DeBergh, J. Robb
Niljianskul, Nootaree
Buchwald, Stephen L.

Synthesis of Aryl Sulfonamides via Palladium-Catalyzed Chlorosulfonylation of Arylboronic Acids

“,
J. Am. Chem. Soc.
,
2013
,
135
(
29
)
,
10638 – 10641
.
Abstract

A palladium-catalyzed method for the preparation of sulfonamides is described. The process exhibits significant functional group tolerance and allows for the preparation of a number of arylsulfonyl chlorides and sulfonamides under mild conditions.