to Palladium(II) Trifluoromethyl Complexes LPd(CF3)X |
Organometallics |
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C. Li*; K. Shin*; R. Y.Liu; S.L. Buchwald |
Engaging Aldehydes in CuH-Catalyzed Reductive Coupling Reactions: Stereoselective Allylation with Unactivated 1,3-Diene Pronucleophiles |
Angew. Chem. Int. Ed. |
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C.C. Wagen; B.T. Ingoglia; S.L. Buchwald |
Unexpected Formation of Hexasubstituted Arenes through a Twofold Palladium-Mediated Ligand Arylation |
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Copper Hydride-Catalyzed Enantioselective Synthesis of Axially Chiral 1,3-Disubstituted Allenes |
J. Am. Chem. Soc. |
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W. Huang; M. Einzinger; A. Maurano; T. Zhu; J. Tiepelt; C. Yu; H.Sik Chae; T. Van Voorhis; M.A. Baldo; S.L. Buchwald |
Large Increase in External Quantum Efficiency by Dihedral Angle Tuning in a Sky-Blue Thermally Activated Delayed Fluorescence Emitter |
Adv. Optical Mater. |
2019 |
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L.M. Baumgartner; J.M. Dennis; N.A. White; S.L. Buchwald; K.F. Jensen |
Use of a Droplet Platform To Optimize Pd-Catalyzed C–N Coupling Reactions Promoted by Organic Bases |
Org. Process Res. Dev. |
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J. Xu; R.Y. Liu; C.S. Yeung; S.L. Buchwald |
Monophosphine Ligands Promote Pd-Catalyzed C–S Cross-Coupling Reactions at Room Temperature with Soluble Bases |
ACS Catalysis |
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Regio- and Enantioselective Synthesis of 1,2-Diamine Derivatives by Copper-Catalyzed Hydroamination |
Org. Lett. |
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B.T. Ingoglia; C.C. Wagen; S.L. Buchwald |
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Pd-Catalyzed C–N Coupling Reactions Facilitated by Organic Bases: Mechanistic Investigation Leads to Enhanced Reactivity in the Arylation of Weakly Binding Amines |
ACS Catalysis |
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C. Li; R.Y. Liu; L.T. Jesikiewicz; Y. Yang; P. Liu; S.L. Buchwald |
CuH-Catalyzed Enantioselective Ketone Allylation with 1,3-Dienes: Scope, Mechanism, and Applications |
J. Am. Chem. Soc. |
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Y. Ye; S.T. Kim; J. Jeong; M.H. Baik; S.L. Buchwald |
CuH-Catalyzed Enantioselective Alkylation of Indole Derivatives with Ligand-Controlled Regiodivergence |
J. Am. Chem. Soc. |
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R.Y. Liu; Y. Zhou; Y. Yang; S.L. Buchwald |
Enantioselective Allylation Using Allene, a Petroleum Cracking Byproduct |
J. Am. Chem. Soc. |
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X.J. Dai; O.D. Engl; T. León; S.L. Buchwald |
Catalytic Asymmetric Synthesis of α-Arylpyrrolidines and Benzo-fused Nitrogen Heterocycles |
Angew. Chem. Int. Ed. |
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M.R. Uehling; R.P. King; S.W. Krska; T. Cernak; S.L. Buchwald |
Pharmaceutical diversification via palladium oxidative addition complexes |
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D.T. Cohen; C. Zhang; C.M. Fadzen; A.J. Mijalis; L. Hie; K.D. Johnson; Z. Shriver; O. Plante; S.J. Miller; S.L. Buchwald; B.L. Pentelute |
A chemoselective strategy for late-stage functionalization of complex small molecules with polypeptides and proteins |
Nat. Chem. |
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C. Zhang; E.V. Vinogradova; A.M. Spokoyny; S.L. Buchwald; B.L. Pentelute |
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Angew. Chem. Int. Ed. |
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A Practical Electrophilic Nitrogen Source for the Synthesis of Chiral Primary Amines by Copper-Catalyzed Hydroamination |
J. Am. Chem. Soc. |
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A.A. Thomas; K. Speck; I. Kevlishvili; Z. Lu; P. Liu; S.L. Buchwald |
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J. Am. Chem. Soc. |
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K.M. Khan; Y. Zhao; T. Scully; S.L. Buchwald |
Catalytic Arylhydroxylation of Dehydroalanine in Continuous Flow for Simple Access to Unnatural Amino Acids |
Chem. Eur. J. |
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S. Ichikawa; S. Zhu; S.L. Buchwald |
A Modified System for the Synthesis of Enantioenriched N‐Arylamines through Copper‐Catalyzed Hydroamination |
Angew. Chem. Int. Ed. |
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Angew. Chem. Int. Ed. |
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Copper-Catalyzed Enantioselective Hydroamination of Alkenes |
Org. Syn. |
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M.W. Gribble; S. Guo; S.L. Buchwald |
Asymmetric Cu-Catalyzed 1,4-Dearomatization of Pyridines and Pyridazines without Preactivation of the Heterocycle or Nucleophile |
J. Am. Chem. Soc. |
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J.M. Dennis; N.A. White; R.Y. Liu; S.L. Buchwald |
Breaking the Base Barrier: An Electron-Deficient Palladium Catalyst Enables the Use of a Common, Soluble Base in C–N Coupling |
J. Am. Chem. Soc. |
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Palladium-Catalyzed C–O Cross-Coupling of Primary Alcohols |
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Molecular Design of Deep Blue Thermally Activated Delayed Fluorescence Materials Employing a Homoconjugative Triptycene Scaffold and Dihedral Angle Tuning |
Chem. Mater. |
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K. Kubota; P. Dai; B.L. Pentelute; S.L. Buchwald |
Palladium Oxidative Addition Complexes for Peptide and Protein Crosslinking |
J. Am. Chem. Soc. |
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Mechanistic Insight Facilitates Discovery of a Mild and Efficient Copper-Catalyzed Dehydration of Primary Amides to Nitriles Using Hydrosilanes |
J. Am. Chem. Soc. |
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CuH-Catalyzed Asymmetric Reduction of α,β-Unsaturated Carboxylic Acids to β-Chiral Aldehydes |
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J. Am. Chem. Soc |
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Water-Soluble Palladium Reagents for Cysteine S-Arylation under Ambient Aqueous Conditions |
Org. Lett. |
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Palladium-Catalyzed Negishi Coupling of α-CF3 Oxiranyl Zincate: Access to Chiral CF3-substituted Benzylic Tertiary Alcohols |
J. Am. Chem. Soc |
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Mechanistic Insight Leads to a Ligand That Facilitates the Pd-Catalyzed Formation of 2-(Hetero)Arylaminooxazoles and 4-(Hetero)Arylaminothiazoles |
Angew. Chem. Int. Ed. |
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CuH-Catalyzed Regioselective Intramolecular Hydroamination for the Synthesis of Alkyl-Substituted Chiral Aziridines |
J. Am. Chem. Soc |
