Guram, Anil S.
Rennels, Roger A.
Buchwald, Stephen L.

A Simple Catalytic Method for the Conversion of Aryl Bromides to Arylamines

“,
Angew. Chem. Int. Ed.
,
1995
,
34
(
12
)
,
1348-1350
.
Abstract

A facile Pd-catalyzed method for the preparation of a wide variety of aryl amines from aryl bromides and amines has been developed [Eq. (a)]. Noteworthy features of this method include the experimental simplicity, the tin/boron-free conditions, and the broad spectrum of potential substrates.