SLB # Authors Title Patent Number Date Issued
49 Buchwald, Stephen L.; Pentelute, Bradley L.; Spokoyny, Alexander M.; Vinogradova, Ekaterina V.; Zhang, Chi Transition metal-based selective functionalization of chalcogens in biomolecules. WO 2016011107 A2 January 21, 2016
48 Linquist, Susan L.; Buchwald, Stephen L.; Tardiff, Daniel; Jui, Nathan Benzimidazole derivatives for treatment of diseases assocd. with protein aggregation and other diseases. WO 2014145887 A1 September 18, 2014
47 Buchwald, Stephen L.; Swager, Timothy M.; Teverovskiy, Georgiy; Su, Mingjuan Organic conductive materials including iptycene-​based structure and devices. WO 2014070888 A1 May 8, 2014
46 Vincent, Benjamin; Whitesell, Luke; Lindquist, Susan L.; Youngsaye, Willmen; Buchwald, Stephen L.; Langlois, Jean-Baptiste; Pu, Jun; Munoz, Benito; Dandapani, Sivaraman Thiohydantoin derivatives for treating a fungal or protozoan infection. WO 2014062852 A2 April 24, 2014
45 Vincent, Benjamin; Whitesell, Luke; Lindquist, Susan L.; Youngsaye, Willmen; Buchwald, Stephen L.; Langlois, Jena-Baptiste; Nag, Partha P.; Ting, Amal; Morgan, Barbara J.; Munoz, Benito Preparation of indazole derivatives as antifungal agents and uses thereof. WO 2014047662 A2 March 27, 2014
44 Bruno, Nicholas C.; Buchwald, Stephen L. Phosphine-​ligated palladium sulfonate palladacycles. WO 2013184198 A1 December 12, 2013
43 Buchwald, Stephen L.; Watson, Donald Allen; Su, Mingjuan; Teverovskiy, Georgiy Metal-​catalyzed carbon-​fluorine bond formation. WO 2011008725 A2 January 20, 2011
42 Buchwald, Stephen L.; Fors, Brett P.; Surry, David S. Ligands for transition-​metal-​catalyzed cross-​couplings, and methods of use thereof. WO2009076622 A3 June 18, 2009
41 Buchwald, S.L. and Anderson, K.W. Transition-metal-catalyzed carbon-nitrogen and carbon-carbon bond-forming reactions. U.S. Patent No. 7,560,596 July 14, 2009
40 Buchwald, S.L.; Old, D.W.; Wolfe, J.P.; Palucki, M.; Kamikawa, K. Ligands for Metals and Improved Metal-Catalyzed Processes Based Thereon. U.S. Patent No. 7,560,582 July 14, 2009
39 Hirsh, J.; Klibanov, A.M.; Swager, T.M.; Buchwald, S.L.; Lo, W.Y.; Fleming, A.B. and Rariy, R.V. Abuse-deterrent Pharmaceutical Compositions of Opiods and Other Drugs. U.S. Patent No 7,399,488 July 15, 2008
38 Buchwald, S.L.; Klapars, A.; Kwong, F.Y.; Strieter, E.R.; Zanon, Z. Copper-catalyzed Formation of Carbon-Heteroatom and Carbon-Carbon Bonds. U.S. Patent No. 7,323,608 January 29, 2008
37 Buchwald, S.L.; Old, D.W.; Wolfe, J.P.; Palucki, M.; Kamikawa, K. Ligands for Metals and Improved Metal-Catalyzed Processes Based Thereon. U.S. Patent No. 7,247,731 July 24, 2007
36 Buchwald, S. L.; Huang, X.; Zim, D. Ligands for metals and improved metal-catalyzed processes based thereon. U.S. Patent No. 7,223,879 May 29, 2007