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Enantioselective CuH-Catalyzed Hydroacylation Employing Unsaturated Carboxylic Acids as Aldehyde Surrogates |
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Angew. Chem. Int. Ed. |
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Oxidative Addition Complexes as Precatalysts for Cross-Coupling Reactions Requiring Extremely Bulky Biarylphosphine Ligands |
Org. Lett. |
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Direct 11CN-Labeling of Unprotected Peptides via Palladium-Mediated Sequential Cross-Coupling Reactions |
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A.J. Rojas; C. Zhang; E.V. Vinogradova; N. Buchwald; J. Reilly; B.L. Pentelute; S.L. Buchwald |
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Chem. Sci. |
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Palladium-Mediated Arylation of Lysine in Unprotected Peptides |
Angew. Chem. Int. Ed. |
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Angew. Chem. Int. Ed. |
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Reaction Chemistry & Engineering |
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Angew. Chem. Int. Ed. |
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Biaryl Phosphine Based Pd(II) Amido Complexes: The Effect of Ligand Structure on Reductive Elimination |
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Rapid Synthesis of Aryl Fluorides in Continuous Flow through the Balz–Schiemann Reaction |
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New Insights into Xantphos/Pd-Catalyzed C−N Bond Forming Reactions: A Structural and Kinetic Study |
Organometallics |
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Expedited Palladium-Catalyzed Amination of Aryl Nonaflates through the Use of Microwave-Irradiation and Soluble Organic Amine Bases |
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Evidence for the Formation and Structure of Palladacycles during Pd-Catalyzed C–N Bond Formation with Catalysts Derived from Bulky Monophosphinobiaryl Ligands |
Angew. Chem. Int. Ed. |
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Combined C−H Functionalization/C−N Bond Formation Route to Carbazoles |
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Industrial-Scale Palladium-Catalyzed Coupling of Aryl Halides and Amines –A Personal Account |
Advanced Synthesis & Catalysis |
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Efficient Pd-Catalyzed Amination of Heteroaryl Halides |
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Synthesis of 4,5-Dianilinophthalimide and Related Analogues for Potential Treatment of Alzheimer's Disease via Palladium-Catalyzed Amination |
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General Catalysts for the Suzuki-Miyaura and Sonogashira Coupling Reactions of Aryl Chlorides and for the Coupling of Challenging Substrate Combinations in Water |
Angew. Chem. Int. Ed. |
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M.P. Rainka; J.E. Milne; S.L. Buchwald |
Dynamic Kinetic Resolution of α,β-Unsaturated Lactones through Asymmetric Copper-Catalyzed Conjugate Reduction: Application to the Total Synthesis of Eupomatilone-3 |
Angew. Chem. Int. Ed. |
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Use of Tunable Ligands Allows for Intermolecular Pd-Catalyzed C−O Bond Formation |
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The Role of Chelating Diamine Ligands in the Goldberg Reaction: A Kinetic Study on the Copper-Catalyzed Amidation of Aryl Iodides |
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Catalysts for Suzuki−Miyaura Coupling Processes: Scope and Studies of the Effect of Ligand Structure |
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One-Pot Sequential Cu-Catalyzed Reduction and Pd-Catalyzed Arylation of Silyl Enol Ethers |
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An extremely active catalyst for the Negishi cross-coupling reaction |
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Efficient Catalyst for the Suzuki−Miyaura Coupling of Potassium Aryl Trifluoroborates with Aryl Chlorides |
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Copper−Diamine-Catalyzed N-Arylation of Pyrroles, Pyrazoles, Indazoles, Imidazoles, and Triazoles |
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M. Murata; S.L. Buchwald |
A general and efficient method for the palladium-catalyzed cross-coupling of thiols and secondary phosphines |
Tetrahedron |
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M.P. Rainka; Y. Aye; S.L. Buchwald |
Copper-catalyzed asymmetric conjugate reduction as a route to novel β-azaheterocyclic acid derivatives |
Proceedings of the National Academy of Sciences of the United States of America |
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Palladium-Catalyzed Regioselective Hydrodebromination of Dibromoindoles: Application to the Enantioselective Synthesis of Indolodioxane U86192A |
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Synthesis of Medium Ring Nitrogen Heterocycles via a Tandem Copper-Catalyzed C−N Bond Formation−Ring-Expansion Process |
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A Rationally Designed Universal Catalyst for Suzuki–Miyaura Coupling Processes |
Angew. Chem. Int. Ed. |
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D. Gelman; S.L. Buchwald |
Efficient Palladium-Catalyzed Coupling of Aryl Chlorides and Tosylates with Terminal Alkynes: Use of a Copper Cocatalyst Inhibits the Reaction |
Angew. Chem. Int. Ed. |
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Insights into the Origin of High Activity and Stability of Catalysts Derived from Bulky, Electron-Rich Monophosphinobiaryl Ligands in the Pd-Catalyzed C−N Bond Formation |
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Palladium-Catalyzed Amination of Aryl Nonaflates |
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Copper-Catalyzed Coupling of Amides and Carbamates with Vinyl Halides |
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H.Nho Nguyen; X. Huang; S.L. Buchwald |
The First General Palladium Catalyst for the Suzuki−Miyaura and Carbonyl Enolate Coupling of Aryl Arenesulfonates |
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E.J. Hennessy; S.L. Buchwald |
Synthesis of Substituted Oxindoles from α-Chloroacetanilides via Palladium-Catalyzed C−H Functionalization |
J. Am. Chem. Soc. |
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C. Enguehard; H. Allouchi; A. Gueiffier; S.L. Buchwald |
Ipso- or Cine-Substitutions of 6-Haloimidazo[1,2-a]pyridine Derivatives with Different Azoles Depending on the Reaction Conditions |
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G. Hughes; M. Kimura; S.L. Buchwald |
Catalytic Enantioselective Conjugate Reduction of Lactones and Lactams |
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Conjugate Reduction of α,β-Unsaturated Carbonyl Compounds Catalyzed by a Copper Carbene Complex |
