2008

An Improved Protocol for the Pd-Catalyzed α-Arylation of Aldehydes with Aryl Halides

R. Martín and Buchwald, S. L. “An Improved Protocol for the Pd-Catalyzed α-Arylation of Aldehydes with Aryl Halides”, Org. Lett., 2008, 10(20), 4561-4564.

Palladium-Catalyzed Suzuki−Miyaura Cross-Coupling Reactions Employing Dialkylbiaryl Phosphine Ligands

R. Martín and Buchwald, S. L. “Palladium-Catalyzed Suzuki−Miyaura Cross-Coupling Reactions Employing Dialkylbiaryl Phosphine Ligands”, Acc. Chem. Res., 2008, 41(11), 1461-1473.

Palladium-Catalyzed γ-Arylation of β,γ-Unsaturated Ketones: Application to a One-Pot Synthesis of Tricyclic Indolines

A. M. Hyde and Buchwald, S. L. “Palladium-Catalyzed γ-Arylation of β,γ-Unsaturated Ketones: Application to a One-Pot Synthesis of Tricyclic Indolines”, Angew. Chem. Int. Ed., 2008, 47(1), 177-180.

Asymmetric Palladium-Catalyzed Intramolecular α-Arylation of Aldehydes

J. García-Fortanet and Buchwald, S. L. “Asymmetric Palladium-Catalyzed Intramolecular α-Arylation of Aldehydes”, Angew. Chem. Int. Ed., 2008, 47(42), 8108-8111.

A Highly Active Catalyst for Pd-Catalyzed Amination Reactions: Cross-Coupling Reactions Using Aryl Mesylates and the Highly Selective Monoarylation of Primary Amines Using Aryl Chlorides

B. P. Fors, Watson, D. A. , Biscoe, M. R. , and Buchwald, S. L. “A Highly Active Catalyst for Pd-Catalyzed Amination Reactions: Cross-Coupling Reactions Using Aryl Mesylates and the Highly Selective Monoarylation of Primary Amines Using Aryl Chlorides”, J. Am. Chem. Soc., 2008, 130(41), 13552-13554.

Water-Mediated Catalyst Preactivation: An Efficient Protocol for C−N Cross-Coupling Reactions

B. P. Fors, Krattiger, P. , Strieter, E. , and Buchwald, S. L. “Water-Mediated Catalyst Preactivation: An Efficient Protocol for C−N Cross-Coupling Reactions”, Org. Lett., 2008, 10(16), 3505-3508.

Twofold C−H Functionalization: Palladium-Catalyzed Ortho Arylation of Anilides

G. Brasche, García-Fortanet, J. , and Buchwald, S. L. “Twofold C−H Functionalization: Palladium-Catalyzed Ortho Arylation of Anilides”, Org. Lett., 2008, 10(11), 2207-2210.

C–H Functionalization/C–N Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines

G. Brasche and Buchwald, S. L. “C–H Functionalization/C–N Bond Formation: Copper-Catalyzed Synthesis of Benzimidazoles from Amidines”, Angew. Chem. Int. Ed., 2008, 47(10), 1932-1934.

A New Class of Easily Activated Palladium Precatalysts for Facile C−N Cross-Coupling Reactions and the Low Temperature Oxidative Addition of Aryl Chlorides

M. R. Biscoe, Fors, B. P. , and Buchwald, S. L. “A New Class of Easily Activated Palladium Precatalysts for Facile C−N Cross-Coupling Reactions and the Low Temperature Oxidative Addition of Aryl Chlorides”, J. Am. Chem. Soc., 2008, 130(21), 6686-6687.

A General and Efficient Method for the Suzuki–Miyaura Coupling of 2-Pyridyl Nucleophiles

K. L. Billingsley and Buchwald, S. L. “A General and Efficient Method for the Suzuki–Miyaura Coupling of 2-Pyridyl Nucleophiles”, Angew. Chem. Int. Ed., 2008, 47(25), 4695-4698.

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