35 Buchwald, S. L.; Klapars, A.; Antilla, J. C.; Job, G. E.; Wolter, M.; Kwong, F. Y.; Nordmann, G.; Hennessy, E. J. Copper-catalyzed Formation of Carbon-heteroatom and Carbon-carbon bonds. U.S. Patent No. 7,115,784 October 3, 2006
34 Buchwald, S.L.; Plante, O.J.; Seeberger, P.H. Protecting Groups Useful in the Synthesis of Polysaccharides, Natural Products, and Combinatorial Libraries U.S. Patent No. 7,102,023 September 5, 2006
33 Rariy, R.V.; Heffernen, H.; Buchwald, S.L.; Swager, T.M. Stereoisomers of p-hydroxy-milnacipran, and Methods of Use Thereof U.S. Patent No. 7,038,085 May 2, 2006
32 Buchwald, S.L.; Old, D.W.; Wolfe, J.P.; Palucki, M.; Kamikawa, K. Ligands for Metals and Improved Metal-catalyzed Processes Based Thereon. U.S. Patent No. 7,026,498 April 11, 2006
31 Buchwald, S.L.; Old, D.W.; Wolfe, J.P.; Palucki, M.; Kamikawa, K. Ligands for Metals and Improved Metal-catalyzed Processes Based Thereon. U.S. Patent No. 6,946,560 September 20, 2005
30 Buchwald, S.L.; Klapars, A.; Kwong, F.Y.; Steiter, E.R.; Zanon, J. Copper-catalyzed Formation of Carbon-heteroatom and Carbon-carbon Bonds. U.S. Patent No. 6,888,032 May 3, 2005
29 Buchwald, S.L.; Fox, J.M. Transition-metal-catalyzed cabon-nitrogen bond-forming methods using carbene ligands. U.S. Patent No. 6,888,029 May 3, 2005
28 Buchwald, S.L.; Wolfe, J.P.; Ahman, J.; Troutman, M.; Palucki, M.; Kamikawa, K.; Chieffi, A. Arylation and vinylation of activated carbons. U.S. Patent No. 6,867,310 March 15, 2005
27 Buchwald, S.L.; Klapars, A.; Antilla, J.C.; Job, Gabriel E.; Wolter, M.; Kwong, Fuk Y.; Nordmann, G.; Hennessy, E. J. Copper-catalyzed Formation of Carbon-heteroatom and Carbon-carbon bonds. U.S. Patent No. 6,867,298 March 15, 2005
26 Buchwald, S.L.; Appella, D.H.; Moritani, Y.; Shintani, R.; Jurkauskas, V. Asymmetric 1,4-reductions of and 1,4-additions to Enolates and Related Systems. U.S. Patent No. 6,787,655 September 7, 2004
25 Marcoux, J.-F.; Doye, S.; Buchwald, S.L. Diaryl Ether Condensation Reactions. U.S. Patent No. 6,762,329 July 13, 2004
24 Buchwald, S.L.; Klapars, A; Antilla, J.C.; Job, G.E.; Wolter, M.; Kwong, F.Y.; Nordmann, G.; Hennessy, E.J. Copper-Catalyzed Formation of Carbon-Heteroatom and Carbon-Carbon Bonds. U.S. Patent No. 6,759,554 July 6, 2004
23 Buchwald, S.L.; Plante, O.J.; Seeberger, P.H. Protecting Groups Useful in the Synthesis of Polysaccharides, Natural products and Combinatorial Libraries. U.S. Patent No. 6,693,178 February, 17, 2004
22 Buchwald, S.L.; Appella, D.H.; Moritani, Y.; Shintani, R.; Jurkauskas, V. Asymmetric 1,4-reductions of and 1,4-additions to Enolates and Related Systems. U.S. Patent No. 6,465,664 October 15, 2002
21 Buchwald, S.L.; Wagaq, S.; Geis, O. Metal-Catalyzed Arylations of Hydrazines, Hydrazones, and Related Substrates. U.S. Patent No. 6,465,693 October 15, 2002