Org. Lett. |
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D. Zim; S.L. Buchwald |
An Air and Thermally Stable One- Component Catalyst for the Amination of Aryl Chlorides |
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D. Gelman; L. Jiang; S.L. Buchwald |
Copper-Catalyzed C−P Bond Construction via Direct Coupling of Secondary Phosphines and Phosphites with Aryl and Vinyl Halides |
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C. Enguehard; H. Allouchi; A. Gueiffier; S.L. Buchwald |
Easy Access to Novel Substituted 6-Aminoimidazo[1,2-a]pyridines Using Palladium- and Copper-Catalyzed Aminations |
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Expanding Pd-Catalyzed C−N Bond-Forming Processes: The First Amidation of Aryl Sulfonates, Aqueous Amination, and Complementarity with Cu-Catalyzed Reactions |
J. Am. Chem. Soc. |
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G. Nordmann; S.L. Buchwald |
A Domino Copper-Catalyzed C−O Coupling−Claisen Rearrangement Process |
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J. Zanon; A. Klapars; S.L. Buchwald |
Copper-Catalyzed Domino Halide Exchange-Cyanation of Aryl Bromides |
J. Am. Chem. Soc. |
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Mild and Efficient Copper-Catalyzed Amination of Aryl Bromides with Primary Alkylamines |
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J.L. Rutherford; M.P. Rainka; S.L. Buchwald |
An Annulative Approach to Highly Substituted Indoles: Unusual Effect of Phenolic Additives on the Success of the Arylation of Ketone Enolates |
J. Am. Chem. Soc. |
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Copper-Catalyzed Halogen Exchange in Aryl Halides: An Aromatic Finkelstein Reaction |
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G.E. Job; S.L. Buchwald |
Copper-Catalyzed Arylation of β-Amino Alcohols |
Org. Lett. |
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A General, Efficient, and Inexpensive Catalyst System for the Coupling of Aryl Iodides and Thiols |
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U.K. Singh; E.R. Strieter; D.G. Blackmond; S.L. Buchwald |
Mechanistic Insights into the Pd(BINAP)-Catalyzed Amination of Aryl Bromides: Kinetic Studies under Synthetically Relevant Conditions |
J. Am. Chem. Soc. |
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The Copper-Catalyzed N-Arylation of Indoles |
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Preparation, Crystal Structure Analysis, and Catalytic Application of [(S)-BINAP]Ni(COD) and [(S)-BINAP]NiBr2 |
Organometallics |
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M.C. Harris; X. Huang; S.L. Buchwald |
Improved Functional Group Compatibility in the Palladium-Catalyzed Synthesis of Aryl Amines |
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A General and Efficient Copper Catalyst for the Amidation of Aryl Halides |
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Pd-Catalyzed Intermolecular Amidation of Aryl Halides: The Discovery that Xantphos Can Be Trans-Chelating in a Palladium Complex |
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S.J. Sturla; S.L. Buchwald |
Cobalt−Phosphite-Catalyzed Asymmetric Pauson−Khand Reaction |
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Nickel-BINAP Catalyzed Enantioselective α-Arylation of α-Substituted γ-Butyrolactones |
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Dynamic Kinetic Resolution via Asymmetric Conjugate Reduction: Enantio- and Diastereoselective Synthesis of 2,4-Dialkyl Cyclopentanones |
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P-Chirogenic Binaphthyl-Substituted Monophosphines: Synthesis and Use in Enolate Vinylation/Arylation Reactions |
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Copper-Catalyzed Coupling of Aryl Iodides with Aliphatic Alcohols |
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Copper-Catalyzed Coupling of Alkylamines and Aryl Iodides: An Efficient System Even in an Air Atmosphere |
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E.J. Hennessy; S.L. Buchwald |
A General and Mild Copper-Catalyzed Arylation of Diethyl Malonate |
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A highly active Suzuki catalyst for the synthesis of sterically hindered biaryls: novel ligand coordination |
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S.J. Sturla; S.L. Buchwald |
Monocyclopentadienyltitanium Aryloxide Complexes: Preparation, Characterization, and Application in Cyclization Reactions |
Organometallics |
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O. Gaertzen; S.L. Buchwald |
Palladium-Catalyzed Intramolecular α-Arylation of α-Amino Acid Esters |
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T. Hamada; A. Chieffi; J.Å. hman; S.L. Buchwald |
An Improved Catalyst for the Asymmetric Arylation of Ketone Enolates |
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Palladium-Catalyzed Intramolecular C−O Bond Formation |
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Palladium-Catalyzed Monoarylation of Nitroalkanes |
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Synthesis of N-Aryl Hydrazides by Copper-Catalyzed Coupling of Hydrazides with Aryl Iodides |
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New Ammonia Equivalents for the Pd-Catalyzed Amination of Aryl Halides |
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An Efficient Intermolecular Palladium-Catalyzed Synthesis of Aryl Ethers |
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S. Kaye; J.M. Fox; F.A. Hicks; S.L. Buchwald |
The Use of Catalytic Amounts of CuCl and Other Improvements in the Benzyne Route to Biphenyl-Based Phosphine Ligands |
Advanced Synthesis & Catalysis |
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J.P. Wolfe; S.L. Buchwald |
Palladium-Catalyzed Amination of Aryl Halides and Aryl Triflates: N-Hexyl-2-methyl-4-methoxy Aniline and N-Methyl-N-(4-chlorophenyl) Aniline |
Org. Syn. |
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A General and Efficient Copper Catalyst for the Amidation of Aryl Halides and the N-Arylation of Nitrogen Heterocycles |
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W.A. Moradi; S.L. Buchwald |
Palladium-Catalyzed α-Arylation of Esters |
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The use of palladium chloride as a precatalyst for the amination of aryl bromides |
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Copper-Catalyzed Coupling of Arylboronic Acids and Amines |
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Catalytic Asymmetric Vinylation of Ketone Enolates |
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Use of Polymer-Supported Dialkylphosphinobiphenyl Ligands for Palladium-Catalyzed Amination and Suzuki Reactions |
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One-Pot Synthesis of Enantiomerically Enriched 2,3-Disubstituted Cyclopentanones via Copper-Catalyzed 1,4-Reduction and Alkylation |
