2015

Versatile Enantioselective Synthesis of Functionalized Lactones via Copper-Catalyzed Radical Oxyfunctionalization of Alkenes

R. Zhu and Buchwald, S. L. “Versatile Enantioselective Synthesis of Functionalized Lactones via Copper-Catalyzed Radical Oxyfunctionalization of Alkenes”, J. Am. Chem. Soc., 2015, 137(25), 8069 - 8077.

Catalytic Asymmetric Hydroamination of Unactivated Internal Olefins to Aliphatic Amines

Y. Yang, Shi, S. - L. , Niu, D. , Liu, P. , and Buchwald, S. L. “Catalytic Asymmetric Hydroamination of Unactivated Internal Olefins to Aliphatic Amines”, Science, 2015, 349(6243), 62 - 66.

Palladium-Catalyzed Intramolecular C-H Difluoroalkylation: Synthesis of Substituted 3,3-Difluoro-2-oxindoles

S. L. Shi and Buchwald, S. L. “Palladium-Catalyzed Intramolecular C-H Difluoroalkylation: Synthesis of Substituted 3,3-Difluoro-2-oxindoles”, Angew. Chem. Int. Ed., 2015, 54, 1646-1650.

Rational Ligand Design for the Arylation of Hindered Primary Amines Guided by Reaction Progress Kinetic Analysis

P. Ruiz-Castillo, Blackmond, D. G. , and Buchwald, S. L. “Rational Ligand Design for the Arylation of Hindered Primary Amines Guided by Reaction Progress Kinetic Analysis”, J. Am. Chem. Soc., 2015, 137, 3085-3092.

Highly Diastereo- and Enantioselective CuH-Catalyzed Synthesis of 2,3-Disubstituted Indolines

E. Ascic and Buchwald, S. L. “Highly Diastereo- and Enantioselective CuH-Catalyzed Synthesis of 2,3-Disubstituted Indolines”, J. Am. Chem. Soc., 2015, 137(14), 4666 - 4669.

Virtually Instantaneous, Room-Temperature [11C]-Cyanation Using Biaryl Phosphine Pd(0) Complexes

H. Geun Lee, Milner, P. J. , Placzek, M. S. , Buchwald, S. L. , and Hooker, J. M. “Virtually Instantaneous, Room-Temperature [11C]-Cyanation Using Biaryl Phosphine Pd(0) Complexes”, J. Am. Chem. Soc., 2015, 137, 648-651.

Mild Palladium-Catalyzed Cyanation of (Hetero)aryl Halides and Triflates in Aqueous Media

D. T. Cohen and Buchwald, S. L. “Mild Palladium-Catalyzed Cyanation of (Hetero)aryl Halides and Triflates in Aqueous Media”, Org. Lett., 2015, 17(2), 202 - 205.

Copper-catalysed Selective Hydroamination Reactions of Alkynes

S. - L. Shi and Buchwald, S. L. “Copper-catalysed Selective Hydroamination Reactions of Alkynes”, Nat. Chem., 2015, 7(1), 38 - 44.

Tim Senter

Stefan Roesner

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