20 Buchwald, S.L.; Plante, O.J.; Seeberger, P.H. Protecting Groups Useful In The Synthesis of Polysaccharides, Natural Products, And Combinatorial Libraries. U.S. Patent No. 6,426,451B1 July 30, 2002
19 Marcoux, J.-F.; Doye, S.; Buchwald, S.L. Diaryl Ether Condensation Reactions. U.S. Patent No. 6, 395,939 May 28, 2002
18 Buchwald, S.L.; Wolfe, J.P.; Old, D.W.; Kamikawa, K.; Palucki, M. Ligands for Metals and Improved Metal-Catalyzed Processes BasedThereon. U.S. Patent No. 6,395,916 May 28, 2002
17 Wolfe, J.P.; Ahman, J.; Sadighi; J.P.; Singer, R.A.; Buchwald, S.L. Arylamine Synthesis. U.S. Patent No. 6,323,366 November 27, 2001
16 Buchwald, S.L.; Old, D.W.; Wolfe, J.P.; Palucki, M.; Kamikawa, K. Ligands for Metals and Improved Metal-Catalyzed Processes Based Thereon. U.S. Patent No. 6,307,087 October 23, 2001
15 Buchwald, S.L.; Singer, R.A.; Sadighi, J.P. Synthesis of Oligoarylamines, and Uses and Reagents Related Thereto. U.S. Patent No. 6,235,871 May 22, 2001
14 Buchwald, S.L.; Wagaw, S.; Geis, O. Metal-Catalyzed Arylations of Hydrazines, Hydrazones, and Related Substrates. U.S. Patent No. 6,235,935 May 22, 2001
13 Molnar, L.K.; Hatton, T.A.; Buchwald, S.L. Replacement Solvents for Use in Chemical Synthesis. U.S. Patent No. 6,231,783 May 15, 2001
12 Buchwald, S.L.; Wolfe, J.P.; Palucki, M Synthesis of Aryl Ethers. U.S. Patent No. 6,166,226 December 26, 2000
11 Verdaguer, X., Lange, U.E.W., Buchwald, S.L. Imine Hydrosilylation, Uses and Reagents Related Thereto. U.S. Patent No. 6,072,085 June 6, 2000
10 Buchwald, S.L.; Wolfe, J.P.; Palucki, M. Synthesis of Aryl Ethers. U.S. Patent No. 5,847,166 December 8, 1998
9 Buchwald, S.L.; Guram, A.S. Preparation of Arylamines. U.S. Patent No. 5,576,460 November 19, 1996
8 Buchwald, S.L.; Broene, R.D. Catalytic Asymmetric Reduction of Trisubstituted Olefins. U.S. Patent No. 5,491,233 February 13, 1996
7 Buchwald, S.L.; Lee, N.E. Catalytic Asymmetric Reduction of Enamines. U.S. Patent No. 5,489,682 February 6, 1996
6 Buchwald, S.L.; Broene, R.D. Catalytic Asymmetric Reduction of Trisubstituted Olefins. U.S. Patent No. 5,442,119 August 15, 1995
5 Buchwald, S.L.; Willoughby, C.A. Catalytic Asymmetric and Non-Asymmetric Reduction of Imines and Oximes Using Metal Catalysts. U.S. Patent No. 5,292,893 March 8, 1994
4 Buchwald, S.L.; Kreutzer, K.A.; Spaltenstein, E. Catalytic Reduction of Organic Carbonyls. U.S. Patent No. 5,286,878 February 15, 1994
3 Buchwald, S.L.; Gutiérrez, A.; Grossman, R.B. Catalytic Asymmetric Reduction of Ketones Using Metal Catalysts. U.S. Patent No. 5,227,538 July 13, 1993
2 Buchwald, S.L.; Gutiérrez, A.; Berk, S.C.; Kreutzer, K.A. Catalytic Reduction of Organic Carbonyls Using Metal Catalysts. U.S. Patent No. 5,220,020 June 15, 1993
1 Buchwald, S.L.; Grossman, R.B. Preparation of Chiral Metallocene Dihalides. U.S. Patent No. 5,004,820 April 2, 1991