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Palladium-Catalyzed Formation of Aryl tert-Butyl Ethers from Unactivated Aryl Halides |
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M.H. Ali; S.L. Buchwald |
An Improved Method for the Palladium-Catalyzed Amination of Aryl Iodides |
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A High-Yield, General Method for the Catalytic Formation of Oxygen Heterocycles |
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A Catalytic Asymmetric Suzuki Coupling for the Synthesis of Axially Chiral Biaryl Compounds |
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Efficient Synthesis of N-Aryl-Aza-Crown Ethers via Palladium-Catalyzed Amination |
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An Improved Synthesis of Functionalized Biphenyl-Based Phosphine Ligands |
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Efficient Synthesis of Well-Defined, High Molecular Weight, and Processible Polyanilines under Mild Conditions via Palladium-Catalyzed Amination |
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Synthesis of β-Alkyl Cyclopentanones in High Enantiomeric Excess via Copper-Catalyzed Asymmetric Conjugate Reduction |
J. Am. Chem. Soc. |
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O.J. Plante; S.L. Buchwald; P.H. Seeberger |
Halobenzyl Ethers as Protecting Groups for Organic Synthesis |
J. Am. Chem. Soc. |
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One-Pot Synthesis of Unsymmetrical Triarylamines from Aniline Precursors |
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T. Hundertmark; A.F. Littke; S.L. Buchwald; G.C. Fu |
Pd(PhCN)2Cl2/P(t-Bu)3: A Versatile Catalyst for Sonogashira Reactions of Aryl Bromides at Room Temperature |
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Palladium-Catalyzed Intermolecular Coupling of Aryl Halides and Amides |
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A method for the asymmetric hydrosilylation of N-aryl imines |
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Kinetic resolution and isomerization of 2,5-disubstituted pyrrolines |
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Highly Active and Selective Catalysts for the Formation of α-Aryl Ketones |
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Efficient Kinetic Resolution in the Asymmetric Hydrosilylation of Imines of 3-Substituted Indanones and 4-Substituted Tetralones |
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A Combined Zirconocene Benzyne−Palladium Cross-Coupling Route to Substituted Biphenyls and Terphenyls |
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Highly Active Palladium Catalysts for Suzuki Coupling Reactions |
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A phosphane-free catalyst system for the Heck arylation of disubstituted alkenes: Application to the synthesis of trisubstituted olefins |
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An Intramolecular Titanium-Catalyzed Asymmetric Pauson−Khand Type Reaction |
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A Highly Active Catalyst for the Room-Temperature Amination and Suzuki Coupling of Aryl Chlorides |
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Catalytic Asymmetric Cyclocarbonylation of Nitrogen-Containing Enynes |
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Titanocene-catalyzed asymmetric ketone hydrosilylation: The effect of catalyst activation protocol and additives on the reaction rate and enantioselectivity |
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Asymmetric Hydrogenation of Unfunctionalized Tetrasubstituted Olefins with a Cationic Zirconocene Catalyst |
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An efficient copper-catalyzed coupling of aryl halides with imidazoles |
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Synthesis of NPS R-568 utilizing titanium-catalyzed asymmetric hydrosilylation |
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144 |
R. Singer; S. Buchwald |
Preparation of 2-amino-2′-hydroxy-1,1′-binaphthyl and N-arylated 2-amino-1,1′-binaphthyl derivatives via palladium-catalyzed amination |
Tet. Lett. |
1999 |
Link |
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143 |
B. Yang; S. Buchwald |
Palladium-Catalyzed Amination of Aryl Halides and Sulfonates |
J. Organomet. Chem. |
1999 |
Link |
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142 |
D.W. Old; J.P. Wolfe; S.L. Buchwald |
A Highly Active Catalyst for Palladium-Catalyzed Cross-Coupling Reactions: Room-Temperature Suzuki Couplings and Amination of Unactivated Aryl Chlorides |
J. Am. Chem. Soc. |
1998 |
Link |
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141 |
S. Akai; A.J. Peat; S.L. Buchwald |
Regioselective, directed meta acylation of aromatic compounds |
J. Am. Chem. Soc. |
1998 |
Link |
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140 |
J.P. Wolfe; S. Wagaw; J.F. Marcoux; S.L. Buchwald |
Rational Development of Practical Catalysts for Aromatic Carbon−Nitrogen Bond Formation |
Acc. Chem. Res. |
1998 |
Link |
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139 |
M.T. Reding; S.L. Buchwald |
Short Enantioselective Total Syntheses of the Piperidine Alkaloids (S)-Coniine and (2R,6R)-trans-Solenopsin A via Catalytic Asymmetric Imine Hydrosilylation |
J. Org. Chem. |
1998 |
Link |
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138 |
S. Wagaw; B.H. Yang; S.L. Buchwald |
A palladium-catalyzed strategy for the preparation of indoles: A novel entry into the Fischer indole synthesis |
J. Am. Chem. Soc. |
1998 |
Link |
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137 |
J.P. Sadighi; M.C. Harris; S.L. Buchwald |
A highly active palladium catalyst system for the arylation of anilines |
Tet. Lett. |
1998 |
Link |
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136 |
R.A. Widenhoefer; S.L. Buchwald |
Electronic Dependence of C−O Reductive Elimination from Palladium (Aryl)neopentoxide Complexes |
J. Am. Chem. Soc. |
1998 |
Link |
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135 |
J.P. Sadighi; R.A. Singer; S.L. Buchwald |
Palladium-catalyzed synthesis of monodisperse, controlled-length, and functionalized oligoanilines |
J. Am. Chem. Soc. |
1998 |
Link |
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134 |
J. Ahman; J.P. Wolfe; M.V. Troutman; M. Palucki; S.L. Buchwald |
Asymmetric arylation of ketone enolates |
J. Am. Chem. Soc. |
1998 |
Link |
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133 |
X. Verdaguer; U.E.W. Lange; S.L. Buchwald |
Amine additives greatly expand the scope of asymmetric hydrosilylation of imines |
Angew. Chem. Int. Ed. |
1998 |
Link |
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132 |
M.C. Hansen; X. Verdaguer; S.L. Buchwald |
Convenient two-step conversion of lactones into cyclic ethers |
