Site-Specific Antibody Prodrugs via S‑Arylation: a Bioconjugation Approach Toward Masked Tyrosine Analogues |
Tao, J. ; Dhanjee, H. H. ; Gribble, Jr., M. W. ; Kottisch, V. ; Rodriguez, J. ; Brown, J. S. ; Schmidt, H. ; Juneja, J. ; Denhez, F. ; Lee, P. S. ; Lipovšek, D. ; Krystek, S. ; Zhang, Y. ; Bousquet, P. ; Zhang, Y. ; Petelute, B. L. ; Buchwald, S. L. . J. Am. Chem. Soc. 2024, 146, 20080-20085. |
Palladium-Mediated Incorporation of Carboranes into Small Molecules, Peptides, and Proteins |
Gazvoda, M. ; Dhanjee, H. H. ; Rodriguez, J. ; Brown, J. S. ; Farquhar, C. E. ; Truex, N. L. ; Loas, A. ; Buchwald, S. L. ; Pentelute, B. L. . J. Am. Chem. Soc. 2022, 144, 7852-7860. |
Palladium Mediated Synthesis of Protein–Polyarene Conjugates |
Rodriguez, J. ; Dhanjee, H. H. ; Pentelute, B. L. ; Buchwald, S. L. . J. Am. Chem. Soc. 2022, 144, 11706-11712. |
Amphiphilic Biaryl Monophosphine Ligands by Regioselective Sulfonation |
Rodriguez, J. ; Dhanjee, H. H. ; Buchwald, S. L. . Org. Lett. 2021, 23, 777-780. |
Oligonucleotide Bioconjugation with Bifunctional Palladium Reagents |
Jbara, M. ; Rodriguez, J. ; Dhanjee, H. H. ; Loas, A. ; Buchwald, S. L. ; Pentelute, B. L. . Angew. Chem., Int. Ed. 2021, 60, 12109-12115. |
Engineering Bioactive Dimeric Transcription Factor Analogs via Palladium Rebound Reagents |
Jbara, M. ; Pomplun, S. ; Schissel, C. K. ; Hawken, S. Wilson; Boija, A. ; Klein, I. ; Rodriguez, J. ; Buchwald, S. L. ; Pentelute, B. L. . J. Am. Chem. Soc. 2021, 143, 11788-11798. |