J. Org. Chem. |
1998 |
Link |
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131 |
K. Aoki; A.J. Peat; S.L. Buchwald |
Titanocene-based method for indole synthesis |
J. Am. Chem. Soc. |
1998 |
Link |
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130 |
R.A. Singer; J.P. Sadighi; S.L. Buchwald |
A general synthesis of end-functionalized oligoanilines via palladium-catalyzed amination |
J. Am. Chem. Soc. |
1998 |
Link |
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129 |
M. Palucki; S.L. Buchwald |
Palladium-catalyzed alpha-arylation of ketones |
J. Am. Chem. Soc. |
1997 |
Link |
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128 |
X. Verdaguer; M.C. Hansen; S.C. Berk; S.L. Buchwald |
Titanocene-Catalyzed Reduction of Lactones to Lactols |
J. Org. Chem. |
1997 |
Link |
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127 |
J.F. Marcoux; S. Doye; S.L. Buchwald |
A general copper-catalyzed synthesis of diaryl ethers |
J. Am. Chem. Soc. |
1997 |
Link |
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126 |
J.P. Wolfe; J. Ahman; J.P. Sadighi; R.A. Singer; S.L. Buchwald |
An ammonia equivalent for the palladium-catalyzed amination of aryl halides and triflates |
Tet. Lett. |
1997 |
Link |
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125 |
J.Å. hman; S.L. Buchwald |
An Improved Method for the Palladium-Catalyzed Amination of Aryl Triflates |
Tet. Lett. |
1997 |
Link |
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124 |
J.P. Wolfe; S.L. Buchwald |
Improved functional group compatibility in the palladium-catalyzed amination of aryl bromides |
Tet. Lett. |
1997 |
Link |
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123 |
S. Wagaw; R.A. Rennels; S.L. Buchwald |
Palladium-Catalyzed Coupling of Optically Active Amines with Aryl Bromides |
J. Am. Chem. Soc. |
1997 |
Link |
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122 |
J.P. Wolfe; S.L. Buchwald |
Room temperature catalytic amination of aryl iodides |
J. Org. Chem. |
1997 |
Link |
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121 |
J.P. Wolfe; S.L. Buchwald |
Nickel-Catalyzed Amination of Aryl Chlorides |
J. Am .Chem .Soc. |
1997 |
Link |
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120 |
R.A. Widenhoefer; H.A. Zhong; S.L. Buchwald |
Direct observation of C-O reductive elimination from palladium aryl alkoxide complexes to form aryl ethers |
J. Am. Chem. Soc. |
1997 |
Link |
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119 |
N.M. Kablaoui; F.A. Hicks; S.L. Buchwald |
Titanocene-catalyzed cyclocarbonylation of o-allyl aryl ketones to gamma-butyrolactones |
J. Am. Chem. Soc. |
1997 |
Link |
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118 |
M. Palucki; J.P. Wolfe; S.L. Buchwald |
Palladium-catalyzed intermolecular carbon-oxygen bond formation: A new synthesis of aryl ethers |
J. Am. Chem. Soc. |
1997 |
Link |
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117 |
J.F. Marcoux; S. Wagaw; S.L. Buchwald |
Palladium-catalyzed amination of aryl bromides: Use of phosphinoether ligands for the efficient coupling of acyclic secondary amines |
J. Org. Chem. |
1997 |
Link |
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116 |
J.P. Wolfe; S.L. Buchwald |
Palladium-Catalyzed Amination of Aryl Triflates |
J. Org. Chem. |
1997 |
Link |
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115 |
B. Chin; S.L. Buchwald |
Improved Procedure for the Preparation of Enantiomerically Pure Ethylenebis(tetrahydroindenyl)zirconium Derivatives |
J. Org. Chem. |
1997 |
Link |
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114 |
F.A. Hicks; S.L. Buchwald |
Highly enantioselective catalytic Pauson-Khand type formation of bicyclic cyclopentenones |
J. Am. Chem. Soc. |
1996 |
Link |
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113 |
M. Palucki; J.P. Wolfe; S.L. Buchwald |
Synthesis of oxygen heterocycles via a palladium-catalyzed C-O bond-forming reaction |
J. Am. Chem. Soc. |
1996 |
Link |
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112 |
F.A. Hicks; N.M. Kablaoui; S.L. Buchwald |
Titanocene-catalyzed cyclocarbonylation of enynes to cyclopentenones |
J. Am. Chem. Soc. |
1996 |
Link |
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111 |
S. Wagaw; S.L. Buchwald |
The Synthesis of Aminopyridines: A Method Employing Palladium-Catalyzed Carbon-Nitrogen Bond Formation |
J. Org. Chem. |
1996 |
Link |
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110 |
N.S. Radu; S.L. Buchwald; B. Scott; C.J. Burns |
Carbon-hydrogen bond activation of aromatic imines by(Cp*2SmH)(2) |
Organometallics |
1996 |
Link |
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109 |
J.P. Wolfe; S. Wagaw; S.L. Buchwald |
An improved catalyst system for aromatic carbon-nitrogen bond formation: The possible involvement of bis(phosphine) palladium complexes as key intermediates |
J. Am. Chem. Soc. |
1996 |
Link |
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108 |
R.A. Widenhoefer; S.L. Buchwald |
Formation of palladium bis(amine) complexes from reaction of amine with palladium tris(o-tolyl)phosphine mono(amine) complexes |
Organometallics |
1996 |
Link |
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107 |
B. Chin; S.L. Buchwald |
An improved procedure for the resolution of (rac)-ethylenebis(tetrahydroindenyl)-titanium derivatives |
J. Org. Chem. |
1996 |
Link |
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106 |
X. Verdaguer; U.E.W. Lange; M.T. Reding; S.L. Buchwald |
Highly enantioselective imine hydrosilylation using (S,S)-ethylenebis(eta(5)-tetrahydroindenyl)titanium difluoride |
J. Am. Chem. Soc. |
1996 |
Link |
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105 |
M. Zhang; S.L. Buchwald |
A Nickel(0)-Catalyzed Process for the Transformation of Enynes to Bicyclic Cyclopentenones |
J. Org. Chem. |
1996 |
Link |
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104 |
S. Bower; K.A. Kreutzer; S.L. Buchwald |
A mild general procedure for the one-pot conversion of amides to aldehydes |
Angew. Chem. Int. Ed. |
1996 |
Link |
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103 |
N.M. Kablaoui; F.A. Hicks; S.L. Buchwald |
Diastereoselective synthesis of gamma-butyrolactones from enones mediated or catalyzed by a titanocene complex |
J. Am. Chem. Soc. |
1996 |
Link |
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102 |
R.A. Widenhoefer; S.L. Buchwald |
Halide and Amine Influence in the Equilibrium Formation of Palladium Tris(o-tolyl)phosphine Mono(amine) Complexes from Palladium Aryl Halide Dimers |
Organometallics |
1996 |
Link |
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101 |
R.A. Widenhoefer; H.A. Zhong; S.L. Buchwald |
Synthesis and solution structure of palladium tris(o-tolyl)phosphine mono(amine) complexes |
Organometallics |
1996 |
Link |
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100 |
N.M. Kablaoui; S.L. Buchwald |
Development of a method for the reductive cyclization of enones by a titanium catalyst |
J. Am. Chem. Soc. |
1996 |
Link |
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99 |
F.A. Hicks; S.C. Berk; S.L. Buchwald |
A Practical Titanium-Catalyzed Synthesis of Bicyclic Cyclopentenones and Allylic Amines |
J. Org. Chem. |
1996 |
Link |
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98 |
J.P. Wolfe; R.A. Rennels; S.L. Buchwald |
Intramolecular palladium-catalyzed aryl amination and aryl amidation |
Tetrahedron |
1996 |
Link |
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97 |
A.J. Peat; S.L. Buchwald |
Novel syntheses of tetrahydropyrroloquinolines: Applications to alkaloid synthesis |
J. Am. Chem. Soc. |
1996 |
Link |
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96 |
J.P. Wolfe; S.L. Buchwald |
Palladium-catalyzed amination of aryl iodides |
J. Org. Chem. |
1996 |
Link |
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95 |
X. Verdaguer; S.C. Berk; S.L. Buchwald |
Catalytic method for the reduction of lactones to lactols |
J. Am. Chem. Soc. |
1995 |
Link |
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94 |
C.A. Willoughby; R.R. Duff; W.M. Davis; S.L. Buchwald |
Preparation of novel titanium complexes bearing o-phosphinophenol ligands |
Organometallics |
1996 |
Link |
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93 |
M.T. Reding; S.L. Buchwald |
An Inexpensive Air-Stable Titanium-Based System for the Conversion of Esters to Primary Alcohols |
J. Org. Chem. |
1995 |
Link |
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92 |
F.M.G. Derege; W.M. Davis; S.L. Buchwald |
Synthesis and Structure of Zirconium Group-13 Heterobimetallic Compounds |
Organometallics |
1995 |
Link |
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91 |
B.P. Warner; S.P. Millar; R.D. Broene; S.L. Buchwald |
Controlled acceleration and inhibition of bergman cyclization by metal chlorides |
Science |
1995 |
Link |
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90 |
J.R. Johnson; G.D. Cuny; S.L. Buchwald |
Rhodium-Catalyzed Hydroformylation of Internal Alkynes to α,β-Unsaturated Aldehydes |
Angew. Chem. Int. Ed. |
1995 |
Link |
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89 |
N.M. Kablaoui; S.L. Buchwald |
Reductive Cyclization of Enones by a Titanium Catalyst |
J. Am. Chem. Soc. |
1995 |
Link |
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88 |
A.S. Guram; R.A. Rennels; S.L. Buchwald |
A Simple Catalytic Method for the Conversion of Aryl Bromides to Arylamines |
Angew. Chem. Int. Ed. |
1995 |
Link |
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87 |
G.D. Cuny; S.L. Buchwald |
Regioselective Olefin Hydroformylation as a Route to Indolizidine and Pyrrolizidine Alkaloids |
Synlett |
1995 |
Link |
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86 |
C.A. Willoughby; W.M. Davis; S.L. Buchwald |
Preparation and X-ray structure of a novel chiral methylene bridged titanocene complex |
J. Organomet. Chem. |
1995 |
Link |
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85 |
J. Campora; S.L. Buchwald; E. Gutierrez-Puebla; A. Monge |
Kinetics and Mechanism of the Reductive Elimination of Cyclic Titanocene Iminoacyls |
Organometallics |
1995 |
Link |
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84 |
F.M.G. de Rege; S.L. Buchwald |
The regioselective synthesis of halophenols |
Tetrahedron |
1995 |
Link |
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83 |
C.A. Willoughby; S.L. Buchwald |
Catalytic Asymmetric Hydrogenation of Imines with a Chiral Titanocene Catalyst: Kinetic and Mechanistic Investigations |
J. Am. Chem. Soc. |
1994 |
Link |
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82 |
J.H. Tidwell; S.L. Buchwald |
Synthesis of Polysubstituted Indoles and Indolines by Means of Zirconocene-Stabilized Benzyne Complexes |
J. Am. Chem. Soc. |
1994 |
Link |
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81 |
J.H. Tidwell; A.J. Peat; S.L. Buchwald |
Synthesis and Reactions of 3-(Bromomethyl)-1-carbethoxy-4-iodoindole: The Preparation of 3,4-Differentially Substituted Indoles |
J. Org. Chem. |
1994 |
Link |
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80 |
E. Spaltenstein; P. Palma; K.A. Kreutzer; C.A. Willoughby; W.M. Davis; S.L. Buchwald |
Preparation and X-ray Structure of Cp2Ti(Ph2SiH2)(PMe3) |
J. Am. Chem. Soc. |
1994 |
Link |
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79 |
M.Beth Carter; B. Schiott; A. Gutierrez; S.L. Buchwald |
Enantioselective Hydrosilylation of Ketones with a Chiral Titanocene Catalyst |
J. Am. Chem. Soc. |
1994 |
Link |
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78 |
A. Viso; N.E. Lee; S.L. Buchwald |
Kinetic resolution of racemic disubstituted 1-pyrrolines via asymmetric reduction with a chiral titanocene catalyst |
J. Am. Chem. Soc. |
1994 |
Link |
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77 |
D.P. Hsu; B.P. Warner; R.A. Fisher; W.M. Davis; S.L. Buchwald |
Synthesis and Structure of a Novel Bis(stibole) |
Organometallics |
1994 |
Link |
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76 |
C.A. Willoughby; S.L. Buchwald |
Catalytic Asymmetric Hydrogenation of Imines with a Chiral Titanocene Catalyst: Scope and Limitations |
J. Am. Chem. Soc. |
1994 |
Link |
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75 |
B.P. Warner; S.L. Buchwald |
A Catalytic Method for the Conversion of Silanes to Stannanes |
J. Org. Chem. |
1994 |
Link |
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74 |
S.C. Berk; R.B. Grossman; S.L. Buchwald |
Development of a Titanocene-Catalyzed Enyne Cyclization/Isocyanide Insertion Reaction |
J. Am. Chem. Soc. |
1994 |
Link |
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73 |
A.F. England; C.J. Burns; S.L. Buchwald |
New Syntheses of Cp*2Th(Ph)2 and Cp*2Th(Me)(aryl) Derivatives |
Organometallics |
1994 |
Link |
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72 |
R.B. Grossman; J.C. Tsai; W.M. Davis; A. Gutierrez; S.L. Buchwald |
Synthesis and Structure of a C2-Symmetric, Doubly Bridged ansa-Titanocene Complex |
Organometallics |
1994 |
Link |
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71 |
A.S. Guram; S.L. Buchwald |
Palladium-Catalyzed Aromatic Aminations with in situ Generated Aminostannanes |
J. Am. Chem. Soc. |
1994 |
Link |
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70 |
K.J. Barr; S.C. Berk; S.L. Buchwald |
Titanocene-Catalyzed Reduction of Esters Using Polymethylhydrosiloxane as the Stoichiometric Reductant |
J. Org. Chem. |
1994 |
Link |
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69 |
N.E. Lee; S.L. Buchwald |
Asymmetric Hydrogenation of Enamines with a Chiral Titanocene Catalyst |
J. Am. Chem. Soc. |
1994 |
Link |
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68 |
B.P. Warner; W.M. Davis; S.L. Buchwald |
Synthesis and X-ray Structure of a Zirconocene Complex of Two Alkynes |
J. Am. Chem. Soc. |
1994 |
Link |
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67 |
C.A. Willoughby; S.L. Buchwald |
Synthesis of highly enantiomerically enriched cyclic amines by the catalytic asymmetric hydrogenation of cyclic imines |
J. Org. Chem. |
1993 |
Link |
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66 |
R.D. Broene; S.L. Buchwald |
Asymmetric hydrogenation of unfunctionalized trisubstituted olefins with a chiral titanocene catalyst |
J. Am. Chem. Soc. |
1993 |
Link |
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65 |
D.P. Hsu; W.M. Davis; S.L. Buchwald |
Synthesis and structure of seven-membered cyclic cumulene |
J. Am. Chem. Soc. |
1993 |
Link |
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64 |
J. Campora; S.L. Buchwald |
Synthesis and reactivity of a titanocene-benzyne complex |
Organometallics |
1993 |
Link |
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63 |
R.D. Broene; S.L. Buchwald |
Zirconocene complexes of unsaturated organic molecules: new vehicles for organic synthesis |
Science |
1993 |
Link |
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62 |
S.C. Berk; R.B. Grossman; S.L. Buchwald |
Titanocene-catalyzed conversion of enynes to bicyclic cyclopentenones |
J. Am. Chem. Soc. |
1993 |
Link |
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61 |
J.H. Tidwell; S.L. Buchwald |
A new approach to the synthesis of the CC-1065/duocarmycin pharmacophore |
J. Org. Chem. |
1992 |
Link |
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60 |
G.D. Cuny; S.L. Buchwald |
Practical, high-yield, regioselective, rhodium-catalyzed hydroformylation of functionalized .alpha.-olefins |
J. Am. Chem. Soc. |
1993 |
Link |
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59 |
R.B. Grossman; S.L. Buchwald |
Reductive cyclization of ester-containing enynes with a practical titanocene reagent. Synthesis of bicyclic cyclopentenones and iminocyclopentenes |
J. Org. Chem. |
1992 |
Link |
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58 |
C.A. Willoughby; S.L. Buchwald |
Asymmetric titanocene-catalyzed hydrogenation of imines |
J. Am. Chem. Soc. |
1992 |
Link |
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57 |
R.E. v H. Spence; D.P. Hsu; S.L. Buchwald |
Synthesis of thermochromic dibismuthines with nonthermochromic distibine analogs |
Organometallics |
1992 |
Link |
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56 |
R.E. v H. Spence; S.L. Buchwald; J.F. Richardson |
The Unexpected Formation of 3,4,7,8-Tetramethyl-1,2,5,6-tetrahydrodicyclobuta[a, e]cyclooctene from a Zirconacyclopentadiene |
Acta Chem. Scand. |
1993 |
Link |
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55 |
S.C. Berk; S.L. Buchwald |
An air-stable catalyst system for the conversion of esters to alcohols |
J. Org. Chem. |
1992 |
Link |
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54 |
K.J. Barr; B.T. Watson; S.L. Buchwald |
Zirconocene(iso-butyl) chloride: In situ generation of a zirconocene(methyl) chloride equivalent for use in organic synthesis |
Tet. Lett. |
1991 |
Link |
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53 |
S.C. Berk; K.A. Kreutzer; S.L. Buchwald |
A catalytic method for the reduction of esters to alcohols |
J. Am. Chem. Soc. |
1991 |
Link |
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52 |
J.H. Tidwell; D.R. Senn; S.L. Buchwald |
Synthesis of 3,4-disubstituted indoles via a sequential olefin-insertion/ene route |
J. Am. Chem. Soc. |
1991 |
Link |
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51 |
S.L. Buchwald; S.J. LaMaire; R.B. Nielsen; B.T. Watson; S.M. King |
Schwartz's Reagent |
Org. Synth. |
1993 |
Link |
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50 |
K.A. Kreutzer; R.A. Fisher; W.M. Davis; E. Spaltenstein; S.L. Buchwald |
Synthesis, characterization, and reactivity of zirconocene and hafnocene silyl hydride complexes |
Organometallics |
1991 |
Link |
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49 |
G.D. Cuny; A. Gutierrez; S.L. Buchwald |
Cis difunctionalization of cyclic olefins with use of organozirconium intermediates |
Organometallics |
1991 |
Link |
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48 |
R.B. Grossman; W.M. Davis; S.L. Buchwald |
Enantioselective, zirconium-mediated synthesis of allylic amines |
J. Am. Chem. Soc. |
1991 |
Link |
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47 |
R.B. Grossman; R.Ann Doyle; S.L. Buchwald |
Syntheses of [ethylene-1,2-bis(.eta.5-4,5,6,7-tetrahydro-1-indenyl)]zirconium and -hafnium hydride complexes. Improved syntheses of the corresponding dichlorides |
Organometallics |
1991 |
Link |
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46 |
R.A. Fisher; R.B. Nielsen; W.M. Davis; S.L. Buchwald |
Stibathiolanes: synthesis, solid-state structure, and solution behavior |
J. Am. Chem. Soc. |
1991 |
Link |
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45 |
S.L. Buchwald; S.M. King |
The regiospecific synthesis of polysubstituted naphthalenes and iodo(acyl)naphthoquinones via zirconocene complexes of naphthalynes |
J. Am. Chem. Soc. |
1991 |
Link |
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44 |
G.D. Cuny; S.L. Buchwald |
Ring-opening reactions of cyclic allylic ethers by zirconocene complexes of cyclic alkynes |
Organometallics |
1991 |
Link |
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43 |
D.P. Hsu; E.A. Lucas; S.L. Buchwald |
Synthesis and reactions of a zirconocene-benzdiyne equivalent |
Tet. Lett. |
1990 |
Link |
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42 |
S.L. Buchwald; R.A. Fisher; B.M. Foxman |
The Synthesis and Structure of Stibaindoles |
Angew. Chem. Int. Ed. |
1990 |
Link |
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41 |
R.A. Fisher; S.L. Buchwald |
Synthesis, structure, and reactivity of a zirconocene complex of cyclobutene |
Organometallics |
1990 |
Link |
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40 |
S.L. Buchwald; K.A. Kreutzer; R.A. Fisher |
Synthesis, reactions, and x-ray crystal structure determination of hafnocene complex Cp2Hf(isobutylene).cntdot.PMe3 |
J. Am. Chem. Soc. |
1990 |
Link |
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39 |
S.L. Buchwald; R.A. Fisher |
Zirconocene Complexes of Unsaturated Organic Molecules |
Chemica Scripta |
1989 |
Link |
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38 |
S.L. Buchwald; R.T. Lum; R.A. Fisher; W.M. Davis |
Synthesis and x-ray crystal structure of a zirconocene complex of a cyclopentyne and its use to prepare bicyclic cyclopentenones |
J. Am. Chem. Soc. |
1989 |
Link |
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37 |
S.L. Buchwald; R.A. Fisher; W.M. Davis |
Synthesis and structure of novel antimony thiametallacycles |
Organometallics |
1989 |
Link |
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36 |
S.L. Buchwald; Q. Fang |
An efficient one-pot method for the preparation of polysubstituted benzothiophenes |
J. Org. Chem. |
1989 |
Link |
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35 |
S.L. Buchwald; R.B. Nielsen; J.C. Dewan |
Synthesis of (alkoxymethyl)zirconocene chlorides: stereochemistry of carbon-carbon bond formation in a zirconocene-Wittig rearrangement |
Organometallics |
1989 |
Link |
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34 |
S.L. Buchwald; B.T. Watson; W. Wannamaker; J.C. Dewan |
Zirconocene complexes of imines. General synthesis, structure, reactivity, and in situ generation to prepare geometrically pure allylic amines |
J. Am. Chem. Soc. |
1989 |
Link |
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33 |
S.L. Buchwald; E.A. Lucas; W.M. Davis |
A bimetallic zirconium complex containing an in-plane bridging aromatic ring |
J. Am. Chem. Soc. |
1989 |
Link |
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32 |
S.L. Buchwald; R.B. Nielsen |
Selective, zirconium-mediated cross-coupling of alkynes: the synthesis of isomerically pure 1,3-dienes and 1,4-diiodo-1,3-dienes |
J. Am. Chem. Soc. |
1989 |
Link |
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31 |
S.L. Buchwald; W. Wannamaker; B.T. Watson |
Synthesis of substituted pyrroles via zirconocene complexes of imines |
J. Am. Chem. Soc. |
1989 |
Link |
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30 |
A. Vaughan; G.L. Hillhouse; R.T. Lum; S.L. Buchwald; A.L. Rheingold |
Oxygen-atom transfer from nitrous oxide. Synthesis and structure of a zirconocene oxametallacyclobutene complex |
J. Am. Chem. Soc. |
1988 |
Link |
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29 |
S.L. Buchwald; R.B. Nielsen |
Group 4 metal complexes of benzynes, cycloalkynes, acyclic alkynes, and alkenes |
Chemical Reviews |
1988 |
Link |
|
28 |
S.L. Buchwald; Q. Fang; S.M. King |
A new method for the preparation of 3,5-disubstituted butenolides |
Tet. Lett. |
1988 |
Link |
|
27 |
S.L. Buchwald; R.B. Nielsen; J.C. Dewan |
Synthesis, structure, and reactions of (1-ethoxyethyl)zirconocene chloride, a stable acyclic secondary zirconocene alkyl |
Organometallics |
1988 |
Link |
|
26 |
S.L. Buchwald; R.B. Nielsen |
Kinetics and substituent effects in the formation of zirconocene thioaldehyde complexes: .beta.-hydride elimination versus cyclometalation |
J. Am. Chem. Soc. |
1988 |
Link |
|
25 |
S.L. Buchwald; B.T. Watson; R.T. Lum; W.A. Nugent |
A general method for the preparation of zirconocene complexes of substituted benzynes: in situ generation, coupling reactions, and use in the synthesis of polyfunctionalized aromatic compounds |
J. Am. Chem. Soc. |
1987 |
Link |
|
24 |
S.L. Buchwald; S.J. LaMaire; R.B. Nielsen; B.T. Watson; S.M. King |
A Modified Procedure for the Preparation of Cp2Zr(H)Cl (Schwartz's Reagent) |
Tet. Lett. |
1987 |
Link |
|
23 |
J.C. Dewan; E.A. Lucas; S.L. Buchwald |
Synthesis, structure, and reactions of a zirconocene-benzdiyne complex |
J. Am. Chem. Soc. |
1987 |
Link |
|
22 |
S.L. Buchwald; A. Sayers; B.T. Watson; J.C. Dewan |
The zirconocene induced coupling of benzyne with nitriles: Synthesis, structure and reactions of novel azametallacyclopentenes |
Tet. Lett. |
1987 |
Link |
|
21 |
S.L. Buchwald; B.T. Watson; J.C. Huffman |
The synthesis, reactions and molecular structure of zirconocene-alkyne complexes |
J. Am. Chem. Soc. |
1987 |
Link |
|
20 |
S.L. Buchwald; R.B. Nielsen; J.C. Dewan |
The synthesis, structure and reactivity of trimethylphosphine-zirconocene thioaldehyde complexes |
J. Am. Chem. Soc. |
1987 |
Link |
|
19 |
S.L. Buchwald; S.J. LaMaire |
A regiospecific method for the hydrocyanation of olefins |
Tet. Lett. |
1987 |
Link |
|
18 |
S.L. Buchwald; R.T. Lum; J.C. Dewan |
Synthesis, structure, and reactions of a zirconocene-cyclohexyne complex |
J. Am. Chem. Soc. |
1986 |
Link |
|
17 |
S.L. Buchwald; B.T. Watson; J.C. Huffman |
Trimethylphosphine adduct of the zirconocene-benzyne complex: synthesis, reactions, and x-ray crystal structure |
J. Am. Chem. Soc. |
1986 |
Link |
|
16 |
L. Clawson; J. Soto; S.L. Buchwald; M.L. Steigerwald; R.H. Grubbs |
Olefin insertion in a metal alkyl in a Ziegler polymerization system |
J. Am. Chem. Soc. |
1985 |
Link |
|
15 |
S.L. Buchwald; E.V. Anslyn; R.H. Grubbs |
Reaction of dicyclopentadienylmethylenetitanium with organic halides: Evidence for a radical mechanism |
J. Am. Chem. Soc. |
1985 |
Link |
|
14 |
L. Clawson; S.L. Buchwald; R.H. Grubbs |
The methylenation of enolizable ketones and esters using organotitanium chemistry |
Tet. Lett. |
1984 |
Link |
|
13 |
S.L. Buchwald; M.S. Saini; J.R. Knowles; R.L. Van Etten |
Stereochemical course of phospho group transfer by human prostatic acid phosphatase |
J. Biol. Chem. |
1984 |
|
|
12 |
S.L. Buchwald; D.H. Pliura; J.R. Knowles |
Stereochemical evidence for pseudorotation in the reaction of a phosphoric monoester |
J. Am. Chem. Soc. |
1984 |
Link |
|
11 |
S.L. Buchwald; J.M. Friedman; J.R. Knowles |
Stereochemistry of nucleophilic displacement on two phosphoric monoesters and a phosphoguanidine: the role of metaphosphate |
J. Am. Chem. Soc. |
1984 |
Link |
|
10 |
K.A. Brown-Wensley; S.L. Buchwald; L. Cannizzo; L. Clawson; H. S.; D. Meinhardt; J.R. Stille; D. Straus; R.H. Grubbs |
CP2TiCH2 Complexes in Synthetic Applications |
Pure Appl. Chem. |
1983 |
Link |
|
9 |
S.L. Buchwald; R.H. Grubbs |
A titanium vinylidene route to substituted allenes |
J. Am. Chem. Soc. |
1983 |
Link |
|
8 |
K.A. Parker; J.J. Petraitis; R.W. Kosley; S.L. Buchwald |
Reactions of propargyl alcohols with amide acetals |
J. Org. Chem. |
1982 |
Link |
|
7 |
S.L. Buchwald; D.H. Pliura; J.R. Knowles |
Stereochemistry and mechanism of an acid-catalyzed 1,2-phospho group migration: evidence for pseudorotation in the reaction of a phosphoric monoester |
J. Am. Chem. Soc. |
1982 |
Link |
|
6 |
S.L. Buchwald; J.R. Knowles |
Nucleophilic displacements on phosphoric monoesters: stereochemical evidence |
J. Am. Chem. Soc. |
1982 |
Link |
|
5 |
S.L. Buchwald; D.E. Hansen; A. Hassett; J.R. Knowles |
Chiral [16O, 17O, 18O]phosphoric monoesters as stereochemical probes of phosphotransferases |
Methods Enzymol. |
1982 |
|
|
4 |
M.S. Saini; S.L. Buchwald; R.L. Van Etten; J.R. Knowles |
Stereochemistry of phospho transfer catalyzed by bovine liver acid phosphatase |
J. Biol. Chem. |
1981 |
|
|
3 |
S.L. Buchwald; J.R. Knowles |
Determination of the absolute configuration of [16O,17O,18O]phosphate monoesters by using phosphorus-31 NMR |
J. Am. Chem. Soc. |
1980 |
Link |
|
2 |
D.E. Cane; S.L. Buchwald |
Application of deuterium magnetic resonance to biosynthetic studies. 1. Biosynthesis of ovalicin |
J. Am. Chem. Soc. |
1977 |
Link |
|
1 |
K.A. Parker; R.W. Kosley; S.L. Buchwald; J.J. Petraitis |
The Reaction of Tertiary Ethynyl Alcohols with Formamide Acetals: Formation of Dienamines and Enamine Orthoformates |
J. Am. Chem. Soc. |
1976 |
Link |
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Submitted |
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